DOP2003000789A - ANALOGS OF 2-QUINAZOLINA SUBSTITUTED-4-YLAMINA - Google Patents

ANALOGS OF 2-QUINAZOLINA SUBSTITUTED-4-YLAMINA

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Publication number
DOP2003000789A
DOP2003000789A DO2003000789A DO2003000789A DOP2003000789A DO P2003000789 A DOP2003000789 A DO P2003000789A DO 2003000789 A DO2003000789 A DO 2003000789A DO 2003000789 A DO2003000789 A DO 2003000789A DO P2003000789 A DOP2003000789 A DO P2003000789A
Authority
DO
Dominican Republic
Prior art keywords
substituted
ylamina
quinazolina
analogs
ligands
Prior art date
Application number
DO2003000789A
Other languages
Spanish (es)
Inventor
Rajagopal Bakthavatchalam
Charles A Blum
Harry Brielmann
Timothy M Caldwell
Stephane De Lombaert
Kevin J Hodgetts
Xiaozhang Zheng
Original Assignee
Neurogen Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Neurogen Corp filed Critical Neurogen Corp
Priority to DO2003000789A priority Critical patent/DOP2003000789A/en
Publication of DOP2003000789A publication Critical patent/DOP2003000789A/en

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Abstract

Certain 2-substituted quinazolin-4-ylamine analogues are provided. Such compounds are ligands that may be used to modulate specific receptor activity in vivo or in vitro, and are particularly useful in the treatment of conditions associated with pathological receptor activation in humans, domesticated companion animals and livestock animals. Pharmaceutical compositions and methods for using them to treat such disorders are provided, as are methods for using such ligands for receptor localization studies.Certain 2-substituted quinazolin-4-ylamine analogues are provided. Such compounds are ligands that may be used to modulate specific receptor activity in vivo or in vitro, and are particularly useful in the treatment of conditions associated with pathological receptor activation in humans, domesticated companion animals and livestock animals. Pharmaceutical compositions and methods for using them to treat such disorders are provided, as are methods for using such ligands for receptor localization studies.

DO2003000789A 2003-12-12 2003-12-12 ANALOGS OF 2-QUINAZOLINA SUBSTITUTED-4-YLAMINA DOP2003000789A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
DO2003000789A DOP2003000789A (en) 2003-12-12 2003-12-12 ANALOGS OF 2-QUINAZOLINA SUBSTITUTED-4-YLAMINA

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DO2003000789A DOP2003000789A (en) 2003-12-12 2003-12-12 ANALOGS OF 2-QUINAZOLINA SUBSTITUTED-4-YLAMINA

Publications (1)

Publication Number Publication Date
DOP2003000789A true DOP2003000789A (en) 2004-06-15

Family

ID=44261274

Family Applications (1)

Application Number Title Priority Date Filing Date
DO2003000789A DOP2003000789A (en) 2003-12-12 2003-12-12 ANALOGS OF 2-QUINAZOLINA SUBSTITUTED-4-YLAMINA

Country Status (1)

Country Link
DO (1) DOP2003000789A (en)

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