EA201692221A1 - Фармацевтическая композиция для профилактики и лечения заболеваний, связанных с повышенной активностью индуцируемой синтазы окиси азота - Google Patents
Фармацевтическая композиция для профилактики и лечения заболеваний, связанных с повышенной активностью индуцируемой синтазы окиси азотаInfo
- Publication number
- EA201692221A1 EA201692221A1 EA201692221A EA201692221A EA201692221A1 EA 201692221 A1 EA201692221 A1 EA 201692221A1 EA 201692221 A EA201692221 A EA 201692221A EA 201692221 A EA201692221 A EA 201692221A EA 201692221 A1 EA201692221 A1 EA 201692221A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- treatment
- prevention
- pharmaceutical composition
- nitrogen oxide
- increased activity
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/4015—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil having oxo groups directly attached to the heterocyclic ring, e.g. piracetam, ethosuximide
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyridine Compounds (AREA)
Abstract
Данное изобретение относится к новому медицинскому применению (4R)-2-(4-фенил-2-оксопирролидин-1-ил)ацетамида для лечения патологических состояний, характеризуемых повышенной экспрессией iNOS гена.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
LVP-14-39A LV15072B (lv) | 2014-05-14 | 2014-05-14 | Farmaceitiska kompozīcija izmantošanai patoloģiska stāvokļa, kam raksturīga paaugstināta iNOS gēna ekspresija, profilaksei un ārstēšanai |
PCT/IB2015/053554 WO2015173763A1 (en) | 2014-05-14 | 2015-05-14 | Pharmaceutical composition for the prevention and treatment of diseases associated with elevated inducible nitric oxide synthase |
Publications (2)
Publication Number | Publication Date |
---|---|
EA201692221A1 true EA201692221A1 (ru) | 2017-05-31 |
EA030563B1 EA030563B1 (ru) | 2018-08-31 |
Family
ID=53716523
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA201692221A EA030563B1 (ru) | 2014-05-14 | 2015-05-14 | Фармацевтическая композиция для профилактики и лечения периферической невропатии |
Country Status (7)
Country | Link |
---|---|
US (1) | US20180064687A1 (ru) |
EP (1) | EP3142662B1 (ru) |
EA (1) | EA030563B1 (ru) |
GE (1) | GEP20186888B (ru) |
LV (1) | LV15072B (ru) |
UA (1) | UA115010C2 (ru) |
WO (1) | WO2015173763A1 (ru) |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
LV13630B (en) | 2006-03-16 | 2007-12-20 | Olainfarm As | Method of preparation and use of pharmaceutically active n-carbamoylmethyl-4(r)-phenyl-2-pyrrolidinone |
TW201408294A (zh) * | 2012-07-05 | 2014-03-01 | Merz Pharma Gmbh & Co Kgaa | (r)-苯基披喇瑟盪於治療帕金森氏症之用除 |
-
2014
- 2014-05-14 LV LVP-14-39A patent/LV15072B/lv unknown
-
2015
- 2015-05-14 WO PCT/IB2015/053554 patent/WO2015173763A1/en active Application Filing
- 2015-05-14 EA EA201692221A patent/EA030563B1/ru not_active IP Right Cessation
- 2015-05-14 EP EP15739673.0A patent/EP3142662B1/en active Active
- 2015-05-14 US US15/309,527 patent/US20180064687A1/en not_active Abandoned
- 2015-05-14 GE GEAP201514335A patent/GEP20186888B/en unknown
- 2015-05-14 UA UAA201611303A patent/UA115010C2/uk unknown
Also Published As
Publication number | Publication date |
---|---|
LV15072A (lv) | 2015-11-20 |
UA115010C2 (uk) | 2017-08-28 |
EP3142662A1 (en) | 2017-03-22 |
WO2015173763A1 (en) | 2015-11-19 |
LV15072B (lv) | 2016-09-20 |
GEP20186888B (en) | 2018-08-27 |
EA030563B1 (ru) | 2018-08-31 |
US20180064687A1 (en) | 2018-03-08 |
EP3142662B1 (en) | 2020-07-08 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
IL255509B (en) | Compounds as modulators of ccr2, pharmaceutical preparations containing them and their use in the treatment of diseases | |
PH12017501306A1 (en) | Inhibitors of histone demethylases | |
PH12016501750A1 (en) | Human plasma kallikrein inhibitors | |
EA201791874A1 (ru) | Фторированные ингибиторы лизилоксидазоподобного фермента-2 и их применение | |
EA201691481A1 (ru) | ИНГИБИТОРЫ C5a ДЛЯ ЛЕЧЕНИЯ ВИРУСНОЙ ПНЕВМОНИИ | |
EA201691447A1 (ru) | 2-амино-3,5,5-трифтор-3,4,5,6-тетрагидропиридины в качестве ингибиторов bace1 для лечения болезни альцгеймера | |
PH12017500401A1 (en) | Therapeutic compounds as inhibitors of the orexin-1 receptor | |
NZ732511A (en) | Small molecule inhibitors of egfr and pi3k | |
MY197440A (en) | Heteroamatic compounds as btk inhibitors | |
GEP20237457B (en) | Nucleotide hemi-sulfate salt for treatment of hepatitis c virus | |
MX2017009417A (es) | Formas solidas de acido 2-(5-(3-fluorofenil)-3-hidroxipicolinamido )acetico, composiciones y usos de las mismas. | |
MY174747A (en) | Bace1 inhibitors | |
EA201690039A1 (ru) | Ингибиторы rorc2 и способы их применения | |
ZA201707951B (en) | Amide compound and use thereof as agent for the treatment and prevention of diseases caused by rna- and/or dna-containing viruses, and concomitant diseases | |
EA201792571A1 (ru) | Терапевтическое применение l-4-хлорокинуренина | |
MX2019006863A (es) | Inhibidores de heparanasa y uso de los mismos. | |
EA201692111A1 (ru) | Фармацевтические композиции, содержащие данириксин, для лечения инфекционных заболеваний | |
CL2017002229A1 (es) | Inhibidores de bace1. | |
MD20180049A2 (ru) | Фармацевтическая композиция | |
MX2016013588A (es) | Complejo de tanato de sitagliptina. | |
MX2018006631A (es) | Compuesto para uso en la prevencion y tratamiento de enfermedades neurodegenerativas. | |
EA201501130A1 (ru) | Офтальмологическая фармацевтическая композиция | |
EA201790020A1 (ru) | Соединения, фармацевтические композиции и их применение при лечении нейродегенеративных заболеваний | |
EA201692221A1 (ru) | Фармацевтическая композиция для профилактики и лечения заболеваний, связанных с повышенной активностью индуцируемой синтазы окиси азота | |
KR20180085033A (ko) | 피부 질환 치료용 약학적 제형 및 이의 제조 방법 |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): AM AZ BY KZ KG TJ TM RU |