EP3237389A4 - 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one as a seed treatment - Google Patents

5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one as a seed treatment Download PDF

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Publication number
EP3237389A4
EP3237389A4 EP15874200.7A EP15874200A EP3237389A4 EP 3237389 A4 EP3237389 A4 EP 3237389A4 EP 15874200 A EP15874200 A EP 15874200A EP 3237389 A4 EP3237389 A4 EP 3237389A4
Authority
EP
European Patent Office
Prior art keywords
alkyl
dihydropyrimidin
arylsulfonyl
imino
fluoro
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
EP15874200.7A
Other languages
German (de)
English (en)
French (fr)
Other versions
EP3237389A1 (en
Inventor
Carla J.R. Klittich
Chenglin Yao
W. John Owen
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Adama Makhteshim Ltd
Original Assignee
Adama Makhteshim Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Adama Makhteshim Ltd filed Critical Adama Makhteshim Ltd
Publication of EP3237389A1 publication Critical patent/EP3237389A1/en
Publication of EP3237389A4 publication Critical patent/EP3237389A4/en
Pending legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01C—PLANTING; SOWING; FERTILISING
    • A01C1/00—Apparatus, or methods of use thereof, for testing or treating seed, roots, or the like, prior to sowing or planting
    • A01C1/06—Coating or dressing seed
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Agronomy & Crop Science (AREA)
  • Soil Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pretreatment Of Seeds And Plants (AREA)
EP15874200.7A 2014-12-23 2015-12-18 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one as a seed treatment Pending EP3237389A4 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201462096301P 2014-12-23 2014-12-23
PCT/US2015/066756 WO2016106138A1 (en) 2014-12-23 2015-12-18 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one as a seed treatment

Publications (2)

Publication Number Publication Date
EP3237389A1 EP3237389A1 (en) 2017-11-01
EP3237389A4 true EP3237389A4 (en) 2018-05-30

Family

ID=56151456

Family Applications (1)

Application Number Title Priority Date Filing Date
EP15874200.7A Pending EP3237389A4 (en) 2014-12-23 2015-12-18 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one as a seed treatment

Country Status (23)

Country Link
US (2) US20180000082A1 (zh)
EP (1) EP3237389A4 (zh)
JP (2) JP2018508468A (zh)
KR (1) KR20170105527A (zh)
CN (2) CN107250117A (zh)
AR (1) AR103283A1 (zh)
AU (1) AU2015369906C1 (zh)
BR (2) BR112017013733B1 (zh)
CA (1) CA2971719C (zh)
CL (1) CL2017001686A1 (zh)
CO (1) CO2017007059A2 (zh)
CR (1) CR20170325A (zh)
EA (1) EA201791444A1 (zh)
EC (1) ECSP17046205A (zh)
IL (1) IL252983B (zh)
MA (1) MA41272A (zh)
MX (1) MX2017008370A (zh)
PE (1) PE20171098A1 (zh)
PH (1) PH12017501171A1 (zh)
TW (1) TWI699162B (zh)
UA (1) UA125789C2 (zh)
WO (1) WO2016106138A1 (zh)
ZA (1) ZA201704838B (zh)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL2938194T3 (pl) 2012-12-28 2020-09-21 Adama Makhteshim Ltd. Pochodne n-podstawionego 5-fluoro-4-imino-3-metylo-2-okso-3,4-dihydropirymidyno-1(2h)-karboksylanu
EP2953463B1 (en) 2012-12-31 2021-03-17 Adama Makhteshim Ltd. 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1h)-one derivatives as fungicides
US9532570B2 (en) 2013-12-31 2017-01-03 Adama Makhteshim Ltd. Synergistic fungicidal mixtures comprising 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2(1H)-one for fungal control in cereals
WO2015103142A1 (en) 2013-12-31 2015-07-09 Dow Agrosciences Llc 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1- (arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation
ME03385B (me) 2014-12-23 2020-01-20 Novartis Ag Triazolopirimidin jedinjenja i njihova upotreba
EP3472166A1 (en) 2016-06-20 2019-04-24 Novartis AG Imidazopyrimidine compounds useful for the treatment of cancer
ES2798424T3 (es) 2016-06-20 2020-12-11 Novartis Ag Compuestos de triazolopiridina y usos de estos
MX2018016331A (es) 2016-06-20 2019-05-20 Novartis Ag Formas cristalinas de compuesto de triazolopirimidina.
TWI801380B (zh) * 2017-05-02 2023-05-11 美商科迪華農業科技有限責任公司 一種非環狀吡啶醯胺化合物作為殺真菌劑以防治在果園、葡萄藤園及農園作物中的植物病原性真菌之用途
TW201902357A (zh) * 2017-05-02 2019-01-16 美商陶氏農業科學公司 用作種子處理之無環吡啶醯胺
TWI774762B (zh) * 2017-05-02 2022-08-21 美商科迪華農業科技有限責任公司 非環狀吡啶醯胺作為一種殺真菌劑以防治蔬菜中植物病原性真菌的用途
TWI801381B (zh) * 2017-05-02 2023-05-11 美商科迪華農業科技有限責任公司 非環狀吡啶醯胺化合物作為殺真菌劑以防治行栽作物中具植物病原性的真菌之用途
CN110996665B (zh) 2017-05-02 2021-10-26 陶氏益农公司 无环吡啶酰胺化合物作为针对草坪草上的真菌病害的杀真菌剂的用途
MA49639A (fr) * 2017-07-17 2020-05-27 Adama Makhteshim Ltd Polymorphes de 5-fluoro-4-imino-3-méthyl-1-tosyl-3,4-dihydropyrimidin-2-one
CA3115684A1 (en) 2018-10-15 2020-04-23 Dow Agrosciences Llc Methods for sythesis of oxypicolinamides
TW202031640A (zh) 2018-11-05 2020-09-01 以色列商亞達瑪馬克天辛有限公司 包括5-氟-4-亞胺基-3-甲基-1-甲苯磺醯基-3,4-二氫嘧啶-2-酮之混合物及組合物，以及其使用方法
CA3145270A1 (en) * 2019-07-22 2021-01-28 Sami SHABTAI Fungicidal combinations, mixtures and compositions and uses thereof
AU2021267206A1 (en) 2020-05-04 2022-12-08 Adama Makhteshim Ltd. Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof
BR112023014997A2 (pt) 2021-01-27 2023-10-03 Adama Makhteshim Ltd 5-fluoro-4-imino-3-metil-1-tosil-3,4-di-hidropirimidin-2(1h)-ona para controle de doenças de plantas
AU2022268726A1 (en) 2021-05-04 2023-11-23 Adama Makhteshim Ltd. Crystalline forms of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4- dihydropyrimidin-2-one, and mixtures, compositions and methods of use thereof
CN114230395B (zh) * 2021-12-16 2022-12-06 河北安格诺农化有限公司 一种缓释药肥组合物及其应用
AR128692A1 (es) 2022-03-03 2024-06-05 Adama Makhteshim Ltd Combinaciones, mezclas y composiciones fungicidas y usos de las mismas
WO2023228148A1 (en) 2022-05-26 2023-11-30 Adama Makhteshim Ltd. Fungicidal combinations, mixtures and compositions and uses thereof

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2015103262A1 (en) * 2013-12-31 2015-07-09 Dow Agrosciences Llc Synergistic fungicidal mixtures for fungal control in cereals

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7687434B2 (en) * 2000-12-22 2010-03-30 Monsanto Technology, Llc Method of improving yield and vigor of plants
UA90209C2 (ru) * 2006-02-09 2010-04-12 Синджента Партисипейшнс Аг Фунгицидная композиция, способ борьбы с заболеваниями полезных растений и способ защиты товаров
SI2563129T1 (sl) * 2010-04-26 2016-12-30 Adama Makhteshim Ltd. N3-substituirani-N1-sulfonil-fluoropirimidinonski derivati
EP2775842B1 (en) * 2011-08-17 2017-10-04 Adama Makhteshim Ltd. 1-substituted-5-fluoro-3,6-dihydro-6-imino-2(1H)-pyrimidinone derivatives as fungicidal agents for use in plant protection
EP2953463B1 (en) * 2012-12-31 2021-03-17 Adama Makhteshim Ltd. 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1h)-one derivatives as fungicides

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2015103262A1 (en) * 2013-12-31 2015-07-09 Dow Agrosciences Llc Synergistic fungicidal mixtures for fungal control in cereals

Also Published As

Publication number Publication date
US20220104489A1 (en) 2022-04-07
US20180000082A1 (en) 2018-01-04
UA125789C2 (uk) 2022-06-08
WO2016106138A1 (en) 2016-06-30
CN117099786A (zh) 2023-11-24
EP3237389A1 (en) 2017-11-01
BR112017013733A2 (pt) 2018-03-13
MA41272A (fr) 2017-10-31
IL252983A0 (en) 2017-08-31
AU2015369906A1 (en) 2017-07-27
CL2017001686A1 (es) 2018-02-02
ZA201704838B (en) 2020-11-25
MX2017008370A (es) 2018-04-30
CA2971719A1 (en) 2016-06-30
TW201628499A (zh) 2016-08-16
CR20170325A (es) 2017-08-29
CA2971719C (en) 2023-09-05
AU2015369906A8 (en) 2017-08-03
JP7075451B2 (ja) 2022-05-25
CN107250117A (zh) 2017-10-13
AR103283A1 (es) 2017-04-26
ECSP17046205A (es) 2017-09-29
PH12017501171A1 (en) 2017-12-11
TWI699162B (zh) 2020-07-21
BR122020000183B1 (pt) 2022-04-26
AU2015369906B2 (en) 2020-03-19
PE20171098A1 (es) 2017-08-07
AU2015369906C1 (en) 2020-10-15
IL252983B (en) 2020-03-31
EA201791444A1 (ru) 2017-11-30
JP2018508468A (ja) 2018-03-29
JP2020196729A (ja) 2020-12-10
BR112017013733B1 (pt) 2021-08-10
KR20170105527A (ko) 2017-09-19
CO2017007059A2 (es) 2017-10-10

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