ECSP951574A - ADHESION RECEPTOR ANTAGONISTS - Google Patents
ADHESION RECEPTOR ANTAGONISTSInfo
- Publication number
- ECSP951574A ECSP951574A ECSP951574A ECSP951574A EC SP951574 A ECSP951574 A EC SP951574A EC SP951574 A ECSP951574 A EC SP951574A EC SP951574 A ECSP951574 A EC SP951574A
- Authority
- EC
- Ecuador
- Prior art keywords
- receptor antagonists
- adhesion receptor
- substituted
- hexahydroazepino
- azetidino
- Prior art date
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Compuestos caracterizados por la fórmula I: en la que: X representa O, S, NH o NA, Y representa un resto de aziridino, azetidino, pirrolidino, piperidino, hexahidroazepino o piperazino sustituído con R2, R1 representa R2 es - Cr-H2r-COOR3, R3 es H, A o Ar, A representa alquilo de 1 a 6 átomos de C, B representa H, A, cicloalquilo de 3 a 7 átomos de C, Ar-Ck H2k- o amidino, Ar representa fenilo o bencilo no sustituído, o bien mono o disustituído con A, CI, Br, I, NO2, CN, OA, OH, NH2, NHA y/o NA2, k es 1,2,3 ó 4, m y r son independientemente 0,1,2,3 ó 4, y n es 2,3 ó 4, y sus sales aceptables desde el punto de vista fisiológico.Compounds characterized by formula I: in which: X represents O, S, NH or NA, Y represents an aziridino, azetidino, pyrrolidino, piperidino, hexahydroazepino or piperazino residue substituted with R2, R1 represents R2 is -Cr-H2r- COOR3, R3 is H, A or Ar, A represents C 1-6 alkyl, B represents H, A, C 3-7 cycloalkyl, Ar-Ck H2k- or amidino, Ar represents phenyl or non-benzyl substituted, or mono or disubstituted with A, CI, Br, I, NO2, CN, OA, OH, NH2, NHA and / or NA2, k is 1,2,3 or 4, m and r are independently 0,1,2 , 3 or 4, and n is 2,3 or 4, and their salts are physiologically acceptable.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP951574 ECSP951574A (en) | 1995-11-08 | 1995-11-08 | ADHESION RECEPTOR ANTAGONISTS |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP951574 ECSP951574A (en) | 1995-11-08 | 1995-11-08 | ADHESION RECEPTOR ANTAGONISTS |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP951574A true ECSP951574A (en) | 1997-04-16 |
Family
ID=42042216
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP951574 ECSP951574A (en) | 1995-11-08 | 1995-11-08 | ADHESION RECEPTOR ANTAGONISTS |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP951574A (en) |
-
1995
- 1995-11-08 EC ECSP951574 patent/ECSP951574A/en unknown
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