DK584283A - Aminoimidazoler, fremgangsmaade til fremstilling deraf og praeparat indeholdende en saadan forbindelse - Google Patents
Aminoimidazoler, fremgangsmaade til fremstilling deraf og praeparat indeholdende en saadan forbindelse Download PDFInfo
- Publication number
- DK584283A DK584283A DK584283A DK584283A DK584283A DK 584283 A DK584283 A DK 584283A DK 584283 A DK584283 A DK 584283A DK 584283 A DK584283 A DK 584283A DK 584283 A DK584283 A DK 584283A
- Authority
- DK
- Denmark
- Prior art keywords
- alkyl
- amino
- acetamido
- chem
- alkoxy
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title 1
- 238000000034 method Methods 0.000 title 1
- 238000002360 preparation method Methods 0.000 title 1
- -1 mono-substituted phenyl Chemical group 0.000 abstract 8
- RAXXELZNTBOGNW-UHFFFAOYSA-N imidazole Natural products C1=CNC=N1 RAXXELZNTBOGNW-UHFFFAOYSA-N 0.000 abstract 5
- 125000006273 (C1-C3) alkyl group Chemical group 0.000 abstract 3
- 125000006274 (C1-C3)alkoxy group Chemical group 0.000 abstract 3
- 125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 3
- 125000006559 (C1-C3) alkylamino group Chemical group 0.000 abstract 2
- 125000006595 (C1-C3) alkylsulfinyl group Chemical group 0.000 abstract 2
- 125000006594 (C1-C3) alkylsulfony group Chemical group 0.000 abstract 2
- 125000004455 (C1-C3) alkylthio group Chemical group 0.000 abstract 2
- 125000006698 (C1-C3) dialkylamino group Chemical group 0.000 abstract 2
- 125000004453 alkoxycarbonyl group Chemical group 0.000 abstract 2
- 125000001589 carboacyl group Chemical group 0.000 abstract 2
- 229910052736 halogen Inorganic materials 0.000 abstract 2
- 150000002367 halogens Chemical class 0.000 abstract 2
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
- 125000001424 substituent group Chemical group 0.000 abstract 2
- 125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 abstract 2
- XAKBSHICSHRJCL-UHFFFAOYSA-N [CH2]C(=O)C1=CC=CC=C1 Chemical group [CH2]C(=O)C1=CC=CC=C1 XAKBSHICSHRJCL-UHFFFAOYSA-N 0.000 abstract 1
- 125000000738 acetamido group Chemical group [H]C([H])([H])C(=O)N([H])[*] 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 125000004429 atom Chemical group 0.000 abstract 1
- 125000003739 carbamimidoyl group Chemical group C(N)(=N)* 0.000 abstract 1
- 125000003917 carbamoyl group Chemical group [H]N([H])C(*)=O 0.000 abstract 1
- 125000003178 carboxy group Chemical group [H]OC(*)=O 0.000 abstract 1
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 1
- 125000002795 guanidino group Chemical group C(N)(=N)N* 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 1
- 150000002460 imidazoles Chemical class 0.000 abstract 1
- 125000002883 imidazolyl group Chemical group 0.000 abstract 1
- 125000001624 naphthyl group Chemical group 0.000 abstract 1
- 125000004923 naphthylmethyl group Chemical group C1(=CC=CC2=CC=CC=C12)C* 0.000 abstract 1
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 1
- 229910052760 oxygen Inorganic materials 0.000 abstract 1
- 125000004076 pyridyl group Chemical group 0.000 abstract 1
- 125000005344 pyridylmethyl group Chemical group [H]C1=C([H])C([H])=C([H])C(=N1)C([H])([H])* 0.000 abstract 1
- 125000005493 quinolyl group Chemical group 0.000 abstract 1
- 229910052717 sulfur Inorganic materials 0.000 abstract 1
- 125000001889 triflyl group Chemical group FC(F)(F)S(*)(=O)=O 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/90—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Tropical Medicine & Parasitology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Emulsifying, Dispersing, Foam-Producing Or Wetting Agents (AREA)
- Plural Heterocyclic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Treatment Of Liquids With Adsorbents In General (AREA)
- Solid-Sorbent Or Filter-Aiding Compositions (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US45084882A | 1982-12-20 | 1982-12-20 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DK584283D0 DK584283D0 (da) | 1983-12-19 |
| DK584283A true DK584283A (da) | 1984-06-21 |
Family
ID=23789738
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK584283A DK584283A (da) | 1982-12-20 | 1983-12-19 | Aminoimidazoler, fremgangsmaade til fremstilling deraf og praeparat indeholdende en saadan forbindelse |
Country Status (8)
| Country | Link |
|---|---|
| EP (1) | EP0113570B1 (da) |
| JP (1) | JPS59118772A (da) |
| AT (1) | ATE25521T1 (da) |
| CA (1) | CA1245660A (da) |
| DE (1) | DE3369845D1 (da) |
| DK (1) | DK584283A (da) |
| ES (1) | ES8505202A1 (da) |
| IE (1) | IE56381B1 (da) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS59167515A (ja) * | 1983-03-15 | 1984-09-21 | Ajinomoto Co Inc | 免疫機能増強剤 |
| EP0151528B1 (en) * | 1984-02-02 | 1990-07-04 | Merck & Co. Inc. | 5-(amino or substituted amino)-1,2,3-triazoles |
| DE3627155A1 (de) * | 1986-08-11 | 1988-02-18 | Schering Ag | Imidazol-derivate |
| FI91754C (fi) * | 1986-12-02 | 1994-08-10 | Tanabe Seiyaku Co | Analogiamenetelmä lääkeaineena käyttökelpoisen imidatsolijohdannaisen valmistamiseksi |
| CA1329614C (en) * | 1987-05-02 | 1994-05-17 | Rainer Buerstinghaus | N-substituted azoles |
| US5359078A (en) * | 1989-05-19 | 1994-10-25 | The United States Of America As Represented By The Department Of Health And Human Services | Signal transduction inhibitor compounds |
| US5635521A (en) * | 1991-09-23 | 1997-06-03 | Sandoz Ltd. | Imidazolylmethyl-pyridines |
| KR100401283B1 (ko) * | 1998-07-13 | 2003-12-31 | 주식회사유한양행 | 라스변이세포성장억제구아니딘유도체 |
| CA2434300A1 (en) * | 2001-01-18 | 2002-07-25 | Schering Corporation | Synthesis of temozolomide and analogs |
| CA2434308C (en) | 2001-01-18 | 2010-09-21 | Schering Corporation | Synthesis of temozolomide and analogs |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4265900A (en) * | 1979-10-29 | 1981-05-05 | Mcneilab, Inc. | N-Aryl-N'-imidazol-2-ylureas |
| JPS5671074A (en) * | 1979-11-12 | 1981-06-13 | Takeda Chem Ind Ltd | 1,2-disubstituted-4-halogenoimidazole-5-acetic acid derivative |
-
1983
- 1983-12-16 DE DE8383307692T patent/DE3369845D1/de not_active Expired
- 1983-12-16 EP EP83307692A patent/EP0113570B1/en not_active Expired
- 1983-12-16 IE IE2975/83A patent/IE56381B1/en not_active IP Right Cessation
- 1983-12-16 AT AT83307692T patent/ATE25521T1/de not_active IP Right Cessation
- 1983-12-19 CA CA000443604A patent/CA1245660A/en not_active Expired
- 1983-12-19 ES ES528159A patent/ES8505202A1/es not_active Expired
- 1983-12-19 DK DK584283A patent/DK584283A/da not_active Application Discontinuation
- 1983-12-20 JP JP58239055A patent/JPS59118772A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| JPS59118772A (ja) | 1984-07-09 |
| EP0113570B1 (en) | 1987-02-25 |
| ES528159A0 (es) | 1985-05-16 |
| DK584283D0 (da) | 1983-12-19 |
| ES8505202A1 (es) | 1985-05-16 |
| EP0113570A1 (en) | 1984-07-18 |
| ATE25521T1 (de) | 1987-03-15 |
| DE3369845D1 (en) | 1987-04-02 |
| IE832975L (en) | 1984-06-20 |
| CA1245660A (en) | 1988-11-29 |
| IE56381B1 (en) | 1991-07-17 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| EP0151529A3 (en) | 5-(amino or substituted amino)-1,2,3-triazoles | |
| FI861995A0 (fi) | Foerfarande foer framstaellning av terapeutiskt anvaendbara 2-(4-benzoyl-1-piperidinyl)-1 -fenylalkanolderivat. | |
| DK584283D0 (da) | Aminoimidazoler, fremgangsmade til fremstilling deraf og praeparat indeholdende en sadan forbindelse | |
| DK81781A (da) | N-phenylpyrazolderivater og herbicid med indhold deraf | |
| KR890003385A (ko) | 항 증식제로서 유용한 5-아미노 또는 치환된 아미도 1,2,3-트리아졸 | |
| ZA826986B (en) | Heterocyclic phenyl ethers,processes for their preparation and herbicidal agents containing them | |
| DK24884D0 (da) | 1-heterocyclyl-2-phenyl-3-(1,2,4-triazol-1-yl)propan-2-ol-forbindelser og farmaceutisk acceptable salte deraf samt farmaceutisk praeparat indeholdende disse forbindelser | |
| DE3479212D1 (en) | New amidine derivatives of 2-substituted 4-phenilimidazole | |
| DK0421227T3 (da) | Derivater af 1-hydroxy-1,2,4-triazoler og fungicider og vækstregulerende midler indeholdende disse |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| AHS | Application shelved for other reasons than non-payment |