EP1135023A4 - Composes aminobenzisoxazole et banques contenant de tels composes - Google Patents

Composes aminobenzisoxazole et banques contenant de tels composes

Info

Publication number
EP1135023A4
EP1135023A4 EP99958891A EP99958891A EP1135023A4 EP 1135023 A4 EP1135023 A4 EP 1135023A4 EP 99958891 A EP99958891 A EP 99958891A EP 99958891 A EP99958891 A EP 99958891A EP 1135023 A4 EP1135023 A4 EP 1135023A4
Authority
EP
European Patent Office
Prior art keywords
libraries
aminobenzisoxazole compounds
aminobenzisoxazole
compounds
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
EP99958891A
Other languages
German (de)
English (en)
Other versions
EP1135023A1 (fr
Inventor
Michael Robert Wiley
Savatore Donato Lepore
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly and Co filed Critical Eli Lilly and Co
Publication of EP1135023A1 publication Critical patent/EP1135023A1/fr
Publication of EP1135023A4 publication Critical patent/EP1135023A4/fr
Withdrawn legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/20—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C40—COMBINATORIAL TECHNOLOGY
    • C40B—COMBINATORIAL CHEMISTRY; LIBRARIES, e.g. CHEMICAL LIBRARIES
    • C40B40/00—Libraries per se, e.g. arrays, mixtures
    • G—PHYSICS
    • G01—MEASURING; TESTING
    • G01N—INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
    • G01N2333/00—Assays involving biological materials from specific organisms or of a specific nature
    • G01N2333/90—Enzymes; Proenzymes
    • G01N2333/914—Hydrolases (3)
    • G01N2333/948—Hydrolases (3) acting on peptide bonds (3.4)
    • G01N2333/974—Thrombin

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
EP99958891A 1998-11-12 1999-11-12 Composes aminobenzisoxazole et banques contenant de tels composes Withdrawn EP1135023A4 (fr)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US10820898P 1998-11-12 1998-11-12
US108208P 1998-11-12
US12915199P 1999-04-14 1999-04-14
US129151P 1999-04-14
US14549299P 1999-07-22 1999-07-22
US145492P 1999-07-22
PCT/US1999/026635 WO2000027199A1 (fr) 1998-11-12 1999-11-12 Composes aminobenzisoxazole et banques contenant de tels composes

Publications (2)

Publication Number Publication Date
EP1135023A1 EP1135023A1 (fr) 2001-09-26
EP1135023A4 true EP1135023A4 (fr) 2003-03-05

Family

ID=27380448

Family Applications (1)

Application Number Title Priority Date Filing Date
EP99958891A Withdrawn EP1135023A4 (fr) 1998-11-12 1999-11-12 Composes aminobenzisoxazole et banques contenant de tels composes

Country Status (3)

Country Link
EP (1) EP1135023A4 (fr)
AU (1) AU1616600A (fr)
WO (1) WO2000027199A1 (fr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6569879B2 (en) * 2000-02-18 2003-05-27 Merck & Co., Inc. Aryloxyacetic acids for diabetes and lipid disorders
DE102005038947A1 (de) 2005-05-18 2006-11-30 Grünenthal GmbH Substituierte Benzo[d]isoxazol-3-yl-amin-Verbindungen und deren Verwendung in Arzneimitteln
CA3142793A1 (fr) * 2019-06-11 2020-12-17 Fresenius Medical Care Holdings, Inc. Systemes et procedes de mesure des caracteristiques electriques de fluides medicaux
CN116685845A (zh) 2021-01-11 2023-09-01 费森尤斯医疗保健控股公司 用于测量医用流体的电特性的系统和方法

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0816376A1 (fr) * 1996-06-25 1998-01-07 Eli Lilly And Company Inhibiteurs de thrombin comme agents anticoagulants
WO1998057951A1 (fr) * 1997-06-19 1998-12-23 Du Pont Pharmaceuticals Company NOUVEAUX IMITATEURS DE GUANIDINE UTILISES EN TANT QU'INHIBITEURS DU FACTEUR Xa
WO2000026210A1 (fr) * 1998-10-30 2000-05-11 Merck & Co., Inc. Inhibiteurs de la thrombine
WO2000027627A1 (fr) * 1998-11-12 2000-05-18 Eli Lilly And Company Lieurs d'aryloxime dans la synthese de la phase solide de 3-aminobenzisoxazoles

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5455274A (en) * 1992-12-09 1995-10-03 Ciba-Geigy Corporation Hydroxyamidine derivatives
WO1996006837A1 (fr) * 1994-08-30 1996-03-07 Sankyo Company, Limited Isoxazoles
JP2891187B2 (ja) * 1995-06-22 1999-05-17 信越半導体株式会社 ワイヤーソー装置及び切断方法
AU4153497A (en) * 1996-08-26 1998-03-19 Eli Lilly And Company Combinatorial process for preparing substituted thiophene libraries

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0816376A1 (fr) * 1996-06-25 1998-01-07 Eli Lilly And Company Inhibiteurs de thrombin comme agents anticoagulants
WO1998057951A1 (fr) * 1997-06-19 1998-12-23 Du Pont Pharmaceuticals Company NOUVEAUX IMITATEURS DE GUANIDINE UTILISES EN TANT QU'INHIBITEURS DU FACTEUR Xa
WO2000026210A1 (fr) * 1998-10-30 2000-05-11 Merck & Co., Inc. Inhibiteurs de la thrombine
WO2000027627A1 (fr) * 1998-11-12 2000-05-18 Eli Lilly And Company Lieurs d'aryloxime dans la synthese de la phase solide de 3-aminobenzisoxazoles

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
See also references of WO0027199A1 *

Also Published As

Publication number Publication date
EP1135023A1 (fr) 2001-09-26
WO2000027199A1 (fr) 2000-05-18
AU1616600A (en) 2000-05-29

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Legal Events

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