EA201201655A1 - ANTI-TUMOR MEDICINE (OPTIONS) - Google Patents

ANTI-TUMOR MEDICINE (OPTIONS)

Info

Publication number
EA201201655A1
EA201201655A1 EA201201655A EA201201655A EA201201655A1 EA 201201655 A1 EA201201655 A1 EA 201201655A1 EA 201201655 A EA201201655 A EA 201201655A EA 201201655 A EA201201655 A EA 201201655A EA 201201655 A1 EA201201655 A1 EA 201201655A1
Authority
EA
Eurasian Patent Office
Prior art keywords
bortezomib
creation
isotopes
minerals
antitumor agent
Prior art date
Application number
EA201201655A
Other languages
Russian (ru)
Inventor
Анастасия Геннадьевна ЧЕЛЯЕВА
Владимир Павлович ЛОБКО
Original Assignee
Ооо "Эн.Си.Фарм"
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ооо "Эн.Си.Фарм" filed Critical Ооо "Эн.Си.Фарм"
Priority to EA201201655A priority Critical patent/EA201201655A1/en
Publication of EA201201655A1 publication Critical patent/EA201201655A1/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Изобретение относится к области фармацевтической промышленности и медицине и может быть использовано при создании и применении противоопухолевых средств, в частности ингибиторов протеасом на основе бортезомиба. Задачей настоящего изобретения является создание эффективного противоопухолевого средства на базе бортезомиба с расширенными свойствами при использовании. Задача решается за счет того, что противоопухолевое средство содержит бортезомиб, минеральные вещества калий, цинк, изотопы углеродаС, изотопы азотаN. Техническими результатами изобретения являются увеличение лечебного эффекта без увеличения концентрации бортезомиба при лечении злокачественных опухолей за счет использования в противоопухолевом средстве изотоповС,N и минеральных веществ; увеличение времени хранения, в том числе в готовом к применению жидком виде.The invention relates to the pharmaceutical industry and medicine and can be used in the creation and application of anticancer drugs, in particular bortezomiba-based proteasome inhibitors. The present invention is the creation of an effective anticancer agent on the basis of bortezomib with enhanced properties during use. The problem is solved due to the fact that the antitumor agent contains bortezomib, minerals potassium, zinc, carbon isotopes, carbon isotopes of nitrogenN. Technical results of the invention are to increase the therapeutic effect without increasing the concentration of bortezomib in the treatment of malignant tumors due to the use in the antitumor agent isotopes C, N and minerals; increase storage time, including in ready-to-use liquid form.

EA201201655A 2012-12-28 2012-12-28 ANTI-TUMOR MEDICINE (OPTIONS) EA201201655A1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
EA201201655A EA201201655A1 (en) 2012-12-28 2012-12-28 ANTI-TUMOR MEDICINE (OPTIONS)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EA201201655A EA201201655A1 (en) 2012-12-28 2012-12-28 ANTI-TUMOR MEDICINE (OPTIONS)

Publications (1)

Publication Number Publication Date
EA201201655A1 true EA201201655A1 (en) 2014-06-30

Family

ID=51013753

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201201655A EA201201655A1 (en) 2012-12-28 2012-12-28 ANTI-TUMOR MEDICINE (OPTIONS)

Country Status (1)

Country Link
EA (1) EA201201655A1 (en)

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