MX9204342A - INDOLES. - Google Patents

INDOLES.

Info

Publication number
MX9204342A
MX9204342A MX9204342A MX9204342A MX9204342A MX 9204342 A MX9204342 A MX 9204342A MX 9204342 A MX9204342 A MX 9204342A MX 9204342 A MX9204342 A MX 9204342A MX 9204342 A MX9204342 A MX 9204342A
Authority
MX
Mexico
Prior art keywords
indoles
formula
present
provides compounds
pharmaceutical salts
Prior art date
Application number
MX9204342A
Other languages
Spanish (es)
Inventor
Julian Blagg
Kelvin Cooper
Peter Lionel Spargo
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of MX9204342A publication Critical patent/MX9204342A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/12—Radicals substituted by oxygen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Abstract

La presente invención provee compuestos de la fórmula (I) y sales farmacéuticas aceptables de los mismos.The present invention provides compounds of formula (I) and acceptable pharmaceutical salts thereof.

MX9204342A 1991-07-24 1992-07-23 INDOLES. MX9204342A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB919115951A GB9115951D0 (en) 1991-07-24 1991-07-24 Indoles

Publications (1)

Publication Number Publication Date
MX9204342A true MX9204342A (en) 1994-03-31

Family

ID=10698873

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9204342A MX9204342A (en) 1991-07-24 1992-07-23 INDOLES.

Country Status (20)

Country Link
EP (2) EP0598750A1 (en)
JP (2) JPH06511483A (en)
CN (2) CN1068816A (en)
AU (2) AU2327192A (en)
BR (1) BR9206306A (en)
CA (2) CA2112689A1 (en)
CZ (1) CZ13694A3 (en)
FI (2) FI940311A (en)
GB (1) GB9115951D0 (en)
HU (1) HU9400199D0 (en)
IE (2) IE922386A1 (en)
IL (2) IL102545A0 (en)
MX (1) MX9204342A (en)
NO (1) NO940237L (en)
NZ (1) NZ243687A (en)
PT (2) PT100718A (en)
SK (1) SK8494A3 (en)
TW (1) TW223060B (en)
WO (2) WO1993002051A1 (en)
ZA (2) ZA925547B (en)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9204024D0 (en) * 1992-02-25 1992-04-08 Fujisawa Pharmaceutical Co Indole derivatives
GB9302577D0 (en) * 1993-02-10 1993-03-24 Fujisawa Pharmaceutical Co Indole derivatives
US5530019A (en) * 1993-04-05 1996-06-25 Fujisawa Pharmaceutical Co., Ltd. Indole derivatives useful as testosterone 5α-reductase inhibitors
GB9310092D0 (en) * 1993-05-17 1993-06-30 Fujisawa Pharmaceutical Co Indole derivatives
GB9317096D0 (en) * 1993-08-17 1993-09-29 Pfizer Ltd Indoles
ES2160158T3 (en) * 1994-03-30 2001-11-01 Zeria Pharm Co Ltd DERIVATIVES OF 4-INDOL-1-IL BUTIRIC ACID, ITS PREPARATION AND ITS USE AS INHIBITORS OF ALFA1-ADRENERGIC RECEPTORS AND TESTOSTERONE 5ALFA-REDUCTASAS.
GB9409583D0 (en) * 1994-05-13 1994-07-06 Pfizer Ltd Indoles
US5543417A (en) * 1994-10-21 1996-08-06 Merck & Co., Inc. Combination method of treating acne using 4-AZA-5α-cholestan-ones and 4-AZA-5α-androstan-ones as selective 5α-reductase inhibitors with anti-bacterial, keratolytic, or anti-inflammatory agents
US6670398B2 (en) 1997-05-14 2003-12-30 Atherogenics, Inc. Compounds and methods for treating transplant rejection
EP0994853B1 (en) 1997-05-14 2005-04-27 Atherogenics, Inc. A monoether of probucol and methods for the inhibition of the expression of vcam-1
US7417063B2 (en) 2004-04-13 2008-08-26 Bristol-Myers Squibb Company Bicyclic heterocycles useful as serine protease inhibitors
FR2893615B1 (en) * 2005-11-18 2008-03-07 Sanofi Aventis Sa 3-ACYLINDOLE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
PE20090159A1 (en) 2007-03-08 2009-02-21 Plexxikon Inc INDOL-PROPIONIC ACID DERIVED COMPOUNDS AS PPARs MODULATORS
US8252840B2 (en) 2007-03-26 2012-08-28 Salutria Pharmaceuticals Llc Methods of derivatives of probucol for the treatment of type II diabetes
US10703969B2 (en) * 2016-09-27 2020-07-07 Kaohsiung Medical University Detection method for quaternary ammonium compound having γ-carboxyl group

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9011335D0 (en) * 1990-05-21 1990-07-11 Fujisawa Pharmaceutical Co Indolebutyric acid derivatives and process for preparation thereof
WO1993005020A1 (en) * 1991-09-06 1993-03-18 Merck & Co., Inc. Indoles as inhibitors of hiv reverse transcriptase

Also Published As

Publication number Publication date
NO940237D0 (en) 1994-01-24
GB9115951D0 (en) 1991-09-11
TW223060B (en) 1994-05-01
JPH06511483A (en) 1994-12-22
ZA925546B (en) 1994-01-24
EP0598754A1 (en) 1994-06-01
AU2327192A (en) 1993-02-23
IL102544A0 (en) 1993-01-14
WO1993002051A1 (en) 1993-02-04
NO940237L (en) 1994-01-24
AU655662B2 (en) 1995-01-05
FI940311A0 (en) 1994-01-21
NZ243687A (en) 1994-12-22
FI940310A0 (en) 1994-01-21
SK8494A3 (en) 1994-11-09
CA2112678A1 (en) 1993-02-04
HU9400199D0 (en) 1994-05-30
PT100718A (en) 1993-08-31
CZ13694A3 (en) 1994-07-13
JPH06509336A (en) 1994-10-20
CA2112689A1 (en) 1993-02-04
FI940310A (en) 1994-01-21
CN1068816A (en) 1993-02-10
WO1993002050A1 (en) 1993-02-04
IE922387A1 (en) 1993-01-27
ZA925547B (en) 1994-01-24
PT100717A (en) 1993-08-31
IL102545A0 (en) 1993-01-14
CN1068817A (en) 1993-02-10
IE922386A1 (en) 1993-01-27
AU2327092A (en) 1993-02-23
FI940311A (en) 1994-01-21
EP0598750A1 (en) 1994-06-01
BR9206306A (en) 1994-11-08

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