ES2174863T3 - PIRIMIDINE COMPOUNDS AND ITS USE AS PHARMACEUTICAL COMPOUNDS. - Google Patents

PIRIMIDINE COMPOUNDS AND ITS USE AS PHARMACEUTICAL COMPOUNDS.

Info

Publication number
ES2174863T3
ES2174863T3 ES94304104T ES94304104T ES2174863T3 ES 2174863 T3 ES2174863 T3 ES 2174863T3 ES 94304104 T ES94304104 T ES 94304104T ES 94304104 T ES94304104 T ES 94304104T ES 2174863 T3 ES2174863 T3 ES 2174863T3
Authority
ES
Spain
Prior art keywords
compounds
formula
pirimidine
pharmaceutical
pyramidine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES94304104T
Other languages
Spanish (es)
Inventor
Gerd Ruhter
Theo Schotten
Wolfgang Stenzel
Michael Paal
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Beiersdorf Lilly GmbH
Original Assignee
Beiersdorf Lilly GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Beiersdorf Lilly GmbH filed Critical Beiersdorf Lilly GmbH
Application granted granted Critical
Publication of ES2174863T3 publication Critical patent/ES2174863T3/en
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Abstract

SE PRESENTAN COMPUESTOS FARMACEUTICOS QUE SON COMPUESTOS DE PIRIMIDINA FUNDIDA EN AZOLO QUE TIENEN LA FORMULA I EN LA CUAL A-B JUNTO CON EL ANILLO DE PIRIMIDINA FORMA (A) UNA PIRAZOLO [1,5A]PIRAMIDINA DE LA FORMULA (A), (B) UNA [1,2,4]TRIAZOLO[1,5A]PIRIMIDINA DE LA FORMULA (B); (C) UNA IMIDAZO[1,5-A]PIRAMIDINA DE LA FORMULA (C); O (D) UNA IMIDAZO[1,2-A]PIRAMIDINA DE LA FORMULA (D).PHARMACEUTICAL COMPOUNDS ARE PRESENTED WHICH ARE PIRIMIDINE COMPOUNDS FOUNDED IN AZOLO THAT HAVE FORMULA I IN WHICH AB NEXT TO THE PYRIMIDINE RING SHAPE (A) A PIRAZOLO [1,5A] PYRAMIDINE OF FORMULA (A), (B) ONE [1,2,4] TRIAZOL [1,5A] PYRIMIDINE OF THE FORMULA (B); (C) AN IMIDAZO [1,5-A] FORMULA PYRAMIDINE (C); OR (D) AN IMIDAZO [1,2-A] FORMULA PYRAMIDINE (D).

ES94304104T 1993-06-10 1994-06-07 PIRIMIDINE COMPOUNDS AND ITS USE AS PHARMACEUTICAL COMPOUNDS. Expired - Lifetime ES2174863T3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP93304513 1993-06-10

Publications (1)

Publication Number Publication Date
ES2174863T3 true ES2174863T3 (en) 2002-11-16

Family

ID=8214429

Family Applications (1)

Application Number Title Priority Date Filing Date
ES94304104T Expired - Lifetime ES2174863T3 (en) 1993-06-10 1994-06-07 PIRIMIDINE COMPOUNDS AND ITS USE AS PHARMACEUTICAL COMPOUNDS.

Country Status (5)

Country Link
US (3) US5571813A (en)
JP (1) JPH072860A (en)
CA (1) CA2125458A1 (en)
DE (1) DE69430279T2 (en)
ES (1) ES2174863T3 (en)

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Also Published As

Publication number Publication date
JPH072860A (en) 1995-01-06
CA2125458A1 (en) 1994-12-11
US5602137A (en) 1997-02-11
DE69430279T2 (en) 2003-03-06
US5571813A (en) 1996-11-05
DE69430279D1 (en) 2002-05-08
US5602136A (en) 1997-02-11

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