EP0730595A4 - Imidazolinobenzodiazepine - Google Patents

Imidazolinobenzodiazepine

Info

Publication number
EP0730595A4
EP0730595A4 EP95901942A EP95901942A EP0730595A4 EP 0730595 A4 EP0730595 A4 EP 0730595A4 EP 95901942 A EP95901942 A EP 95901942A EP 95901942 A EP95901942 A EP 95901942A EP 0730595 A4 EP0730595 A4 EP 0730595A4
Authority
EP
European Patent Office
Prior art keywords
imidazolinobenzodiazepines
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
EP95901942A
Other languages
English (en)
French (fr)
Other versions
EP0730595A1 (de
Inventor
Mark G Bock
Roger M Freidinger
Robert M Dipardo
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck and Co Inc
Original Assignee
Merck and Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck and Co Inc filed Critical Merck and Co Inc
Publication of EP0730595A1 publication Critical patent/EP0730595A1/de
Publication of EP0730595A4 publication Critical patent/EP0730595A4/de
Withdrawn legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Anesthesiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
EP95901942A 1993-11-22 1994-11-18 Imidazolinobenzodiazepine Withdrawn EP0730595A4 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US15621093A 1993-11-22 1993-11-22
US156210 1993-11-22
PCT/US1994/013325 WO1995014693A1 (en) 1993-11-22 1994-11-18 Imidazolinobenzodiazepines

Publications (2)

Publication Number Publication Date
EP0730595A1 EP0730595A1 (de) 1996-09-11
EP0730595A4 true EP0730595A4 (de) 1997-07-16

Family

ID=22558586

Family Applications (1)

Application Number Title Priority Date Filing Date
EP95901942A Withdrawn EP0730595A4 (de) 1993-11-22 1994-11-18 Imidazolinobenzodiazepine

Country Status (5)

Country Link
EP (1) EP0730595A4 (de)
JP (1) JP2840453B2 (de)
AU (1) AU1099695A (de)
CA (1) CA2176017A1 (de)
WO (1) WO1995014693A1 (de)

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0272866A1 (de) * 1986-12-23 1988-06-29 Merck & Co. Inc. 1,4-Benzodiazepine mit 5-gliedrigen heterocyclischen Ringen
EP0518484A2 (de) * 1991-05-14 1992-12-16 Merck & Co. Inc. Mit fünf- oder sechsgliedrigen heterozyklischen Ringverbindungen kondensierte 1,4-Benzodiazepine zur Behandlung von Angstzuständen, Schmerz, Pupillenkontraktion, Entzugserscheinungen oder onkologischen Erkrankungen
WO1995014472A1 (en) * 1993-11-22 1995-06-01 Merck & Co., Inc. Antiarrhythmic benzodiazepines

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4847248A (en) * 1986-12-23 1989-07-11 Merck & Co., Inc. 1,4-Benzodiazepines with 5- and 6-membered heterocyclic rings and their use as cholecystokinins and gastrin antagonists
US5177071A (en) * 1991-06-17 1993-01-05 Merck & Co., Inc. 1,4-benzodiazepines with 6-membered heterocyclic rings to treat panic and anxiety disorder

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0272866A1 (de) * 1986-12-23 1988-06-29 Merck & Co. Inc. 1,4-Benzodiazepine mit 5-gliedrigen heterocyclischen Ringen
EP0518484A2 (de) * 1991-05-14 1992-12-16 Merck & Co. Inc. Mit fünf- oder sechsgliedrigen heterozyklischen Ringverbindungen kondensierte 1,4-Benzodiazepine zur Behandlung von Angstzuständen, Schmerz, Pupillenkontraktion, Entzugserscheinungen oder onkologischen Erkrankungen
WO1995014472A1 (en) * 1993-11-22 1995-06-01 Merck & Co., Inc. Antiarrhythmic benzodiazepines

Non-Patent Citations (3)

* Cited by examiner, † Cited by third party
Title
MARK G. BOCK ET AL.: "CHOLECYSTOKININ ANTAGONISTS.", JOURNAL OF MEDICINAL CHEMISTRY, vol. 31, 1988, WASHINGTON US, pages 176 - 180, XP002030790 *
MARK G. BOCK ET AL.: "SELECTIVE NON PEPTIDE LIGANDS FOR A ACCOMODATING PEPTIDE RECEPTOR.", BIOORGANIC & MEDICINAL CHEMISTRY, vol. 2, no. 9, 1994, GREAT BRITAIN, pages 987 - 998, XP000671854 *
See also references of WO9514693A1 *

Also Published As

Publication number Publication date
EP0730595A1 (de) 1996-09-11
JP2840453B2 (ja) 1998-12-24
CA2176017A1 (en) 1995-06-01
JPH09501444A (ja) 1997-02-10
AU1099695A (en) 1995-06-13
WO1995014693A1 (en) 1995-06-01

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Legal Events

Date Code Title Description
PUAI Public reference made under article 153(3) epc to a published international application that has entered the european phase

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17P Request for examination filed

Effective date: 19960624

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STAA Information on the status of an ep patent application or granted ep patent

Free format text: STATUS: THE APPLICATION IS DEEMED TO BE WITHDRAWN

18D Application deemed to be withdrawn

Effective date: 19991110