ECSP951529A - PHARMACEUTICAL COMPOUNDS - Google Patents
PHARMACEUTICAL COMPOUNDSInfo
- Publication number
- ECSP951529A ECSP951529A ECSP951529A ECSP951529A EC SP951529 A ECSP951529 A EC SP951529A EC SP951529 A ECSP951529 A EC SP951529A EC SP951529 A ECSP951529 A EC SP951529A
- Authority
- EC
- Ecuador
- Prior art keywords
- optionally substituted
- alkyl
- phenyl
- hydrogen
- naphthyl
- Prior art date
Links
Abstract
Un compuesto de la fórmula: en la cual R1 y R7 son cada uno halo, trifluorometilo, alquilo C1-6, alcoxi C1-6, fenilo opcionalmente sustituido, naftilo opcionalmente sustituido o heteroarilo opcionalmente sustituido, R2 y R3 son cada uno hidrógeno o alquilo C1-6, R4 y R5 son cada uno hidrógeno, halo, trifluorometilo, alquilo C1-6, alcoxi C1-6, fenilo opcionalmente sustituido, naftilo opcionalmente sustituido o heteroarilo opcionalmente sustituido, R6 es hidrógeno, alquilo C1-6, fenilo opcionalmente sustituido, naftilo opcionalmente sustituido, heteroarilo opcionalmente sustituido, fenilo C1-6 alquilo opcionalmente sustituido o -CO2R8 donde R8 es un grupo éster, m y p son cada uno 0,1,2,3, o 4, n es 1,2,3 o 4; Z es Donde R9 y R10 son cada uno hidrógeno, alquilo C1-6 o fenilo C1-6 alquilo opcionalmente sustituido, X es oxígeno o azufre y Y es Donde R11 y R12 son cada uno hidrógeno, alquilo C1-6, trifluorometilo, fenilo opcionalmente sustituido, naftilo opcionalmente sustituido o heteroarilo opcionalmente sustituido; y sales y solvatos de los mismos.A compound of the formula: in which R1 and R7 are each halo, trifluoromethyl, C1-6 alkyl, C1-6 alkoxy, optionally substituted phenyl, optionally substituted naphthyl or optionally substituted heteroaryl, R2 and R3 are each hydrogen or alkyl C1-6, R4 and R5 are each hydrogen, halo, trifluoromethyl, C1-6 alkyl, C1-6 alkoxy, optionally substituted phenyl, optionally substituted naphthyl or optionally substituted heteroaryl, R6 is hydrogen, C1-6 alkyl, optionally substituted phenyl , optionally substituted naphthyl, optionally substituted heteroaryl, C1-6 phenyl optionally substituted alkyl or -CO2R8 where R8 is an ester group, m and p are each 0,1,2,3, or 4, n is 1,2,3 or 4 ; Z is Where R9 and R10 are each hydrogen, optionally substituted C1-6 alkyl or phenyl C1-6 alkyl, X is oxygen or sulfur and Y is Where R11 and R12 are each hydrogen, optionally C1-6 alkyl, trifluoromethyl, phenyl substituted, optionally substituted naphthyl or optionally substituted heteroaryl; and salts and solvates thereof.
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ECSP951529 ECSP951529A (en) | 1995-09-05 | 1995-09-05 | PHARMACEUTICAL COMPOUNDS |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ECSP951529 ECSP951529A (en) | 1995-09-05 | 1995-09-05 | PHARMACEUTICAL COMPOUNDS |
Publications (1)
Publication Number | Publication Date |
---|---|
ECSP951529A true ECSP951529A (en) | 1997-05-16 |
Family
ID=42042171
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ECSP951529 ECSP951529A (en) | 1995-09-05 | 1995-09-05 | PHARMACEUTICAL COMPOUNDS |
Country Status (1)
Country | Link |
---|---|
EC (1) | ECSP951529A (en) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US11130755B2 (en) | 2016-11-07 | 2021-09-28 | Sanofi | Substituted pyrido[3,4-b]indoles for the treatment of cartilage disorders |
-
1995
- 1995-09-05 EC ECSP951529 patent/ECSP951529A/en unknown
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US11130755B2 (en) | 2016-11-07 | 2021-09-28 | Sanofi | Substituted pyrido[3,4-b]indoles for the treatment of cartilage disorders |
US11827633B2 (en) | 2016-11-07 | 2023-11-28 | Sanofi | Substituted pyrido[3,4-b]indoles for the treatment of cartilage disorders |
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