AU4566589A - Beta-amino-boronic acid derivatives - Google Patents

Beta-amino-boronic acid derivatives

Info

Publication number
AU4566589A
AU4566589A AU45665/89A AU4566589A AU4566589A AU 4566589 A AU4566589 A AU 4566589A AU 45665/89 A AU45665/89 A AU 45665/89A AU 4566589 A AU4566589 A AU 4566589A AU 4566589 A AU4566589 A AU 4566589A
Authority
AU
Australia
Prior art keywords
beta
amino
acid derivatives
boronic acid
boronic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU45665/89A
Other versions
AU616819B2 (en
Inventor
Heinz-Werner Kleemann
Dieter Ruppert
Bernward Scholkens
Hansjorg Urbach
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Hoechst AG
Original Assignee
Hoechst AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst AG filed Critical Hoechst AG
Publication of AU4566589A publication Critical patent/AU4566589A/en
Application granted granted Critical
Publication of AU616819B2 publication Critical patent/AU616819B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic System
    • C07F5/02—Boron compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic System
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N
AU45665/89A 1988-12-01 1989-11-30 Beta-amino-boronic acid derivatives Ceased AU616819B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE3840452 1988-12-01
DE3840452A DE3840452A1 (en) 1988-12-01 1988-12-01 (BETA) -amino-boronic acid DERIVATIVES

Publications (2)

Publication Number Publication Date
AU4566589A true AU4566589A (en) 1990-06-07
AU616819B2 AU616819B2 (en) 1991-11-07

Family

ID=6368210

Family Applications (1)

Application Number Title Priority Date Filing Date
AU45665/89A Ceased AU616819B2 (en) 1988-12-01 1989-11-30 Beta-amino-boronic acid derivatives

Country Status (14)

Country Link
EP (1) EP0371467A3 (en)
JP (1) JPH02193997A (en)
KR (1) KR900009663A (en)
AU (1) AU616819B2 (en)
CA (1) CA2004303A1 (en)
DE (1) DE3840452A1 (en)
DK (1) DK605489A (en)
FI (1) FI895718A0 (en)
IL (1) IL92497A0 (en)
NO (1) NO894790L (en)
NZ (1) NZ231578A (en)
PH (1) PH26584A (en)
PT (1) PT92442A (en)
ZA (1) ZA899152B (en)

Cited By (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU616968B2 (en) * 1988-05-11 1991-11-14 Du Pont Merck Pharmaceutical Company, The Peptide-drug compositions containing alpha-aminoboronic acid derivatives
AU635800B2 (en) * 1989-12-14 1993-04-01 Chevron Research And Technology Company Fungicidal imidazole diphenylaliphaticboranes
AU643312B2 (en) * 1990-08-13 1993-11-11 Novartis Ag Improvements in or relating to organic chemistry
WO1995007269A1 (en) * 1993-09-10 1995-03-16 Narhex Limited Polar-substituted hydrocarbons
US5679688A (en) * 1992-03-11 1997-10-21 Narhex Limited Quinaldoyl-amine derivatives of oxo-and hydroxy-substituted hydrocarbons
US5888992A (en) * 1992-03-11 1999-03-30 Narhex Limited Polar substituted hydrocarbons
US6071895A (en) * 1992-03-11 2000-06-06 Narhex Limited Polar-substituted hydrocarbons
US6258806B1 (en) 1992-03-11 2001-07-10 Narhex Limited Amine derivatives of oxo- and hydroxy- substituted hydrocarbons

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9024775D0 (en) * 1990-11-14 1991-01-02 Axis Research Chemical compounds
US5554728A (en) * 1991-07-23 1996-09-10 Nexstar Pharmaceuticals, Inc. Lipid conjugates of therapeutic peptides and protease inhibitors
US6825169B1 (en) 1991-10-22 2004-11-30 Trustees Of Tufts College Inhibitors of dipeptidyl-aminopeptidase type IV
US5559256A (en) * 1992-07-20 1996-09-24 E. R. Squibb & Sons, Inc. Aminediol protease inhibitors
US5442100A (en) * 1992-08-14 1995-08-15 The Procter & Gamble Company β-aminoalkyl and β-N-peptidylaminoalkyl boronic acids
US5354491A (en) * 1992-08-14 1994-10-11 The Procter & Gamble Company Liquid detergent compositions containing protease and certain β-aminoalkylboronic acids and esters
EP0655068B1 (en) * 1992-08-14 1997-12-17 The Procter & Gamble Company Process for synthesizing a beta-aminoalkylboronic acid and ester thereof
TR28578A (en) * 1993-08-13 1996-11-04 Procter & Gamble Liquid detergent compositions containing protease and some of -aminoalkylboronic acid and esters.
US5431842A (en) * 1993-11-05 1995-07-11 The Procter & Gamble Company Liquid detergents with ortho-substituted phenylboronic acids for inhibition of proteolytic enzyme
US5965532A (en) 1996-06-28 1999-10-12 Trustees Of Tufts College Multivalent compounds for crosslinking receptors and uses thereof
US6040145A (en) 1997-05-07 2000-03-21 Tufts University Potentiation of the immune response
US6100234A (en) 1997-05-07 2000-08-08 Tufts University Treatment of HIV
CN1163594C (en) 1997-09-29 2004-08-25 尖端医疗有限公司 stimulation of hematopoietic cells in vitro
TWI252107B (en) 1998-05-04 2006-04-01 Piint Therapeutics Inc Pharmaceutical compositions and kits for hematopoietic usage
US6890904B1 (en) 1999-05-25 2005-05-10 Point Therapeutics, Inc. Anti-tumor agents
US20150018311A1 (en) * 2012-01-09 2015-01-15 University of Tromsø Therapeutic boron-containing compounds

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4499082A (en) * 1983-12-05 1985-02-12 E. I. Du Pont De Nemours And Company α-Aminoboronic acid peptides
US4537773A (en) * 1983-12-05 1985-08-27 E. I. Du Pont De Nemours And Company α-Aminoboronic acid derivatives

Cited By (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU616968B2 (en) * 1988-05-11 1991-11-14 Du Pont Merck Pharmaceutical Company, The Peptide-drug compositions containing alpha-aminoboronic acid derivatives
AU635800B2 (en) * 1989-12-14 1993-04-01 Chevron Research And Technology Company Fungicidal imidazole diphenylaliphaticboranes
AU643312B2 (en) * 1990-08-13 1993-11-11 Novartis Ag Improvements in or relating to organic chemistry
US5679688A (en) * 1992-03-11 1997-10-21 Narhex Limited Quinaldoyl-amine derivatives of oxo-and hydroxy-substituted hydrocarbons
US5888992A (en) * 1992-03-11 1999-03-30 Narhex Limited Polar substituted hydrocarbons
US6071895A (en) * 1992-03-11 2000-06-06 Narhex Limited Polar-substituted hydrocarbons
US6258806B1 (en) 1992-03-11 2001-07-10 Narhex Limited Amine derivatives of oxo- and hydroxy- substituted hydrocarbons
WO1995007269A1 (en) * 1993-09-10 1995-03-16 Narhex Limited Polar-substituted hydrocarbons

Also Published As

Publication number Publication date
NZ231578A (en) 1992-02-25
AU616819B2 (en) 1991-11-07
EP0371467A2 (en) 1990-06-06
NO894790L (en) 1990-06-05
DE3840452A1 (en) 1990-06-07
ZA899152B (en) 1990-09-26
EP0371467A3 (en) 1991-04-03
IL92497A0 (en) 1990-08-31
FI895718A0 (en) 1989-11-29
NO894790D0 (en) 1989-11-30
DK605489D0 (en) 1989-11-30
JPH02193997A (en) 1990-07-31
PT92442A (en) 1990-06-29
PH26584A (en) 1992-08-19
KR900009663A (en) 1990-07-05
DK605489A (en) 1990-06-02
CA2004303A1 (en) 1990-06-01

Similar Documents

Publication Publication Date Title
AU5578390A (en) Dioxothiazolidine derivatives
AU1741788A (en) Azolylmethyl-cyclopropyl derivatives
AU3613089A (en) Amino acid derivatives
AU3079789A (en) Amino acid derivatives
AU616819B2 (en) Beta-amino-boronic acid derivatives
AU3910389A (en) Indazole-3-carboxylic acid derivatives
AU8297787A (en) 1h-imadazole-5-carboxylic acid derivatives
AU8292687A (en) Thiol-carboxylic acid derivatives
AU1415188A (en) New ribofuranuronic acid derivatives
AU3301689A (en) 1-azabicyclo-alkyl derivatives
AU587108B2 (en) Imidazolecarboxylic acid derivatives
AU6892291A (en) 4-hydroxyquinaldic acid derivatives
AU2055488A (en) 7-Acylaminocephalosporin derivatives
AU2150088A (en) Isoxazole-beta-carboline derivatives
AU2963389A (en) Pyranobenzoxadiazole derivatives
AU616039B2 (en) Benzopyranol derivatives
AU3315889A (en) Phosphonoalkylpurine derivatives
AU1862088A (en) Hydroxyethyl-Azolyl derivatives
AU3579289A (en) 1,1-dioxo-cephem-4-carbothiolic acid derivatives
AU3329289A (en) Amino acid derivatives
AU3255589A (en) Amino acid derivatives
AU3330789A (en) Arylpropanamine derivatives
AU3301589A (en) Oxadiazole-1-azabicyclo-alkane derivatives
AU3156989A (en) Androst-4-ene derivatives
AU8314987A (en) 1-methyl-1h-imidazole-5-carboxylic acid derivatives