ES2120185T3 - Procedimiento para preparar (1h-tetrazol-5-il)tetrazolo(1,5-a)quinolinas y naftiridinas. - Google Patents

Procedimiento para preparar (1h-tetrazol-5-il)tetrazolo(1,5-a)quinolinas y naftiridinas.

Info

Publication number
ES2120185T3
ES2120185T3 ES95910282T ES95910282T ES2120185T3 ES 2120185 T3 ES2120185 T3 ES 2120185T3 ES 95910282 T ES95910282 T ES 95910282T ES 95910282 T ES95910282 T ES 95910282T ES 2120185 T3 ES2120185 T3 ES 2120185T3
Authority
ES
Spain
Prior art keywords
tetrazole
naphtiridines
quinolins
preparing
procedure
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES95910282T
Other languages
English (en)
Inventor
Kay K Olmstead
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Aventis Pharmaceuticals Inc
Original Assignee
Merrell Dow Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merrell Dow Pharmaceuticals Inc filed Critical Merrell Dow Pharmaceuticals Inc
Application granted granted Critical
Publication of ES2120185T3 publication Critical patent/ES2120185T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Paper (AREA)
  • Luminescent Compositions (AREA)

Abstract

UN PROCESO DE ACUERDO AL ESQUEMA DE REACCION (I), EN DONDE N ES 0, 1 O 2, R ES ALQUILO C{SUB,1-4}, ALCOXI C{SUB,1-4}, HALOGENO, METILMERCAPTO, METILSULFONILO, O DOS R`S PUEDEN ESTAR COMBINADOS COMO METILENDIOXI; B ES NITROGENO O CH; Y X ES UN GRUPO SALIENTE ADECUADO; M ES UN CATION DE UN METAL ALCALINO BAJO, CON LA CONDICION DE QUE CUANDO R SEA METILMERCAPTO O METILSULFONILO, ENTONCES N DEBE SER 1.
ES95910282T 1994-03-25 1995-02-16 Procedimiento para preparar (1h-tetrazol-5-il)tetrazolo(1,5-a)quinolinas y naftiridinas. Expired - Lifetime ES2120185T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US21828094A 1994-03-25 1994-03-25

Publications (1)

Publication Number Publication Date
ES2120185T3 true ES2120185T3 (es) 1998-10-16

Family

ID=22814477

Family Applications (1)

Application Number Title Priority Date Filing Date
ES95910282T Expired - Lifetime ES2120185T3 (es) 1994-03-25 1995-02-16 Procedimiento para preparar (1h-tetrazol-5-il)tetrazolo(1,5-a)quinolinas y naftiridinas.

Country Status (18)

Country Link
EP (1) EP0751945B1 (es)
JP (1) JPH09510968A (es)
KR (1) KR970702278A (es)
CN (1) CN1043644C (es)
AT (1) ATE167863T1 (es)
AU (1) AU686761B2 (es)
CA (1) CA2184694A1 (es)
DE (1) DE69503229T2 (es)
DK (1) DK0751945T3 (es)
ES (1) ES2120185T3 (es)
FI (1) FI963808L (es)
GR (1) GR3027563T3 (es)
HU (1) HUP9774612A2 (es)
IL (1) IL113075A0 (es)
NO (1) NO964009L (es)
NZ (1) NZ281496A (es)
WO (1) WO1995026348A1 (es)
ZA (1) ZA952287B (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH08325248A (ja) * 1995-05-26 1996-12-10 Chugoku Kayaku Kk テトラゾール類の新規な合成試薬及びそれを用いたテトラゾール類の製造方法
GB0316546D0 (en) 2003-07-15 2003-08-20 Novartis Ag Process for the manufacture of organic compounds
JP2007506788A (ja) * 2003-09-26 2007-03-22 ライジェル ファーマシューティカルズ, インコーポレイテッド Hcv感染阻害剤とその使用法
WO2005121138A2 (en) * 2004-06-03 2005-12-22 Rigel Pharmaceuticals, Inc. Heterotricyclic compounds for use as hcv inhibitors

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3764681A (en) * 1970-07-08 1973-10-09 Lilly Co Eli Certain tetrazolo-(1,5-a) quinoline compounds as fungus control agents
US4496569A (en) * 1983-03-25 1985-01-29 The Dow Chemical Company Antiallergic (1H-tetrazol-5-yl)tetrazolo[1,5-a]quinolines and derivatives thereof
US4581455A (en) * 1984-10-10 1986-04-08 Merrell Dow Pharmaceuticals Inc. Tetrazolothienopyridines

Also Published As

Publication number Publication date
ATE167863T1 (de) 1998-07-15
DE69503229T2 (de) 1998-12-24
CN1043644C (zh) 1999-06-16
WO1995026348A1 (en) 1995-10-05
DE69503229D1 (de) 1998-08-06
IL113075A0 (en) 1995-06-29
EP0751945B1 (en) 1998-07-01
CN1144527A (zh) 1997-03-05
NZ281496A (en) 1998-02-26
AU686761B2 (en) 1998-02-12
ZA952287B (en) 1996-01-09
HUP9774612A2 (en) 1997-01-28
KR970702278A (ko) 1997-05-13
AU1845495A (en) 1995-10-17
FI963808A0 (fi) 1996-09-24
GR3027563T3 (en) 1998-11-30
CA2184694A1 (en) 1995-10-05
NO964009D0 (no) 1996-09-24
EP0751945A1 (en) 1997-01-08
FI963808A7 (fi) 1996-09-24
FI963808L (fi) 1996-09-24
JPH09510968A (ja) 1997-11-04
DK0751945T3 (da) 1999-04-12
HU9602614D0 (en) 1996-11-28
NO964009L (no) 1996-11-22

Similar Documents

Publication Publication Date Title
HU9602721D0 (en) Use of serotonin antagonists (5ht3) for treating fibromyalgia
ES2124373T3 (es) Procedimiento para la preparacion de derivados del acido n-acil-n,n',n'-etilendiamintriacetico.
AU594488B2 (en) Agents for the treatment of arthroses
TR199801348T2 (xx) Heterosikl-kondanse morfinoid t�revleri(II).
TW353067B (en) Isoquinolines
NO901536L (no) Fremgangsmaate ved desoxydasjon av vann, spesielt sjoevann.
ES2029787T3 (es) Procedimiento para la preparacion de (2,2)-paraciclofanos halogenados y mezclas de (2,2)-paraciclofanos halogenados resultantes.
ES8603351A1 (es) Un metodo para someter a tratamiento un sistema acuoso susceptible de ser sujeto a contaminacion biologica
ES2120185T3 (es) Procedimiento para preparar (1h-tetrazol-5-il)tetrazolo(1,5-a)quinolinas y naftiridinas.
ES2038127T3 (es) Procedimiento para preparar monosulfactamas.
TW278071B (es)
ES8500058A1 (es) Procedimiento para preparar soluciones miscibles en agua de un agente controlador de la coccidiosis
ES8705421A1 (es) Un procedimiento para la preparacion de 4-amino-2-fenil-quinolinas
NZ219032A (en) Method for preservation of wood with substituted phenol derivatives
ES2013025A6 (es) Un metodo para preparar 24r-escimnol.
MY101961A (en) 4-nitrogen substituted isoquinolinol compounds having cardiotonic, phosphodiesterease fraction iii inhibiting properties and/or renal vasodilating properties
EP0194977A3 (en) Method of lighting generic interiors, in particular so-called open-space work interiors
SU1540328A1 (ru) Ингибитор сероводородной коррозии стали
ZA929175B (en) 5,6-dihydro-dibenz(b,e)azepine-6,11-dione-11-oximes.
TR199701011A2 (xx) 1-karba-(detia)-sefalosforin t�revleri.
NO862930L (no) Fremgangsmaate for belegning av staalkonstruksjoner i vann.
UA10395C2 (uk) Спосіб одержаhhя модифікатора гуми
MX9603722A (es) Nuevos pseudopeptidos sustituidos con heterociclos.
DK488288A (da) Fremgangsmaade til bekaempelse af korrosion i vaeskebeholdere indeholdende carbonhydrider
ES8500214A1 (es) "procedimiento para la obtencion de derivados de 2-metilamino-benzofenona"

Legal Events

Date Code Title Description
FG2A Definitive protection

Ref document number: 751945

Country of ref document: ES