EP1122261A3 - 13- und 14-Gliederige Antibakterielle-Makroliden - Google Patents

13- und 14-Gliederige Antibakterielle-Makroliden Download PDF

Info

Publication number
EP1122261A3
EP1122261A3 EP01300521A EP01300521A EP1122261A3 EP 1122261 A3 EP1122261 A3 EP 1122261A3 EP 01300521 A EP01300521 A EP 01300521A EP 01300521 A EP01300521 A EP 01300521A EP 1122261 A3 EP1122261 A3 EP 1122261A3
Authority
EP
European Patent Office
Prior art keywords
membered
antibacterial
compounds
antiprotozoal
relates
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
EP01300521A
Other languages
English (en)
French (fr)
Other versions
EP1122261A2 (de
Inventor
Takushi Kaneko
William Thomas Mcmillen
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Products Inc
Original Assignee
Pfizer Products Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc filed Critical Pfizer Products Inc
Publication of EP1122261A2 publication Critical patent/EP1122261A2/de
Publication of EP1122261A3 publication Critical patent/EP1122261A3/de
Withdrawn legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/02—Heterocyclic radicals containing only nitrogen as ring hetero atoms

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
EP01300521A 2000-01-31 2001-01-22 13- und 14-Gliederige Antibakterielle-Makroliden Withdrawn EP1122261A3 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US17932400P 2000-01-31 2000-01-31
US179324P 2000-01-31

Publications (2)

Publication Number Publication Date
EP1122261A2 EP1122261A2 (de) 2001-08-08
EP1122261A3 true EP1122261A3 (de) 2001-09-26

Family

ID=22656089

Family Applications (1)

Application Number Title Priority Date Filing Date
EP01300521A Withdrawn EP1122261A3 (de) 2000-01-31 2001-01-22 13- und 14-Gliederige Antibakterielle-Makroliden

Country Status (4)

Country Link
EP (1) EP1122261A3 (de)
JP (1) JP2001213893A (de)
BR (1) BR0100228A (de)
CA (1) CA2332686C (de)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4043191B2 (ja) 1998-11-03 2008-02-06 ファイザー・プロダクツ・インク 新規なマクロライド抗生物質
EP1147121B1 (de) 1999-01-27 2003-12-17 Pfizer Products Inc. Ketolid-antibiotika
WO2000071557A1 (en) 1999-05-24 2000-11-30 Pfizer Products Inc. 13-methyl-erythromycin derivatives
WO2003022289A1 (fr) * 2001-09-05 2003-03-20 Hokuriku Seiyaku Co., Ltd. Medicament contenant de l'erythromycine pour traiter ou prevenir la tuberculose
AU2003211113B2 (en) 2002-02-15 2007-08-09 Merckle Gmbh Antibiotic conjugates
AU2003215245A1 (en) 2002-02-15 2003-09-09 Sympore Gmbh Conjugates of biologically active compounds, methods for their preparation and use, formulation and pharmaceutical applications thereof
EP1483277A4 (de) 2002-02-15 2007-10-03 Merckle Gmbh Konjugate biologisch aktiver verbindungen, verfahren zu deren herstellung und anwendung, formulierung und pharmazeutische anwendungen davon
BRPI0519135A2 (pt) 2004-12-21 2008-12-23 Pfizer Prod Inc macrolÍdeos
WO2010086351A1 (en) * 2009-01-30 2010-08-05 Glaxosmithkline Istrazivacki Centar Zagreb D.O.O. 3'-n-substituted 9-deoxo-9a-methyl-9a-aza-homoerythromycin having antimalarial activity

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1992018134A1 (en) * 1991-04-09 1992-10-29 Abbott Laboratories Macrocyclic lactam prokinetic agents

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1992018134A1 (en) * 1991-04-09 1992-10-29 Abbott Laboratories Macrocyclic lactam prokinetic agents

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
FAGHIH R ET AL: "Preparation of 9-deoxo-4-deoxy-6,9-epoxyerythromycin lactams motilactides: potent and orally active prokinetic agents", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,GB,OXFORD, vol. 8, no. 7, 7 April 1998 (1998-04-07), pages 805 - 810, XP004136969, ISSN: 0960-894X *

Also Published As

Publication number Publication date
JP2001213893A (ja) 2001-08-07
CA2332686C (en) 2005-06-07
BR0100228A (pt) 2001-08-28
CA2332686A1 (en) 2001-07-31
EP1122261A2 (de) 2001-08-08

Similar Documents

Publication Publication Date Title
CA2316919A1 (en) Novel macrolides
WO2004080391A3 (en) Novel antibacterial agents
WO2001058412A3 (de) Extrakte von rückständen aus der weinherstellung
MXPA03003168A (es) Composicion antibiotica topica para el tratamiento de infeccion de los ojos.
WO2002048147A3 (en) Pyrazolopyridines
CA2343236A1 (en) 4,4-biarylpiperidine derivatives
CA2359354A1 (en) Medicament for the treatment, prevention and diagnosis of infection due to chlamydia pneumoniae
CA2303498A1 (en) Dioxocyclopentyl hydroxamic acids
CA2359708A1 (en) Ketolide antibiotics
WO2001035950A3 (en) Benzamide therapeutics and methods for treating inflammatory bowel disease
HUP0400832A3 (en) New amidoalkyl-piperidine and amidoalkyl-piperazine derivatives, and pharmaceutical compositions containing such derivatives as active ingredients
WO2000026224A3 (en) Novel macrolide antibiotics
CA2415354A1 (en) Phospholipid derivatives of valproic acid and mixtures thereof
WO2002042315A3 (en) Macrolide solvates
EP1122261A3 (de) 13- und 14-Gliederige Antibakterielle-Makroliden
WO2003018059A3 (de) Kombinationspräparate von arylsubstituierten propanolaminderivaten mit weiteren wirkstoffen und deren verwendung
EP1114826A3 (de) Antibakterielle und prokinetische Makroliden
AU2001289714A1 (en) Benzofuran derivatives and their use as antibacterial agents
MXPA04001773A (es) Derivados de 6,7-dihidroxitetrahidroisquinolinas 3-sustituidas parta uso como agentes antibacterianos.
WO2000040232A3 (en) Bretylium compositions and kits, and their use in preventing and treating cardiovascular conditions
WO2003024996A3 (de) Antibakterielle makrozyklen
CA2351829A1 (en) Macrolide antibiotics
CA2299036A1 (en) 4-phenyl-4-heteroarylpiperidine derivatives
GB0025688D0 (en) Macrolides
WO2002070537A3 (en) Fusidic acid derivatives

Legal Events

Date Code Title Description
PUAI Public reference made under article 153(3) epc to a published international application that has entered the european phase

Free format text: ORIGINAL CODE: 0009012

17P Request for examination filed

Effective date: 20010122

AK Designated contracting states

Kind code of ref document: A2

Designated state(s): AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU NL PT SE TR

Kind code of ref document: A2

Designated state(s): AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR

AX Request for extension of the european patent

Free format text: AL;LT;LV;MK;RO;SI

PUAL Search report despatched

Free format text: ORIGINAL CODE: 0009013

AK Designated contracting states

Kind code of ref document: A3

Designated state(s): AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR

AX Request for extension of the european patent

Free format text: AL;LT;LV;MK;RO;SI

AKX Designation fees paid

Free format text: AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR

RBV Designated contracting states (corrected)

Designated state(s): AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU NL PT SE TR

17Q First examination report despatched

Effective date: 20020702

STAA Information on the status of an ep patent application or granted ep patent

Free format text: STATUS: THE APPLICATION IS DEEMED TO BE WITHDRAWN

18D Application deemed to be withdrawn

Effective date: 20030114