ECSP066441A - ?15-d-homoesteroides que tienen un efecto androgénico - Google Patents

?15-d-homoesteroides que tienen un efecto androgénico

Info

Publication number
ECSP066441A
ECSP066441A EC2006006441A ECSP066441A ECSP066441A EC SP066441 A ECSP066441 A EC SP066441A EC 2006006441 A EC2006006441 A EC 2006006441A EC SP066441 A ECSP066441 A EC SP066441A EC SP066441 A ECSP066441 A EC SP066441A
Authority
EC
Ecuador
Prior art keywords
homosteroids
androgenic effect
compounds
general formula
androgenic
Prior art date
Application number
EC2006006441A
Other languages
English (en)
Inventor
Ralf Wyrwa
Sven Ring
Guenter Kaufmann
Walter Elger
Birgitt Schneider
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE10339532A external-priority patent/DE10339532A1/de
Application filed by Schering Ag filed Critical Schering Ag
Publication of ECSP066441A publication Critical patent/ECSP066441A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J63/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by expansion of only one ring by one or two atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/26—Androgens
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/30—Oestrogens
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J75/00—Processes for the preparation of steroids in general

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Reproductive Health (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pregnancy & Childbirth (AREA)
  • Epidemiology (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La invención se relaciona con ?15-D-homoesteroides de la fórmula general (I), con métodos para producirlos y con composiciones farmacéuticas que contienen dichos compuestos. Se proporcionan compuestos de la fórmula general (I) de la invención con actividad androgénica.
EC2006006441A 2003-08-21 2006-03-20 ?15-d-homoesteroides que tienen un efecto androgénico ECSP066441A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US49666903P 2003-08-21 2003-08-21
DE10339532A DE10339532A1 (de) 2003-08-21 2003-08-21 Delta 15-D-Homosteroide mit androgener Wirkung

Publications (1)

Publication Number Publication Date
ECSP066441A true ECSP066441A (es) 2006-09-18

Family

ID=34276519

Family Applications (1)

Application Number Title Priority Date Filing Date
EC2006006441A ECSP066441A (es) 2003-08-21 2006-03-20 ?15-d-homoesteroides que tienen un efecto androgénico

Country Status (11)

Country Link
US (1) US7388003B2 (es)
EP (1) EP1658306A1 (es)
JP (1) JP2007502801A (es)
KR (1) KR20060091295A (es)
AU (1) AU2004268040A1 (es)
BR (1) BRPI0413787A (es)
CA (1) CA2534831A1 (es)
EC (1) ECSP066441A (es)
IL (1) IL173608A0 (es)
MX (1) MXPA06002034A (es)
WO (1) WO2005021573A1 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW200745156A (en) * 2005-06-17 2007-12-16 Organon Nv Steroids having a mixed androgenic and progestagenic profile

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1054262A (es) *
IL50854A (en) * 1975-11-11 1979-12-30 Sparamedica Ag D-homosteroids their manufacture and pharmaceutical compositions containing them
IL51468A (en) * 1976-02-23 1981-01-30 Sparamedica Ag 17 -hydroxy- -d-homosteroid derivatives,their preparation and pharmaceutical compositions containing them
NL7703448A (nl) * 1976-04-13 1977-10-17 Hoffmann La Roche Nieuwe d-homosteroiden.
DE10247399A1 (de) * 2002-10-08 2004-04-29 Schering Ag Pharmazeutische Zubereitungen, Verwendung dieser Zubereitung und Verfahren zur Erhöhung der Bioverfügbarkeit von peroral zu applizierenden Arzneistoffen

Also Published As

Publication number Publication date
CA2534831A1 (en) 2005-03-10
JP2007502801A (ja) 2007-02-15
AU2004268040A1 (en) 2005-03-10
MXPA06002034A (es) 2006-05-17
EP1658306A1 (de) 2006-05-24
US20050131076A1 (en) 2005-06-16
US7388003B2 (en) 2008-06-17
WO2005021573A1 (de) 2005-03-10
BRPI0413787A (pt) 2006-11-07
KR20060091295A (ko) 2006-08-18
IL173608A0 (en) 2006-07-05

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