ES2131219T3 - Solvatos estables de compuestos de avermectina. - Google Patents
Solvatos estables de compuestos de avermectina.Info
- Publication number
- ES2131219T3 ES2131219T3 ES94931307T ES94931307T ES2131219T3 ES 2131219 T3 ES2131219 T3 ES 2131219T3 ES 94931307 T ES94931307 T ES 94931307T ES 94931307 T ES94931307 T ES 94931307T ES 2131219 T3 ES2131219 T3 ES 2131219T3
- Authority
- ES
- Spain
- Prior art keywords
- avermectin compounds
- avermectin
- compounds
- disclosed
- solvates
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
- C07D493/22—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains four or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/14—Ectoparasiticides, e.g. scabicides
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Tropical Medicine & Parasitology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Saccharide Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- External Artificial Organs (AREA)
- Polysaccharides And Polysaccharide Derivatives (AREA)
- Separation Of Suspended Particles By Flocculating Agents (AREA)
Abstract
SE PRESENTA UNA NUEVA FORMA DE COMPUESTOS DE AVERMECTINA EN LA QUE LOS COMPUESTOS DE AVERMECTINA SE CRISTALIZAN COMO SOLVATOS DE ALCOHOL PARA MEJORAR GRATAMENTE LA ESTABILIDAD DE LA DROGA DE AVERMECTINA DURANTE SU ALMACENAMIENTO A LARGO PLAZO. LOS COMPUESTOS DE AVERMECTINA TIENEN UTILIDAD COMO AGENTES ANTIPARASITICOS, INSECTICIDAS Y ANTIHELMINTICOS ALTAMENTE POTENTES Y TAMBIEN SE PRESENTAN COMPOSICIONES PARA ESTOS USOS.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US08/133,494 US5380838A (en) | 1993-10-08 | 1993-10-08 | Stable solvates of avermectin compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
ES2131219T3 true ES2131219T3 (es) | 1999-07-16 |
Family
ID=22458871
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES94931307T Expired - Lifetime ES2131219T3 (es) | 1993-10-08 | 1994-10-04 | Solvatos estables de compuestos de avermectina. |
Country Status (10)
Country | Link |
---|---|
US (1) | US5380838A (es) |
EP (1) | EP0722454B1 (es) |
JP (1) | JP2938974B2 (es) |
AT (1) | ATE179985T1 (es) |
AU (1) | AU681916B2 (es) |
CA (1) | CA2171871C (es) |
DE (1) | DE69418469T2 (es) |
ES (1) | ES2131219T3 (es) |
WO (1) | WO1995010525A1 (es) |
ZA (1) | ZA947863B (es) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9716567D0 (en) * | 1997-08-05 | 1997-10-08 | Pfizer | Process |
EP1043324B1 (en) | 1997-11-12 | 2004-06-16 | Mitsubishi Chemical Corporation | Purine derivatives and medicine containing the same as the active ingredient |
KR100747106B1 (ko) | 1999-05-11 | 2007-08-08 | 미쯔비시 가가꾸 가부시끼가이샤 | 퓨린 유도체 이수화물, 이를 유효성분으로 함유하는 의약및 이의 제조 중간체 |
WO2004063147A1 (en) * | 2003-01-10 | 2004-07-29 | Novo Nordisk A/S | Salts and solvates of glucagon antagonists |
Family Cites Families (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SE434277B (sv) * | 1976-04-19 | 1984-07-16 | Merck & Co Inc | Sett att framstella nya antihelmintiskt verkande foreningar genom odling av streptomyces avermitilis |
PH15982A (en) * | 1977-10-03 | 1983-05-18 | Merck & Co Inc | Selective hydrogenation producta of c-076 compounds and derivatives thereof |
US4199569A (en) * | 1977-10-03 | 1980-04-22 | Merck & Co., Inc. | Selective hydrogenation products of C-076 compounds and derivatives thereof |
NZ188459A (en) * | 1977-10-03 | 1982-09-07 | Merck & Co Inc | Derivatives of c-076 compounds and pesticidal compositions |
US4206205A (en) * | 1977-10-03 | 1980-06-03 | Merck & Co., Inc. | Monosaccharide and aglycone derivatives of C-076 |
US4171314A (en) * | 1977-12-19 | 1979-10-16 | Merck & Co., Inc. | 13-Halo and 13-deoxy C-076 compounds |
US4734375A (en) * | 1980-05-27 | 1988-03-29 | Miles Laboratories, Inc. | Ion specific test method |
US4457920A (en) * | 1981-09-03 | 1984-07-03 | Merck & Co., Inc. | 4a-Substituted avermectin compounds |
US4657854A (en) * | 1983-05-05 | 1987-04-14 | Ivan Endre Modrovich | Assay systems based on magnesium-responsive enzymes |
ATE51003T1 (de) * | 1985-09-13 | 1990-03-15 | Biotechnolog Forschung Gmbh | Makrozyklische antibiotika. |
US4812400A (en) * | 1986-07-14 | 1989-03-14 | Steinman Gary D | Process for measuring sodium levels in biological fluids |
JPH0612999B2 (ja) * | 1986-11-17 | 1994-02-23 | 関東化学株式会社 | 塩素イオン定量用試薬 |
-
1993
- 1993-10-08 US US08/133,494 patent/US5380838A/en not_active Expired - Lifetime
-
1994
- 1994-10-04 AT AT94931307T patent/ATE179985T1/de not_active IP Right Cessation
- 1994-10-04 CA CA002171871A patent/CA2171871C/en not_active Expired - Lifetime
- 1994-10-04 AU AU80130/94A patent/AU681916B2/en not_active Expired
- 1994-10-04 EP EP94931307A patent/EP0722454B1/en not_active Expired - Lifetime
- 1994-10-04 ES ES94931307T patent/ES2131219T3/es not_active Expired - Lifetime
- 1994-10-04 DE DE69418469T patent/DE69418469T2/de not_active Expired - Lifetime
- 1994-10-04 JP JP7511881A patent/JP2938974B2/ja not_active Expired - Lifetime
- 1994-10-04 WO PCT/US1994/011247 patent/WO1995010525A1/en active IP Right Grant
- 1994-10-07 ZA ZA947863A patent/ZA947863B/xx unknown
Also Published As
Publication number | Publication date |
---|---|
AU8013094A (en) | 1995-05-04 |
ZA947863B (en) | 1995-05-22 |
ATE179985T1 (de) | 1999-05-15 |
CA2171871A1 (en) | 1995-04-20 |
CA2171871C (en) | 1999-08-03 |
EP0722454B1 (en) | 1999-05-12 |
US5380838A (en) | 1995-01-10 |
JP2938974B2 (ja) | 1999-08-25 |
DE69418469T2 (de) | 1999-12-16 |
WO1995010525A1 (en) | 1995-04-20 |
AU681916B2 (en) | 1997-09-11 |
JPH09503521A (ja) | 1997-04-08 |
DE69418469D1 (de) | 1999-06-17 |
EP0722454A1 (en) | 1996-07-24 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FG2A | Definitive protection |
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