EP1494674A4 - Derives de carboximide utiles comme bloqueurs uroselectifs du recepteur adrenergique alpha-sb-1a - Google Patents
Derives de carboximide utiles comme bloqueurs uroselectifs du recepteur adrenergique alpha-sb-1aInfo
- Publication number
- EP1494674A4 EP1494674A4 EP02720343A EP02720343A EP1494674A4 EP 1494674 A4 EP1494674 A4 EP 1494674A4 EP 02720343 A EP02720343 A EP 02720343A EP 02720343 A EP02720343 A EP 02720343A EP 1494674 A4 EP1494674 A4 EP 1494674A4
- Authority
- EP
- European Patent Office
- Prior art keywords
- uro
- useful
- selective alpha
- adrenoceptor blockers
- carboximide derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
- C07D295/125—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
- C07D295/13—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Heart & Thoracic Surgery (AREA)
- Urology & Nephrology (AREA)
- Cardiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
PCT/IB2002/001108 WO2003084541A1 (fr) | 2002-04-08 | 2002-04-08 | Derives de carboximide utiles comme bloqueurs uroselectifs du recepteur adrenergique $g(a)1a |
Publications (2)
Publication Number | Publication Date |
---|---|
EP1494674A1 EP1494674A1 (fr) | 2005-01-12 |
EP1494674A4 true EP1494674A4 (fr) | 2006-04-12 |
Family
ID=28686909
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EP02720343A Withdrawn EP1494674A4 (fr) | 2002-04-08 | 2002-04-08 | Derives de carboximide utiles comme bloqueurs uroselectifs du recepteur adrenergique alpha-sb-1a |
Country Status (8)
Country | Link |
---|---|
EP (1) | EP1494674A4 (fr) |
JP (1) | JP2005532282A (fr) |
CN (1) | CN1627946A (fr) |
AU (1) | AU2002251409A1 (fr) |
BR (1) | BR0215686A (fr) |
EA (1) | EA200401335A1 (fr) |
MX (1) | MXPA04009821A (fr) |
WO (1) | WO2003084541A1 (fr) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU2003259391A1 (en) * | 2003-08-25 | 2005-03-10 | Ranbaxy Laboratories Limited | Metabolites of 1-{3-4`4-(2-methoxyphenyl) piperazin-1-yl!-propyl}-piperidine-2, 6-dione for use in the treatment of benign prostatic hyperplasia |
WO2005037281A1 (fr) * | 2003-10-15 | 2005-04-28 | Ranbaxy Laboratories Limited | Derives de 1-alkylpiperazinyl-pyrrolidin-2,5-dione utiles comme antagonistes du recepteur adrenergique |
Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1997037983A1 (fr) * | 1996-04-05 | 1997-10-16 | Societe De Conseils De Recherches Et D'applications Scientifiques (S.C.R.A.S.) | ANTAGONISTES DU RECEPTEUR α1-ADRENERGIQUE |
WO1999006384A1 (fr) * | 1997-08-01 | 1999-02-11 | Recordati S.A., Chemical And Pharmaceutical Company | Derives de 1-(n-phenylaminoalkyl)-piperazine substitues a la position 2 du cycle phenyle |
US6083950A (en) * | 1997-11-13 | 2000-07-04 | Ranbaxy Laboratories Limited | 1-(4-arylpiperazin-1-yl)-ω-[n-(α,ω-dicarboximido)]-alka nes useful as uro-selective α1-adrenoceptor blockers |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2781220B1 (fr) * | 1998-07-17 | 2000-10-13 | Lafon Labor | Piperazinones substituees en beta |
-
2002
- 2002-04-08 CN CNA028290976A patent/CN1627946A/zh active Pending
- 2002-04-08 WO PCT/IB2002/001108 patent/WO2003084541A1/fr active Application Filing
- 2002-04-08 BR BR0215686-5A patent/BR0215686A/pt not_active IP Right Cessation
- 2002-04-08 JP JP2003581781A patent/JP2005532282A/ja not_active Withdrawn
- 2002-04-08 AU AU2002251409A patent/AU2002251409A1/en not_active Abandoned
- 2002-04-08 EP EP02720343A patent/EP1494674A4/fr not_active Withdrawn
- 2002-04-08 MX MXPA04009821A patent/MXPA04009821A/es not_active Application Discontinuation
- 2002-04-08 EA EA200401335A patent/EA200401335A1/ru unknown
Patent Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO1997037983A1 (fr) * | 1996-04-05 | 1997-10-16 | Societe De Conseils De Recherches Et D'applications Scientifiques (S.C.R.A.S.) | ANTAGONISTES DU RECEPTEUR α1-ADRENERGIQUE |
WO1999006384A1 (fr) * | 1997-08-01 | 1999-02-11 | Recordati S.A., Chemical And Pharmaceutical Company | Derives de 1-(n-phenylaminoalkyl)-piperazine substitues a la position 2 du cycle phenyle |
US6083950A (en) * | 1997-11-13 | 2000-07-04 | Ranbaxy Laboratories Limited | 1-(4-arylpiperazin-1-yl)-ω-[n-(α,ω-dicarboximido)]-alka nes useful as uro-selective α1-adrenoceptor blockers |
Non-Patent Citations (1)
Title |
---|
See also references of WO03084541A1 * |
Also Published As
Publication number | Publication date |
---|---|
JP2005532282A (ja) | 2005-10-27 |
EP1494674A1 (fr) | 2005-01-12 |
BR0215686A (pt) | 2005-02-22 |
EA200401335A1 (ru) | 2006-02-24 |
WO2003084541A1 (fr) | 2003-10-16 |
AU2002251409A1 (en) | 2003-10-20 |
MXPA04009821A (es) | 2004-12-13 |
CN1627946A (zh) | 2005-06-15 |
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Legal Events
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PUAI | Public reference made under article 153(3) epc to a published international application that has entered the european phase |
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A4 | Supplementary search report drawn up and despatched |
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GRAS | Grant fee paid |
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RAP1 | Party data changed (applicant data changed or rights of an application transferred) |
Owner name: RANBAXY LABORATORIES LIMITED |
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STAA | Information on the status of an ep patent application or granted ep patent |
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