ECSP15032906A - PHARMACEUTICAL COMPOSITION INCLUDING DROSPIRENONE AND CONTRACEPTIVE KIT (DIVISIONAL 2 APPLICATION No. SP-12-12359 PCT) - Google Patents
PHARMACEUTICAL COMPOSITION INCLUDING DROSPIRENONE AND CONTRACEPTIVE KIT (DIVISIONAL 2 APPLICATION No. SP-12-12359 PCT)Info
- Publication number
- ECSP15032906A ECSP15032906A ECIEPI201532906A ECPI201532906A ECSP15032906A EC SP15032906 A ECSP15032906 A EC SP15032906A EC IEPI201532906 A ECIEPI201532906 A EC IEPI201532906A EC PI201532906 A ECPI201532906 A EC PI201532906A EC SP15032906 A ECSP15032906 A EC SP15032906A
- Authority
- EC
- Ecuador
- Prior art keywords
- pharmaceutical composition
- divisional
- pct
- application
- drospirenone
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
- A61K31/585—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin containing lactone rings, e.g. oxandrolone, bufalin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Medicinal Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
La presente invención se refiere al campo de las composiciones farmacéuticas y métodos anticonceptivos. La presente invención proporciona una composición farmacéutica que comprende drospirenona caracterizada por una velocidad de disolución lenta de la drospirenona in vitro y un perfil farmacocinético mejorado. Está asimismo prevista la utilización de dicha composición en los métodos anticonceptivos y en los kits.The present invention relates to the field of pharmaceutical compositions and contraceptive methods. The present invention provides a pharmaceutical composition comprising drospirenone characterized by a slow dissolution rate of drospirenone in vitro and an improved pharmacokinetic profile. The use of said composition in contraceptive methods and kits is also planned.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP10305708 | 2010-06-29 | ||
US36839610P | 2010-07-28 | 2010-07-28 | |
PCT/EP2011/060795 WO2012000981A1 (en) | 2010-06-29 | 2011-06-28 | Pharmaceutical composition comprising drospirenone and contraceptive kit |
Publications (1)
Publication Number | Publication Date |
---|---|
ECSP15032906A true ECSP15032906A (en) | 2016-01-29 |
Family
ID=48802149
Family Applications (3)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ECSP12012359 ECSP12012359A (en) | 2010-06-29 | 2012-10-27 | PHARMACEUTICAL COMPOSITION INCLUDING DROSPIRENONE AND ANTI-CONCEPTIVE KIT |
ECIEPI201532906A ECSP15032906A (en) | 2010-06-29 | 2015-07-28 | PHARMACEUTICAL COMPOSITION INCLUDING DROSPIRENONE AND CONTRACEPTIVE KIT (DIVISIONAL 2 APPLICATION No. SP-12-12359 PCT) |
ECIEPI201532911A ECSP15032911A (en) | 2010-06-29 | 2015-07-28 | PHARMACEUTICAL COMPOSITION INCLUDING DROSPIRENONE AND CONTRACEPTIVE KIT (DIVISIONAL 1 APPLICATION No. SP-12-12359 PCT) |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ECSP12012359 ECSP12012359A (en) | 2010-06-29 | 2012-10-27 | PHARMACEUTICAL COMPOSITION INCLUDING DROSPIRENONE AND ANTI-CONCEPTIVE KIT |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ECIEPI201532911A ECSP15032911A (en) | 2010-06-29 | 2015-07-28 | PHARMACEUTICAL COMPOSITION INCLUDING DROSPIRENONE AND CONTRACEPTIVE KIT (DIVISIONAL 1 APPLICATION No. SP-12-12359 PCT) |
Country Status (14)
Country | Link |
---|---|
KR (1) | KR102210982B1 (en) |
BR (1) | BR122019008317A2 (en) |
CL (1) | CL2012003685A1 (en) |
CO (1) | CO6640328A2 (en) |
DK (1) | DK2588114T3 (en) |
EC (3) | ECSP12012359A (en) |
ES (1) | ES2777886T3 (en) |
GT (3) | GT201200336BA (en) |
HR (1) | HRP20200155T1 (en) |
HU (1) | HUE047689T2 (en) |
LT (2) | LT2588114T (en) |
MX (3) | MX364971B (en) |
PT (1) | PT2588114T (en) |
ZA (1) | ZA201209743B (en) |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2009138224A1 (en) * | 2008-05-14 | 2009-11-19 | Helm Ag | Pharmaceutical composition comprising drospirenone |
-
2011
- 2011-06-28 BR BR122019008317-7A patent/BR122019008317A2/en not_active Application Discontinuation
- 2011-06-28 MX MX2015008884A patent/MX364971B/en unknown
- 2011-06-28 DK DK11727985.1T patent/DK2588114T3/en active
- 2011-06-28 PT PT117279851T patent/PT2588114T/en unknown
- 2011-06-28 MX MX2012014629A patent/MX339952B/en active IP Right Grant
- 2011-06-28 LT LTEP11727985.1T patent/LT2588114T/en unknown
- 2011-06-28 HU HUE11727985A patent/HUE047689T2/en unknown
- 2011-06-28 ES ES11727985T patent/ES2777886T3/en active Active
- 2011-06-28 KR KR1020197017379A patent/KR102210982B1/en active IP Right Grant
-
2012
- 2012-10-27 EC ECSP12012359 patent/ECSP12012359A/en unknown
- 2012-12-12 GT GT201200336BL patent/GT201200336BA/en unknown
- 2012-12-12 GT GT201200336A patent/GT201200336A/en unknown
- 2012-12-12 GT GT201200336AK patent/GT201200336AA/en unknown
- 2012-12-13 MX MX2019004393A patent/MX2019004393A/en unknown
- 2012-12-21 ZA ZA2012/09743A patent/ZA201209743B/en unknown
- 2012-12-26 CL CL2012003685A patent/CL2012003685A1/en unknown
- 2012-12-28 CO CO12235600A patent/CO6640328A2/en not_active Application Discontinuation
-
2015
- 2015-07-28 EC ECIEPI201532906A patent/ECSP15032906A/en unknown
- 2015-07-28 EC ECIEPI201532911A patent/ECSP15032911A/en unknown
-
2020
- 2020-01-30 HR HRP20200155TT patent/HRP20200155T1/en unknown
-
2021
- 2021-10-14 LT LTPA2021523C patent/LTPA2021523I1/lt unknown
Also Published As
Publication number | Publication date |
---|---|
ZA201209743B (en) | 2014-03-26 |
ES2777886T3 (en) | 2020-08-06 |
CO6640328A2 (en) | 2013-03-22 |
CL2012003685A1 (en) | 2013-07-05 |
BR122019008317A2 (en) | 2020-09-29 |
LT2588114T (en) | 2020-02-25 |
MX364971B (en) | 2019-05-16 |
GT201200336A (en) | 2014-01-14 |
GT201200336AA (en) | 2017-10-23 |
HUE047689T2 (en) | 2020-05-28 |
HRP20200155T1 (en) | 2020-05-01 |
KR102210982B1 (en) | 2021-02-02 |
MX2019004393A (en) | 2019-09-09 |
DK2588114T3 (en) | 2020-02-17 |
KR20190073598A (en) | 2019-06-26 |
LTPA2021523I1 (en) | 2021-11-10 |
ECSP15032911A (en) | 2016-01-29 |
PT2588114T (en) | 2020-02-20 |
MX2012014629A (en) | 2013-05-06 |
MX339952B (en) | 2016-06-20 |
ECSP12012359A (en) | 2013-03-28 |
GT201200336BA (en) | 2017-10-23 |
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