EA200501830A1 - NEW LINCOMYCIN DERIVATIVES WITH ANTIMICROBIAL ACTIVITY - Google Patents

NEW LINCOMYCIN DERIVATIVES WITH ANTIMICROBIAL ACTIVITY

Info

Publication number
EA200501830A1
EA200501830A1 EA200501830A EA200501830A EA200501830A1 EA 200501830 A1 EA200501830 A1 EA 200501830A1 EA 200501830 A EA200501830 A EA 200501830A EA 200501830 A EA200501830 A EA 200501830A EA 200501830 A1 EA200501830 A1 EA 200501830A1
Authority
EA
Eurasian Patent Office
Prior art keywords
new
lincomycin derivatives
antimicrobial activity
lincomycin
compounds
Prior art date
Application number
EA200501830A
Other languages
Russian (ru)
Inventor
Джейсон Густаф Льюис
Сампат-Кумар Анандан
Хардвин О` Доуд
Михаил Федорович Гордеев
Original Assignee
Викьюрон Фармасьютикалз, Инк.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US10/642,807 external-priority patent/US7164011B2/en
Priority claimed from US10/777,455 external-priority patent/US7199105B2/en
Application filed by Викьюрон Фармасьютикалз, Инк. filed Critical Викьюрон Фармасьютикалз, Инк.
Priority claimed from PCT/US2004/019689 external-priority patent/WO2005012320A2/en
Publication of EA200501830A1 publication Critical patent/EA200501830A1/en

Links

Abstract

Описаны новые производные линкомицина. Эти производные линкомицина проявляют антибактериальную активность. Соединения данного изобретения могут обладать усиленной активностью против бактерий, в том числе грамположительных организмов, и могут быть полезными антибактериальными агентами. Описаны также способы синтеза и применение этих соединений.New lincomycin derivatives have been described. These lincomycin derivatives exhibit antibacterial activity. The compounds of this invention may have enhanced activity against bacteria, including gram-positive organisms, and may be useful antibacterial agents. Methods for the synthesis and use of these compounds are also described.

EA200501830A 2003-06-17 2004-06-17 NEW LINCOMYCIN DERIVATIVES WITH ANTIMICROBIAL ACTIVITY EA200501830A1 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US47950203P 2003-06-17 2003-06-17
US47929603P 2003-06-17 2003-06-17
US10/642,807 US7164011B2 (en) 2002-08-15 2003-08-15 Lincomycin derivatives possessing antibacterial activity
US10/777,455 US7199105B2 (en) 2002-08-15 2004-02-11 Lincomycin derivatives possessing antibacterial activity
PCT/US2004/019689 WO2005012320A2 (en) 2003-06-17 2004-06-17 Novel lincomycin derivatives possessing antimicrobial activity

Publications (1)

Publication Number Publication Date
EA200501830A1 true EA200501830A1 (en) 2006-06-30

Family

ID=58707227

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200501830A EA200501830A1 (en) 2003-06-17 2004-06-17 NEW LINCOMYCIN DERIVATIVES WITH ANTIMICROBIAL ACTIVITY

Country Status (1)

Country Link
EA (1) EA200501830A1 (en)

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