ECSP993013A - DERIVATIVES OF 3- (2-OXO- [1,3 '] BIPIRROLIDINIL- 3-ILIDENMETIL) - CEFEMES - Google Patents
DERIVATIVES OF 3- (2-OXO- [1,3 '] BIPIRROLIDINIL- 3-ILIDENMETIL) - CEFEMESInfo
- Publication number
- ECSP993013A ECSP993013A ECSP993013A ECSP993013A EC SP993013 A ECSP993013 A EC SP993013A EC SP993013 A ECSP993013 A EC SP993013A EC SP993013 A ECSP993013 A EC SP993013A
- Authority
- EC
- Ecuador
- Prior art keywords
- hydrogen
- compounds
- ocor
- salts
- cooch
- Prior art date
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
La presente invención se refiere a los compuestos de fórmula I (gráfico), donde R1 es un hidrógeno, C1-6-alquilo, sustituido opcionalmente por flúor, o bien el C3-6-cicloalquilo; R2 es un hidrogeno o un grupo elegido entre -CH2C(=CHR)-COOR, -CH2OCOR, -CH(R)OCOR, -CH(R)OCOOR, CH(OCOR)OCOR, -CH2COCH2OCOR y (gráfico), R3 es un hidrógeno o un grupo elegido entre -CH2C(=CH2)-COOR, -COOCH2C(=CHR)-COOR, -COOCH2OCOR, -COOCH(R)OCOR, -COOCH(R) OCOOR, -COOCH(OCOR) OCOR, -COOCH2COCH2OCOR, y (gráfico), con la condición de que R2 o R3 sea un hidrógeno y el otro R2 o R3 sea distinto de un hidrógeno, R es hidrógeno o C1-6-alquilo; R4 es un hidrógeno o un grupo hidroxi, R5 es un hidrógeno o un w-hidroxialquilo; y X es CH ó N, asi como sales de dichos compuestos aceptables farmacéuticamente e hidratos de los compuestos de fórmula I y sus sales, y con el uso de compuestos de fórmula I y de sales de dichos compuestos aceptables desde un punto de vista farmacéutico e hidratos de dichos compuestos y desus sales para la fabricación de preparados farmacéuticos que contengan dichos compuestos.The present invention refers to the compounds of formula I (graph), where R1 is a hydrogen, C1-6-alkyl, optionally substituted by fluorine, or C3-6-cycloalkyl; R2 is a hydrogen or a group chosen from -CH2C (= CHR) -COOR, -CH2OCOR, -CH (R) OCOR, -CH (R) OCOOR, CH (OCOR) OCOR, -CH2COCH2OCOR and (graph), R3 is a hydrogen or a group chosen from -CH2C (= CH2) -COOR, -COOCH2C (= CHR) -COOR, -COOCH2OCOR, -COOCH (R) OCOR, -COOCH (R) OCOOR, -COOCH (OCOR) OCOR, - COOCH2COCH2OCOR, and (graph), provided that R2 or R3 is a hydrogen and the other R2 or R3 is other than a hydrogen, R is hydrogen or C1-6-alkyl; R4 is a hydrogen or a hydroxy group, R5 is a hydrogen or a w-hydroxyalkyl; and X is CH or N, as well as salts of said pharmaceutically acceptable compounds and hydrates of the compounds of formula I and their salts, and with the use of compounds of formula I and of salts of said pharmaceutically acceptable compounds and hydrates of said compounds and their salts for the manufacture of pharmaceutical preparations containing said compounds.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP993013 ECSP993013A (en) | 1999-06-15 | 1999-06-15 | DERIVATIVES OF 3- (2-OXO- [1,3 '] BIPIRROLIDINIL- 3-ILIDENMETIL) - CEFEMES |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP993013 ECSP993013A (en) | 1999-06-15 | 1999-06-15 | DERIVATIVES OF 3- (2-OXO- [1,3 '] BIPIRROLIDINIL- 3-ILIDENMETIL) - CEFEMES |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP993013A true ECSP993013A (en) | 2000-01-27 |
Family
ID=42044002
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP993013 ECSP993013A (en) | 1999-06-15 | 1999-06-15 | DERIVATIVES OF 3- (2-OXO- [1,3 '] BIPIRROLIDINIL- 3-ILIDENMETIL) - CEFEMES |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP993013A (en) |
-
1999
- 1999-06-15 EC ECSP993013 patent/ECSP993013A/en unknown
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