DK95489D0 - Anvendelse af quinolizin- og quinolizinonderivater til fremstilling af et laegemiddel - Google Patents

Anvendelse af quinolizin- og quinolizinonderivater til fremstilling af et laegemiddel

Info

Publication number
DK95489D0
DK95489D0 DK095489A DK95489A DK95489D0 DK 95489 D0 DK95489 D0 DK 95489D0 DK 095489 A DK095489 A DK 095489A DK 95489 A DK95489 A DK 95489A DK 95489 D0 DK95489 D0 DK 95489D0
Authority
DK
Denmark
Prior art keywords
quinolizin
medicine
derivatives
preparation
quinolizin derivatives
Prior art date
Application number
DK095489A
Other languages
English (en)
Other versions
DK95489A (da
Inventor
Maurice W Gittos
Original Assignee
Merrell Dow Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merrell Dow Pharma filed Critical Merrell Dow Pharma
Publication of DK95489D0 publication Critical patent/DK95489D0/da
Publication of DK95489A publication Critical patent/DK95489A/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/18Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DK095489A 1988-03-01 1989-02-28 Anvendelse af quinolizin- og quinolizinonderivater til fremstilling af et laegemiddel DK95489A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP88400482A EP0330788A1 (en) 1988-03-01 1988-03-01 Use of quinolizine and quinolizinone derivatives in the manufacture of medicaments for the treatment of cardiac arrhythmia

Publications (2)

Publication Number Publication Date
DK95489D0 true DK95489D0 (da) 1989-02-28
DK95489A DK95489A (da) 1989-09-02

Family

ID=8200359

Family Applications (1)

Application Number Title Priority Date Filing Date
DK095489A DK95489A (da) 1988-03-01 1989-02-28 Anvendelse af quinolizin- og quinolizinonderivater til fremstilling af et laegemiddel

Country Status (6)

Country Link
EP (2) EP0330788A1 (da)
JP (1) JPH01268634A (da)
KR (1) KR890014112A (da)
AU (1) AU3028589A (da)
DK (1) DK95489A (da)
ZA (1) ZA891366B (da)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0329932B1 (en) * 1988-02-23 1995-10-18 Merrell Pharmaceuticals Inc. Use of quinolizine and quinolizinone derivatives in the manufacture of medicaments
US4992446A (en) * 1989-09-05 1991-02-12 G. D. Searle & Co. Tricyclic quinolizine amides
EP0492020A1 (en) * 1990-12-21 1992-07-01 Merrell Dow Pharmaceuticals Inc. Use of certain esters of hexahydro-8-hydroxy-2,6-methano-2H-quinolizin-3(4H)-one and related compounds for treating cognitive disorders
EP0517984A1 (en) * 1991-06-11 1992-12-16 Merrell Dow Pharmaceuticals Inc. Derivatives of amide analogs of certain methano bridged quinolizines
US5955470A (en) * 1991-06-11 1999-09-21 Merrell Pharmaceuticals, Inc. Derivatives of amide analogs of certain methano bridged quinolizines
US20080275241A1 (en) * 2005-12-23 2008-11-06 Tarur Venkatasubramanian Radha Polymorphic Forms of Dolasetron Base and Processes of Preparing Dolasetron Base, Its Polymorphic Forms and Salt Thereof
WO2007081909A2 (en) * 2006-01-05 2007-07-19 Teva Gyogyszergyar Zartkoruen Mukodo Forms of dolasetron mesylate and processes for their preparation
CN102203089A (zh) 2008-09-05 2011-09-28 伊兰医药品公司 N-磺酰氨基多环吡唑基化合物
WO2011102388A1 (ja) * 2010-02-16 2011-08-25 株式会社エーピーアイ コーポレーション 1-アミノ-1-アルコキシカルボニル-2-ビニルシクロプロパンの製造方法
CN102180878B (zh) * 2010-07-02 2013-06-26 成都新恒创药业有限公司 一种多拉司琼异构体或其盐及其制备方法和其应用

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0220011A3 (en) * 1985-10-12 1990-01-03 Beecham Group Plc Use of azabicloalkylbenzamides in the treatment of gastrointestinal motility disorders, migraine, emesis, cluster headaches, trigeminal neuralgia and arrhythmia
ZA878096B (en) * 1986-11-03 1988-04-26 Merrell Dow Pharmaceuticals Inc. Esters of hexahydro-8-hydroxy-2,6-methano-2h-quinolizin-3(4h)-one and related compounds

Also Published As

Publication number Publication date
KR890014112A (ko) 1989-10-21
EP0330824A1 (en) 1989-09-06
ZA891366B (en) 1989-11-29
AU3028589A (en) 1989-09-07
JPH01268634A (ja) 1989-10-26
DK95489A (da) 1989-09-02
EP0330788A1 (en) 1989-09-06

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Legal Events

Date Code Title Description
AHB Application shelved due to non-payment