EA201991008A1 - NEW DERIVATIVES OF NAFTIRIDINONE AND THEIR APPLICATION IN TREATMENT OF ARRHYTHMIA - Google Patents

NEW DERIVATIVES OF NAFTIRIDINONE AND THEIR APPLICATION IN TREATMENT OF ARRHYTHMIA

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Publication number
EA201991008A1
EA201991008A1 EA201991008A EA201991008A EA201991008A1 EA 201991008 A1 EA201991008 A1 EA 201991008A1 EA 201991008 A EA201991008 A EA 201991008A EA 201991008 A EA201991008 A EA 201991008A EA 201991008 A1 EA201991008 A1 EA 201991008A1
Authority
EA
Eurasian Patent Office
Prior art keywords
naftiridinone
arrhythmia
treatment
application
new derivatives
Prior art date
Application number
EA201991008A
Other languages
Russian (ru)
Other versions
EA038455B1 (en
Inventor
Гийом Барб
Грегори Рэймонд Бебернитц
Сыцун Гэн
Хатидже Белгин Гулгезе Эффимиу
Лв Ляо
Фупэн Ма
Жовэй Мо
Дэвид Томас Паркер
Юньшань Пэн
Штефан Пойкерт
Кен Ямада
Кайо Ясосима
Original Assignee
Новартис Аг
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Новартис Аг filed Critical Новартис Аг
Priority claimed from PCT/IB2017/056515 external-priority patent/WO2018073788A1/en
Publication of EA201991008A1 publication Critical patent/EA201991008A1/en
Publication of EA038455B1 publication Critical patent/EA038455B1/en

Links

Abstract

Настоящее изобретение предусматривает соединение формулы (I) или его фармацевтически приемлемую соль:где R, R-R, Xи Xопределены в данном документе, способ получения соединений по настоящему изобретению и пути их терапевтического применения. В настоящем изобретении дополнительно предусмотрены комбинация фармакологически активных средств и фармацевтическая композиция.The present invention provides a compound of formula (I) or a pharmaceutically acceptable salt thereof: wherein R, R-R, X, and X are defined herein, a process for preparing the compounds of the present invention, and methods for their therapeutic use. The present invention further provides a combination of pharmacologically active agents and a pharmaceutical composition.

EA201991008A 2016-10-26 2017-10-19 Novel naphthyridinone derivatives and their use in the treatment of arrhythmia EA038455B1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201662413292P 2016-10-26 2016-10-26
PCT/IB2017/056515 WO2018073788A1 (en) 2016-10-21 2017-10-19 Naphthyridinone derivatives and their use in the treatment of arrhythmia

Publications (2)

Publication Number Publication Date
EA201991008A1 true EA201991008A1 (en) 2019-09-30
EA038455B1 EA038455B1 (en) 2021-08-31

Family

ID=68000223

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201991008A EA038455B1 (en) 2016-10-26 2017-10-19 Novel naphthyridinone derivatives and their use in the treatment of arrhythmia

Country Status (1)

Country Link
EA (1) EA038455B1 (en)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1432710A1 (en) * 2001-09-26 2004-06-30 Bayer Pharmaceuticals Corporation 1, 8-naphthyridine derivatives as antidiabetics
DK2254873T3 (en) * 2008-02-22 2014-06-30 Otsuka Pharma Co Ltd Benzodiazepine Compound and Pharmaceutical Composition.

Also Published As

Publication number Publication date
EA038455B1 (en) 2021-08-31

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