DK605489A - BETA-AMINO-BORONIC ACID DERIVATIVES, THEIR PREPARATION AND USE - Google Patents

BETA-AMINO-BORONIC ACID DERIVATIVES, THEIR PREPARATION AND USE Download PDF

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Publication number
DK605489A
DK605489A DK605489A DK605489A DK605489A DK 605489 A DK605489 A DK 605489A DK 605489 A DK605489 A DK 605489A DK 605489 A DK605489 A DK 605489A DK 605489 A DK605489 A DK 605489A
Authority
DK
Denmark
Prior art keywords
beta
amino
preparation
acid derivatives
boronic acid
Prior art date
Application number
DK605489A
Other languages
Danish (da)
Other versions
DK605489D0 (en
Inventor
Heinz-Werner Kleemann
Hansjoerg Urbach
Dieter Ruppert
Bernward Schoelkens
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of DK605489D0 publication Critical patent/DK605489D0/en
Publication of DK605489A publication Critical patent/DK605489A/en

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic System
    • C07F5/02—Boron compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic System
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N
DK605489A 1988-12-01 1989-11-30 BETA-AMINO-BORONIC ACID DERIVATIVES, THEIR PREPARATION AND USE DK605489A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE3840452A DE3840452A1 (en) 1988-12-01 1988-12-01 (BETA) -amino-boronic acid DERIVATIVES

Publications (2)

Publication Number Publication Date
DK605489D0 DK605489D0 (en) 1989-11-30
DK605489A true DK605489A (en) 1990-06-02

Family

ID=6368210

Family Applications (1)

Application Number Title Priority Date Filing Date
DK605489A DK605489A (en) 1988-12-01 1989-11-30 BETA-AMINO-BORONIC ACID DERIVATIVES, THEIR PREPARATION AND USE

Country Status (14)

Country Link
EP (1) EP0371467A3 (en)
JP (1) JPH02193997A (en)
KR (1) KR900009663A (en)
AU (1) AU616819B2 (en)
CA (1) CA2004303A1 (en)
DE (1) DE3840452A1 (en)
DK (1) DK605489A (en)
FI (1) FI895718A0 (en)
IL (1) IL92497A0 (en)
NO (1) NO894790L (en)
NZ (1) NZ231578A (en)
PH (1) PH26584A (en)
PT (1) PT92442A (en)
ZA (1) ZA899152B (en)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL90244A (en) * 1988-05-11 1993-05-13 Du Pont Merck Pharma Peptide-drug compositions, for buccal and nasal administration, containing :-aminoboronic acid derivatives
US4983589A (en) * 1989-12-14 1991-01-08 Chevron Research And Technology Company Fungicidal imidazole diphenylaliphaticboranes and derivatives thereof
GB9017694D0 (en) * 1990-08-13 1990-09-26 Sandoz Ltd Improvements in or relating to organic chemistry
GB9024775D0 (en) * 1990-11-14 1991-01-02 Axis Research Chemical compounds
US5554728A (en) * 1991-07-23 1996-09-10 Nexstar Pharmaceuticals, Inc. Lipid conjugates of therapeutic peptides and protease inhibitors
US6825169B1 (en) 1991-10-22 2004-11-30 Trustees Of Tufts College Inhibitors of dipeptidyl-aminopeptidase type IV
MXPA93002392A (en) 1992-03-11 2005-02-04 Narhex Ltd Amine derivatives of oxo- and hydroxy-substitued hydrocarbons.
US6071895A (en) * 1992-03-11 2000-06-06 Narhex Limited Polar-substituted hydrocarbons
US5888992A (en) * 1992-03-11 1999-03-30 Narhex Limited Polar substituted hydrocarbons
RU2126794C1 (en) * 1992-03-11 1999-02-27 Нархекс Лимитед Amino-derivatives of oxo- or hydroxy-substituted hydrazines, method of their synthesis and pharmaceutical compositions for inhibition of retrovirus protease
US5559256A (en) * 1992-07-20 1996-09-24 E. R. Squibb & Sons, Inc. Aminediol protease inhibitors
US5442100A (en) * 1992-08-14 1995-08-15 The Procter & Gamble Company β-aminoalkyl and β-N-peptidylaminoalkyl boronic acids
US5354491A (en) * 1992-08-14 1994-10-11 The Procter & Gamble Company Liquid detergent compositions containing protease and certain β-aminoalkylboronic acids and esters
EP0655068B1 (en) * 1992-08-14 1997-12-17 The Procter & Gamble Company Process for synthesizing a beta-aminoalkylboronic acid and ester thereof
TR28578A (en) * 1993-08-13 1996-11-04 Procter & Gamble Liquid detergent compositions containing protease and some of -aminoalkylboronic acid and esters.
IL110898A0 (en) * 1993-09-10 1994-11-28 Narhex Australia Pty Ltd Polar-substituted hydrocarbons
US5431842A (en) * 1993-11-05 1995-07-11 The Procter & Gamble Company Liquid detergents with ortho-substituted phenylboronic acids for inhibition of proteolytic enzyme
US5965532A (en) 1996-06-28 1999-10-12 Trustees Of Tufts College Multivalent compounds for crosslinking receptors and uses thereof
US6040145A (en) 1997-05-07 2000-03-21 Tufts University Potentiation of the immune response
US6100234A (en) 1997-05-07 2000-08-08 Tufts University Treatment of HIV
CN1163594C (en) 1997-09-29 2004-08-25 尖端医疗有限公司 stimulation of hematopoietic cells in vitro
TWI252107B (en) 1998-05-04 2006-04-01 Piint Therapeutics Inc Pharmaceutical compositions and kits for hematopoietic usage
US6890904B1 (en) 1999-05-25 2005-05-10 Point Therapeutics, Inc. Anti-tumor agents
US20150018311A1 (en) * 2012-01-09 2015-01-15 University of Tromsø Therapeutic boron-containing compounds

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4499082A (en) * 1983-12-05 1985-02-12 E. I. Du Pont De Nemours And Company α-Aminoboronic acid peptides
US4537773A (en) * 1983-12-05 1985-08-27 E. I. Du Pont De Nemours And Company α-Aminoboronic acid derivatives

Also Published As

Publication number Publication date
NZ231578A (en) 1992-02-25
AU616819B2 (en) 1991-11-07
EP0371467A2 (en) 1990-06-06
NO894790L (en) 1990-06-05
DE3840452A1 (en) 1990-06-07
ZA899152B (en) 1990-09-26
EP0371467A3 (en) 1991-04-03
IL92497A0 (en) 1990-08-31
FI895718A0 (en) 1989-11-29
NO894790D0 (en) 1989-11-30
DK605489D0 (en) 1989-11-30
JPH02193997A (en) 1990-07-31
PT92442A (en) 1990-06-29
PH26584A (en) 1992-08-19
AU4566589A (en) 1990-06-07
KR900009663A (en) 1990-07-05
CA2004303A1 (en) 1990-06-01

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