ES2509869T3 - Formulaciones farmacéuticas de estatinas transportadas utilizando el transporte mediado por portadores y uso de las mismas. - Google Patents
Formulaciones farmacéuticas de estatinas transportadas utilizando el transporte mediado por portadores y uso de las mismas. Download PDFInfo
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- ES2509869T3 ES2509869T3 ES04791793.5T ES04791793T ES2509869T3 ES 2509869 T3 ES2509869 T3 ES 2509869T3 ES 04791793 T ES04791793 T ES 04791793T ES 2509869 T3 ES2509869 T3 ES 2509869T3
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- statin
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Vascular Medicine (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Urology & Nephrology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US51677003P | 2003-11-04 | 2003-11-04 | |
| US516770P | 2003-11-04 | ||
| US967167 | 2004-10-19 | ||
| US10/967,167 US8987322B2 (en) | 2003-11-04 | 2004-10-19 | Pharmaceutical formulations for carrier-mediated transport statins and uses thereof |
| PCT/IB2004/003849 WO2005041939A1 (en) | 2003-11-04 | 2004-10-29 | Pharmaceutical formulations for carrier-mediated transport statins and uses thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2509869T3 true ES2509869T3 (es) | 2014-10-20 |
Family
ID=34556205
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES04791793.5T Expired - Lifetime ES2509869T3 (es) | 2003-11-04 | 2004-10-29 | Formulaciones farmacéuticas de estatinas transportadas utilizando el transporte mediado por portadores y uso de las mismas. |
| ES10185149.1T Expired - Lifetime ES2500924T3 (es) | 2003-11-04 | 2004-10-29 | Formulaciones farmacéuticas de estatinas transportadas utilizando el transporte mediado por portadores y uso de las mismas |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES10185149.1T Expired - Lifetime ES2500924T3 (es) | 2003-11-04 | 2004-10-29 | Formulaciones farmacéuticas de estatinas transportadas utilizando el transporte mediado por portadores y uso de las mismas |
Country Status (9)
| Country | Link |
|---|---|
| US (2) | US8987322B2 (enExample) |
| EP (2) | EP1682095B1 (enExample) |
| JP (1) | JP2007510714A (enExample) |
| AU (1) | AU2004284884A1 (enExample) |
| CA (1) | CA2543716C (enExample) |
| ES (2) | ES2509869T3 (enExample) |
| IL (1) | IL175134A0 (enExample) |
| NO (1) | NO20062432L (enExample) |
| WO (1) | WO2005041939A1 (enExample) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7658938B2 (en) | 1999-02-22 | 2010-02-09 | Merrion Reasearch III Limited | Solid oral dosage form containing an enhancer |
| CA2628666A1 (en) * | 2005-11-21 | 2007-05-24 | Teva Pharmaceutical Industries Ltd. | Atorvastatin formulation |
| AU2006329006B2 (en) * | 2005-12-20 | 2013-02-28 | Lek Pharmaceuticals D.D. | Pharmaceutical composition comprising (E)-7-[4-(4-fluorophenyl)-6-isopropyl-2-[methyl(methylsulfonyl)amino]pyrimidin-5-yl]-(3R,5S)-3,5-dihydroxyhept-6-enoic acid |
| MX2008011418A (es) * | 2006-03-06 | 2008-09-22 | Teva Pharma | Composiciones de ezetimibe. |
| US7704977B2 (en) * | 2006-04-07 | 2010-04-27 | Merrion Research Iii Limited | Solid oral dosage form containing an enhancer |
| ES2300188B1 (es) * | 2006-05-24 | 2009-05-01 | Ferrer Internacional, S.A. | Comprimido bicapa para la prevencion de los accidentes cardiovasculares. |
| JP2010529142A (ja) * | 2007-06-08 | 2010-08-26 | アドレネクス・ファーマシューティカルズ，インコーポレイテッド | アドレナリン調節異常症を治療する徐放性の製剤および方法 |
| US20090082315A1 (en) * | 2007-09-05 | 2009-03-26 | Raif Tawakol | Compositions and Methods for Controlling Cholesterol Levels |
| TR200800269A2 (tr) * | 2008-01-15 | 2009-08-21 | Bi̇li̇m İlaç Sanayi̇ Ti̇caret A.Ş. | Stabil farmasötik formülasyon ve hazırlama yöntemleri |
| TWI391150B (zh) * | 2008-01-22 | 2013-04-01 | Taiwan Biotech Co Ltd | 腸溶性長效塗覆芯與藥物劑型及其製造方法 |
| US20110003837A1 (en) * | 2008-01-30 | 2011-01-06 | Lupin Limited | Modified release formulations of hmg coa reductase inhibitors |
| JP5671451B2 (ja) | 2008-05-07 | 2015-02-18 | メリオン・リサーチ・Ｉｉｉ・リミテッド | ＧｎＲＨ関連化合物の組成物および調製プロセス |
| WO2010099255A1 (en) * | 2009-02-25 | 2010-09-02 | Merrion Research Iii Limited | Composition and drug delivery of bisphosphonates |
| US20110182985A1 (en) * | 2010-01-28 | 2011-07-28 | Coughlan David C | Solid Pharmaceutical Composition with Enhancers and Methods of Preparing thereof |
| WO2011120033A1 (en) * | 2010-03-26 | 2011-09-29 | Merrion Research Iii Limited | Pharmaceutical compositions of selective factor xa inhibitors for oral administration |
| US8802114B2 (en) | 2011-01-07 | 2014-08-12 | Merrion Research Iii Limited | Pharmaceutical compositions of iron for oral administration |
| CN107205948B (zh) | 2015-01-29 | 2021-12-14 | 诺和诺德股份有限公司 | 包含glp-1激动剂和肠溶衣的片剂 |
Family Cites Families (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3845770A (en) | 1972-06-05 | 1974-11-05 | Alza Corp | Osmatic dispensing device for releasing beneficial agent |
| US3916899A (en) | 1973-04-25 | 1975-11-04 | Alza Corp | Osmotic dispensing device with maximum and minimum sizes for the passageway |
| GB1478759A (en) | 1974-11-18 | 1977-07-06 | Alza Corp | Process for forming outlet passageways in pills using a laser |
| US4088884A (en) * | 1976-01-26 | 1978-05-09 | The United States Of America As Represented By The Secretary Of The Navy | Wide aperture optical communications detector |
| US4200098A (en) | 1978-10-23 | 1980-04-29 | Alza Corporation | Osmotic system with distribution zone for dispensing beneficial agent |
| US4557925A (en) | 1982-07-08 | 1985-12-10 | Ab Ferrosan | Membrane-coated sustained-release tablets and method |
| SE8601624D0 (sv) * | 1986-04-11 | 1986-04-11 | Haessle Ab | New pharmaceutical preparations |
| US4904474A (en) * | 1988-01-25 | 1990-02-27 | Alza Corporation | Delivery of drug to colon by oral disage form |
| EP0465096A1 (en) | 1990-06-26 | 1992-01-08 | Merck & Co. Inc. | Plasma cholesterol level lowering composition |
| US6764697B1 (en) * | 1991-06-27 | 2004-07-20 | Alza Corporation | System for delaying drug delivery up to seven hours |
| US5573776A (en) | 1992-12-02 | 1996-11-12 | Alza Corporation | Oral osmotic device with hydrogel driving member |
| US5916595A (en) * | 1997-12-12 | 1999-06-29 | Andrx Pharmaceutials, Inc. | HMG co-reductase inhibitor |
| CO5140079A1 (es) | 1998-10-14 | 2002-03-22 | Novartis Ag | Composicion farmaceutica de liberacion sostenida y metodo para liberar un agente farmaceuticamente activo de liberacion sostenida y metodo para liberar un agente far- maceuticamente activo |
| US6248363B1 (en) * | 1999-11-23 | 2001-06-19 | Lipocine, Inc. | Solid carriers for improved delivery of active ingredients in pharmaceutical compositions |
| US6569461B1 (en) * | 1999-03-08 | 2003-05-27 | Merck & Co., Inc. | Dihydroxy open-acid and salts of HMG-CoA reductase inhibitors |
| AU2866400A (en) | 1999-03-08 | 2000-09-28 | Merck & Co., Inc. | Dihydroxy open-acid and salts of hmg-co-a reductase inhibitors |
| SI20425A (sl) * | 1999-12-10 | 2001-06-30 | LEK tovarna farmacevtskih in kemi�nih izdelkov d.d. | Priprava amorfnega atorvastatina |
| AU2001253401B2 (en) * | 2000-04-11 | 2006-12-07 | Atherogenics, Inc | Compounds and methods to increase plasma hdl cholesterol levels and improve hdl functionality |
| US20020147232A1 (en) * | 2000-05-26 | 2002-10-10 | Claus Sundgreen | Pharmaceutical compositions comprising desglymidodrine as an active drug substance |
| IL156552A0 (en) * | 2000-12-21 | 2004-01-04 | Aventis Pharma Gmbh | Diphenyl azetidinone derivatives, method for the production thereof, medicaments containing these compounds, and their use |
| FR2834212B1 (fr) * | 2001-12-27 | 2004-07-09 | Besins Int Belgique | Utilisation d'une poudre a liberation immediate dans des compositions pharmaceutiques et nutraceutiques |
| EP1465605A1 (en) | 2002-01-11 | 2004-10-13 | Athpharma Limited | Pravastatin pharmaceutical formulations and methods of their use |
| MXPA05002074A (es) | 2002-09-03 | 2005-06-08 | Biovail Lab Int Srl | Formulaciones farmaceuticas y metodos para la liberacion modificada de farmacos de estatina. |
| PL375712A1 (en) | 2002-09-03 | 2005-12-12 | Biovail Laboratories Inc. | Pravastatin pharmaceutical formulations and methods of their use |
-
2004
- 2004-10-19 US US10/967,167 patent/US8987322B2/en not_active Expired - Fee Related
- 2004-10-29 EP EP04791793.5A patent/EP1682095B1/en not_active Expired - Lifetime
- 2004-10-29 JP JP2006538993A patent/JP2007510714A/ja active Pending
- 2004-10-29 EP EP10185149.1A patent/EP2319501B1/en not_active Expired - Lifetime
- 2004-10-29 WO PCT/IB2004/003849 patent/WO2005041939A1/en not_active Ceased
- 2004-10-29 AU AU2004284884A patent/AU2004284884A1/en not_active Abandoned
- 2004-10-29 ES ES04791793.5T patent/ES2509869T3/es not_active Expired - Lifetime
- 2004-10-29 ES ES10185149.1T patent/ES2500924T3/es not_active Expired - Lifetime
- 2004-10-29 CA CA2543716A patent/CA2543716C/en not_active Expired - Fee Related
-
2006
- 2006-04-24 IL IL175134A patent/IL175134A0/en unknown
- 2006-05-29 NO NO20062432A patent/NO20062432L/no not_active Application Discontinuation
-
2015
- 2015-02-23 US US14/629,232 patent/US20150164893A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| CA2543716C (en) | 2016-05-31 |
| US20050119331A1 (en) | 2005-06-02 |
| ES2500924T3 (es) | 2014-10-01 |
| EP1682095B1 (en) | 2014-07-02 |
| WO2005041939A1 (en) | 2005-05-12 |
| EP2319501A1 (en) | 2011-05-11 |
| IL175134A0 (en) | 2006-09-05 |
| CA2543716A1 (en) | 2005-05-12 |
| NO20062432L (no) | 2006-08-04 |
| JP2007510714A (ja) | 2007-04-26 |
| US20150164893A1 (en) | 2015-06-18 |
| US8987322B2 (en) | 2015-03-24 |
| AU2004284884A1 (en) | 2005-05-12 |
| EP2319501B1 (en) | 2014-06-18 |
| EP1682095A1 (en) | 2006-07-26 |
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