ES413937A1 - Un procedimiento para preparar 6 - (2 - aril - 2 - 3 (3- guanil - 1 - ureidoalcanoilamino) acetamido) penecilanico. - Google Patents

Un procedimiento para preparar 6 - (2 - aril - 2 - 3 (3- guanil - 1 - ureidoalcanoilamino) acetamido) penecilanico.

Info

Publication number
ES413937A1
ES413937A1 ES413937A ES413937A ES413937A1 ES 413937 A1 ES413937 A1 ES 413937A1 ES 413937 A ES413937 A ES 413937A ES 413937 A ES413937 A ES 413937A ES 413937 A1 ES413937 A1 ES 413937A1
Authority
ES
Spain
Prior art keywords
carbon atoms
formula
alpha
see formula
alkylene containing
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES413937A
Other languages
English (en)
Spanish (es)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc filed Critical Pfizer Inc
Publication of ES413937A1 publication Critical patent/ES413937A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C275/00Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
    • C07C275/04Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to acyclic carbon atoms
    • C07C275/06Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to acyclic carbon atoms of an acyclic and saturated carbon skeleton
    • C07C275/16Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to acyclic carbon atoms of an acyclic and saturated carbon skeleton being further substituted by carboxyl groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C279/00Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups
    • C07C279/28Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of guanidine groups bound to cyano groups, e.g. cyanoguanidines, dicyandiamides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C335/00Thioureas, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
    • C07C335/30Isothioureas
    • C07C335/34Isothioureas having sulfur atoms of isothiourea groups bound to carbon atoms of rings other than six-membered aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C335/00Thioureas, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
    • C07C335/30Isothioureas
    • C07C335/38Isothioureas containing any of the groups, X being a hetero atom, Y being any atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/28Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/30Oxygen or sulfur atoms
    • C07D233/42Sulfur atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/28Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/44Nitrogen atoms not forming part of a nitro radical
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/28Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/44Nitrogen atoms not forming part of a nitro radical
    • C07D233/46Nitrogen atoms not forming part of a nitro radical with only hydrogen atoms attached to said nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Cephalosporin Compounds (AREA)
ES413937A 1972-05-16 1973-04-19 Un procedimiento para preparar 6 - (2 - aril - 2 - 3 (3- guanil - 1 - ureidoalcanoilamino) acetamido) penecilanico. Expired ES413937A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US00253856A US3838153A (en) 1972-05-16 1972-05-16 6-(alpha-(guanylureidoalkanoylamino)aracylamino)penicillanic acids

Publications (1)

Publication Number Publication Date
ES413937A1 true ES413937A1 (es) 1976-06-01

Family

ID=22961983

Family Applications (1)

Application Number Title Priority Date Filing Date
ES413937A Expired ES413937A1 (es) 1972-05-16 1973-04-19 Un procedimiento para preparar 6 - (2 - aril - 2 - 3 (3- guanil - 1 - ureidoalcanoilamino) acetamido) penecilanico.

Country Status (23)

Country Link
US (1) US3838153A (US20100292554A1-20101118-C00004.png)
JP (1) JPS5533712B2 (US20100292554A1-20101118-C00004.png)
AR (1) AR195914A1 (US20100292554A1-20101118-C00004.png)
AT (1) AT325767B (US20100292554A1-20101118-C00004.png)
AU (1) AU475922B2 (US20100292554A1-20101118-C00004.png)
BE (1) BE798170A (US20100292554A1-20101118-C00004.png)
CA (1) CA1010444A (US20100292554A1-20101118-C00004.png)
CH (1) CH573434A5 (US20100292554A1-20101118-C00004.png)
DE (1) DE2318986A1 (US20100292554A1-20101118-C00004.png)
DK (1) DK137046B (US20100292554A1-20101118-C00004.png)
ES (1) ES413937A1 (US20100292554A1-20101118-C00004.png)
FI (1) FI56534C (US20100292554A1-20101118-C00004.png)
FR (1) FR2184609B1 (US20100292554A1-20101118-C00004.png)
GB (1) GB1404469A (US20100292554A1-20101118-C00004.png)
IE (1) IE37491B1 (US20100292554A1-20101118-C00004.png)
IL (1) IL41937A (US20100292554A1-20101118-C00004.png)
NL (1) NL7305355A (US20100292554A1-20101118-C00004.png)
PH (1) PH10024A (US20100292554A1-20101118-C00004.png)
PL (1) PL89245B1 (US20100292554A1-20101118-C00004.png)
SE (1) SE415976B (US20100292554A1-20101118-C00004.png)
SU (1) SU504491A3 (US20100292554A1-20101118-C00004.png)
YU (1) YU36965B (US20100292554A1-20101118-C00004.png)
ZA (1) ZA732343B (US20100292554A1-20101118-C00004.png)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1462421A (en) * 1973-12-14 1977-01-26 Pfizer 6-a-amidino-and -'midoylaminoalkanoylamino aracylamino-penicillanic acids and their preparation
US3994965A (en) * 1974-08-09 1976-11-30 Pfizer Inc. D-N-(guanylureidoacetyl)-α-aminophenyl acetic acid and D-N-(guanylureidoacetyl)-α-aminophenyl acetyl chloride
JPS5562537U (US20100292554A1-20101118-C00004.png) * 1978-10-20 1980-04-28
DE3014353A1 (de) * 1980-04-15 1982-01-21 Bayer Ag, 5090 Leverkusen Trisubstituierte cyanguanidine, verfahren zu ihrer herstellung sowie ihre verwendung als fungizide
JPS56161152A (en) * 1980-05-12 1981-12-11 Tachikawa Spring Co Manufacture of steel band with resin
AU9028298A (en) 1997-08-21 1999-03-08 Quark Biotech, Inc. Hypoxia-regulated genes
US20030104973A1 (en) * 1997-08-21 2003-06-05 Quark Biotech, Inc. Hypoxia-regulated genes
US7973156B2 (en) * 1997-08-21 2011-07-05 Quark Pharmaceuticals Inc. Hypoxia-regulated genes

Also Published As

Publication number Publication date
FR2184609B1 (US20100292554A1-20101118-C00004.png) 1976-10-22
BE798170A (fr) 1973-10-15
FI56534B (fi) 1979-10-31
AR195914A1 (es) 1973-11-15
PH10024A (en) 1976-07-13
JPS5533712B2 (US20100292554A1-20101118-C00004.png) 1980-09-02
CA1010444A (en) 1977-05-17
SU504491A3 (ru) 1976-02-25
AU475922B2 (en) 1976-09-09
SE415976B (sv) 1980-11-17
NL7305355A (US20100292554A1-20101118-C00004.png) 1973-11-20
DK137046C (US20100292554A1-20101118-C00004.png) 1978-06-12
JPS4924991A (US20100292554A1-20101118-C00004.png) 1974-03-05
IE37491B1 (en) 1977-08-03
GB1404469A (en) 1975-08-28
DK137046B (da) 1978-01-09
FR2184609A1 (US20100292554A1-20101118-C00004.png) 1973-12-28
DE2318986A1 (de) 1973-12-06
AU5428373A (en) 1974-10-10
AT325767B (de) 1975-11-10
IL41937A0 (en) 1973-06-29
YU97773A (en) 1982-06-18
ZA732343B (en) 1974-01-30
ATA341573A (de) 1975-01-15
CH573434A5 (US20100292554A1-20101118-C00004.png) 1976-03-15
IE37491L (en) 1973-11-16
PL89245B1 (US20100292554A1-20101118-C00004.png) 1976-11-30
YU36965B (en) 1984-08-31
US3838153A (en) 1974-09-24
IL41937A (en) 1976-10-31
FI56534C (fi) 1980-02-11

Similar Documents

Publication Publication Date Title
ES369005A1 (es) Procedimiento para producir compuestos de o-amino - ciclo- hexadienilalrohilenopenicilina y cefalosporinas.
ES431057A1 (es) Procedimiento para la preparacion de nuevos n-(metoximetil - furilmetil)-6, 7-benzomorfanos y -morfinanos.
ES425626A1 (es) Un procedimiento para preparar compuestos de acil-xilidida.
ES413937A1 (es) Un procedimiento para preparar 6 - (2 - aril - 2 - 3 (3- guanil - 1 - ureidoalcanoilamino) acetamido) penecilanico.
ES444804A1 (es) Procedimiento para la obtencion de derivados de tetrahidroi-soquinolina.
ES410190A1 (es) Procedimiento para la obtencion de pigmentos heterocicli- cos.
ES8507450A1 (es) Un procedimiento para la preparacion de nuevos derivados de difeniletanona.
ES411038A1 (es) Un procedimiento para la preparacion de compuestos semisin-teticos intermedios en la produccion de cefalosporinas, pe- nicilinas y antibioticos relacionados de beta-lactama.
ES404745A1 (es) Un procedimiento para preparar cefalosporinas.
GB806914A (en) Manufacture of basic ketones
ES437790A1 (es) Procedimiento para preparar composiciones farmaceuticas y veterinarias.
ES435351A1 (es) Procedimiento para preparar 1-(3-fenil-propil)-4-furoilpi- perazinas.
ES441257A1 (es) Procedimiento para preparar aminocicloles.
ES393554A1 (es) Un procedimiento para la preparacion de derivados de tia- zol.
ES335707A1 (es) Procedimiento para la preparacion de derivados de la tebaina
ES340825A1 (es) Un procedimiento para preparar 1-aminoalcohil-1-arilinde- nos.
ES414805A1 (es) Un procedimiento para preparar monoesteres de alfa-carboxi-bencilpenicilina.
ES417461A1 (es) Un procedimiento para preparar acidos 6-(alfa-(amidino-e imidoilaminoalcanoilamino) aracilamino) penicilanicos.
ES437041A1 (es) Un procedimiento para preparar derivados de 1-ftalazona.
ES451820A1 (es) Procedimiento para preparar tetrahidrobenzo (b) tienilureas y tetrahidro-7-oxobenzo (b) tienlureas.
ES423230A1 (es) Un procedimiento para la preparacion de poliarilimidazolas.
ES411184A1 (es) Procedimiento para preparar derivados de penicilinas y ce- falosporinas.
ES376034A1 (es) Procedimiento para la preparacion de nuevos compuestos qui-micos utilizables como medicamentos de accion psicotropa.
GB963050A (en) Improvements in or relating to substituted pyrimido-[4,5-d]pyrimidines
ES450586A1 (es) Procedimiento para preparar 1-azidoalquilimidazoles.