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Priority to ECSP961876priorityCriticalpatent/ECSP961876A/en
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Pharmaceuticals Containing Other Organic And Inorganic Compounds
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Medicinal Preparation
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Abstract
El invento proporciona una forma de dosificación farmacéutica adaptada para la administración en el tracto gastrointestinal de un paciente que comprende darifenacina, o una de sus sales farmacéuticamente aceptable y un adyuvante diluyente o vehículo farmacéuticamente aceptable caracterizada porque la forma de dosificación está adaptada para liberar al menos el 10% en peso de la darifenacina o de su sal farmacéuticamente aceptable, en el tracto gastrointestinal inferior del paciente. La formulación minimiza los efectos secundarios indeseados y aumenta la biodisponibilidad de la darifenacina.The invention provides a pharmaceutical dosage form adapted for administration to the gastrointestinal tract of a patient comprising darifenacin, or a pharmaceutically acceptable salt thereof and a diluting adjuvant or pharmaceutically acceptable carrier characterized in that the dosage form is adapted to release at least 10% by weight of darifenacin or its pharmaceutically acceptable salt, in the patient's lower gastrointestinal tract. The formulation minimizes unwanted side effects and increases the bioavailability of darifenacin.
LACTAMA COMPOUND (N) - ((S) -2-HIDROXI-3-METHYLBUTIRILE) -1- (L-ALANINIL) - (S) -1-AMINO-3-METHYL-4,5,6,7-TETRAHYDRO -2H-3-BENZAZEPIN-2-ONA, PHARMACEUTICAL COMPOSITION THAT INCLUDES IT, PROCEDURE FOR THE INHIBITION OF THE B-AMYLOID PEPTIDE RELEASE AND / OR ITS SYNTHESIS THAT USES IT AND ITS USE FOR THE FABR
1ALFA, 26 DIHIDROXI-D-HOMO-VITAMIN D3, A PHARMACEUTICAL COMPOSITION THAT INCLUDES IT, A PROCEDURE FOR ITS PREPARATION AND USE OF THEM IN THE ELABORATION OF A MEDICINAL PRODUCT
DERIVATIVE OF NAFTIRIDIN-DIBENZO [A, D] CICLOHEPTENO-10-ACETICO, PHARMACEUTICAL COMPOSITION, AND THE USE OF THAT DERIVATIVE FOR THE MANUFACTURE OF A MEDICINAL PRODUCT.
A BENZAMIDE COMPOUND, A MEDICINAL PRODUCT CONTAINING IT, AND USE FOR THE MANUFACTURE OF A MEDICINAL PRODUCT FOR THE TREATMENT OR PREVENTION OF A DIGESTIVE DISEASE OR TO IMPROVE THE MOBILITY OF THE GASTROINTESTINAL TRACT.