CO6640328A2 - Pharmaceutical composition comprising drospirenone and contraceptive kit - Google Patents
Pharmaceutical composition comprising drospirenone and contraceptive kitInfo
- Publication number
- CO6640328A2 CO6640328A2 CO12235600A CO12235600A CO6640328A2 CO 6640328 A2 CO6640328 A2 CO 6640328A2 CO 12235600 A CO12235600 A CO 12235600A CO 12235600 A CO12235600 A CO 12235600A CO 6640328 A2 CO6640328 A2 CO 6640328A2
- Authority
- CO
- Colombia
- Prior art keywords
- drospirenone
- pharmaceutical composition
- contraceptive kit
- present
- contraceptive
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
- A61K31/585—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin containing lactone rings, e.g. oxandrolone, bufalin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Molecular Biology (AREA)
- Biophysics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
La presente invención se refiere al campo de las composiciones farmacéuticas y métodos anticonceptivos. La presente invención proporciona una composición farmacéutica que comprende drospirenona caracterizada por una velocidad de disolución lenta de la drospirenona in vitro y un perfil farmacocinético mejorado. Está asimismo prevista la utilización de dicha composición en los métodos anticonceptivos y en los kits.The present invention relates to the field of pharmaceutical compositions and contraceptive methods. The present invention provides a pharmaceutical composition comprising drospirenone characterized by a slow dissolution rate of drospirenone in vitro and an improved pharmacokinetic profile. It is also planned to use said composition in contraceptive methods and in kits.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP10305708 | 2010-06-29 | ||
US36839610P | 2010-07-28 | 2010-07-28 |
Publications (1)
Publication Number | Publication Date |
---|---|
CO6640328A2 true CO6640328A2 (en) | 2013-03-22 |
Family
ID=48802149
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CO12235600A CO6640328A2 (en) | 2010-06-29 | 2012-12-28 | Pharmaceutical composition comprising drospirenone and contraceptive kit |
Country Status (14)
Country | Link |
---|---|
KR (1) | KR102210982B1 (en) |
BR (1) | BR122019008317A2 (en) |
CL (1) | CL2012003685A1 (en) |
CO (1) | CO6640328A2 (en) |
DK (1) | DK2588114T3 (en) |
EC (3) | ECSP12012359A (en) |
ES (1) | ES2777886T3 (en) |
GT (3) | GT201200336A (en) |
HR (1) | HRP20200155T1 (en) |
HU (1) | HUE047689T2 (en) |
LT (2) | LT2588114T (en) |
MX (3) | MX339952B (en) |
PT (1) | PT2588114T (en) |
ZA (1) | ZA201209743B (en) |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2009138224A1 (en) * | 2008-05-14 | 2009-11-19 | Helm Ag | Pharmaceutical composition comprising drospirenone |
-
2011
- 2011-06-28 MX MX2012014629A patent/MX339952B/en active IP Right Grant
- 2011-06-28 DK DK11727985.1T patent/DK2588114T3/en active
- 2011-06-28 ES ES11727985T patent/ES2777886T3/en active Active
- 2011-06-28 PT PT117279851T patent/PT2588114T/en unknown
- 2011-06-28 BR BR122019008317-7A patent/BR122019008317A2/en not_active Application Discontinuation
- 2011-06-28 LT LTEP11727985.1T patent/LT2588114T/en unknown
- 2011-06-28 HU HUE11727985A patent/HUE047689T2/en unknown
- 2011-06-28 MX MX2015008884A patent/MX364971B/en unknown
- 2011-06-28 KR KR1020197017379A patent/KR102210982B1/en active IP Right Grant
-
2012
- 2012-10-27 EC ECSP12012359 patent/ECSP12012359A/en unknown
- 2012-12-12 GT GT201200336A patent/GT201200336A/en unknown
- 2012-12-12 GT GT201200336BL patent/GT201200336BA/en unknown
- 2012-12-12 GT GT201200336AK patent/GT201200336AA/en unknown
- 2012-12-13 MX MX2019004393A patent/MX2019004393A/en unknown
- 2012-12-21 ZA ZA2012/09743A patent/ZA201209743B/en unknown
- 2012-12-26 CL CL2012003685A patent/CL2012003685A1/en unknown
- 2012-12-28 CO CO12235600A patent/CO6640328A2/en not_active Application Discontinuation
-
2015
- 2015-07-28 EC ECIEPI201532906A patent/ECSP15032906A/en unknown
- 2015-07-28 EC ECIEPI201532911A patent/ECSP15032911A/en unknown
-
2020
- 2020-01-30 HR HRP20200155TT patent/HRP20200155T1/en unknown
-
2021
- 2021-10-14 LT LTPA2021523C patent/LTPA2021523I1/lt unknown
Also Published As
Publication number | Publication date |
---|---|
ES2777886T3 (en) | 2020-08-06 |
HRP20200155T1 (en) | 2020-05-01 |
ECSP15032906A (en) | 2016-01-29 |
KR102210982B1 (en) | 2021-02-02 |
MX339952B (en) | 2016-06-20 |
HUE047689T2 (en) | 2020-05-28 |
PT2588114T (en) | 2020-02-20 |
KR20190073598A (en) | 2019-06-26 |
ZA201209743B (en) | 2014-03-26 |
GT201200336BA (en) | 2017-10-23 |
DK2588114T3 (en) | 2020-02-17 |
GT201200336AA (en) | 2017-10-23 |
GT201200336A (en) | 2014-01-14 |
BR122019008317A2 (en) | 2020-09-29 |
MX2019004393A (en) | 2019-09-09 |
MX2012014629A (en) | 2013-05-06 |
CL2012003685A1 (en) | 2013-07-05 |
MX364971B (en) | 2019-05-16 |
ECSP15032911A (en) | 2016-01-29 |
LT2588114T (en) | 2020-02-25 |
LTPA2021523I1 (en) | 2021-11-10 |
ECSP12012359A (en) | 2013-03-28 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FC | Application refused |