EP0812196A4 - ANTAGONISTES DU RECEPTEUR ALPHA-1a-ADRENERGIQUE - Google Patents

ANTAGONISTES DU RECEPTEUR ALPHA-1a-ADRENERGIQUE

Info

Publication number
EP0812196A4
EP0812196A4 EP96905575A EP96905575A EP0812196A4 EP 0812196 A4 EP0812196 A4 EP 0812196A4 EP 96905575 A EP96905575 A EP 96905575A EP 96905575 A EP96905575 A EP 96905575A EP 0812196 A4 EP0812196 A4 EP 0812196A4
Authority
EP
European Patent Office
Prior art keywords
alpha
receptor antagonists
adrenergic receptor
adrenergic
antagonists
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
EP96905575A
Other languages
German (de)
English (en)
Other versions
EP0812196A1 (fr
Inventor
Ben E Evans
Gerald S Ponticello
Jacob M Hoffman
Raymond S L Chang
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck and Co Inc
Original Assignee
Merck and Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9603457.4A external-priority patent/GB9603457D0/en
Application filed by Merck and Co Inc filed Critical Merck and Co Inc
Publication of EP0812196A1 publication Critical patent/EP0812196A1/fr
Publication of EP0812196A4 publication Critical patent/EP0812196A4/fr
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
EP96905575A 1995-02-23 1996-02-23 ANTAGONISTES DU RECEPTEUR ALPHA-1a-ADRENERGIQUE Ceased EP0812196A4 (fr)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US39269995A 1995-02-23 1995-02-23
US392699 1995-02-23
US253495P 1995-08-18 1995-08-18
US2534 1995-08-18
GB9603457 1996-02-19
GBGB9603457.4A GB9603457D0 (fr) 1996-02-19 1996-02-19
PCT/US1996/002534 WO1996025934A1 (fr) 1995-02-23 1996-02-23 ANTAGONISTES DU RECEPTEUR ALPHA-1a-ADRENERGIQUE

Publications (2)

Publication Number Publication Date
EP0812196A1 EP0812196A1 (fr) 1997-12-17
EP0812196A4 true EP0812196A4 (fr) 1998-05-20

Family

ID=26308756

Family Applications (1)

Application Number Title Priority Date Filing Date
EP96905575A Ceased EP0812196A4 (fr) 1995-02-23 1996-02-23 ANTAGONISTES DU RECEPTEUR ALPHA-1a-ADRENERGIQUE

Country Status (4)

Country Link
EP (1) EP0812196A4 (fr)
JP (1) JPH11508536A (fr)
AU (1) AU700559B2 (fr)
CA (1) CA2213192A1 (fr)

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4110449A (en) * 1977-05-23 1978-08-29 E. R. Squibb & Sons, Inc. 2-substituted benzisothiazol-3-ones
WO1995028397A1 (fr) * 1994-04-14 1995-10-26 Merck & Co., Inc. Antagonistes du recepteur adrenergique alpha1c
US5462942A (en) * 1993-07-05 1995-10-31 Duphar International Research B.V. 2,3-dihydro-1,4-benzodioxin-5-yl-piperazine derivatives having 5-HT 1A-antagonistic activity

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4110449A (en) * 1977-05-23 1978-08-29 E. R. Squibb & Sons, Inc. 2-substituted benzisothiazol-3-ones
US5462942A (en) * 1993-07-05 1995-10-31 Duphar International Research B.V. 2,3-dihydro-1,4-benzodioxin-5-yl-piperazine derivatives having 5-HT 1A-antagonistic activity
WO1995028397A1 (fr) * 1994-04-14 1995-10-26 Merck & Co., Inc. Antagonistes du recepteur adrenergique alpha1c

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
See also references of WO9625934A1 *

Also Published As

Publication number Publication date
AU700559B2 (en) 1999-01-07
CA2213192A1 (fr) 1996-08-29
JPH11508536A (ja) 1999-07-27
AU4930196A (en) 1996-09-11
EP0812196A1 (fr) 1997-12-17

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Legal Events

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