DK565676A - PROCEDURE FOR THE PREPARATION OF KLAVAM DERIVATIVES - Google Patents

PROCEDURE FOR THE PREPARATION OF KLAVAM DERIVATIVES

Info

Publication number
DK565676A
DK565676A DK565676A DK565676A DK565676A DK 565676 A DK565676 A DK 565676A DK 565676 A DK565676 A DK 565676A DK 565676 A DK565676 A DK 565676A DK 565676 A DK565676 A DK 565676A
Authority
DK
Denmark
Prior art keywords
klavam
derivatives
procedure
preparation
klavam derivatives
Prior art date
Application number
DK565676A
Other languages
Danish (da)
Inventor
P C Cherry
G I Gregory
P Ward
Original Assignee
Glaxo Lab Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Lab Ltd filed Critical Glaxo Lab Ltd
Publication of DK565676A publication Critical patent/DK565676A/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/429Thiazoles condensed with heterocyclic ring systems
    • A61K31/43Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D503/00Heterocyclic compounds containing 4-oxa-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxapenicillins, clavulanic acid derivatives; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Cephalosporin Compounds (AREA)
DK565676A 1975-12-17 1976-12-16 PROCEDURE FOR THE PREPARATION OF KLAVAM DERIVATIVES DK565676A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB51688/75A GB1573503A (en) 1975-12-17 1975-12-17 Clavulanic acid derivatives

Publications (1)

Publication Number Publication Date
DK565676A true DK565676A (en) 1977-06-18

Family

ID=10461003

Family Applications (1)

Application Number Title Priority Date Filing Date
DK565676A DK565676A (en) 1975-12-17 1976-12-16 PROCEDURE FOR THE PREPARATION OF KLAVAM DERIVATIVES

Country Status (10)

Country Link
JP (1) JPS5293792A (en)
AU (1) AU2064576A (en)
BE (1) BE849475A (en)
DE (1) DE2657048A1 (en)
DK (1) DK565676A (en)
FR (1) FR2335222A1 (en)
GB (1) GB1573503A (en)
NL (1) NL7613965A (en)
SE (1) SE7614181L (en)
ZA (1) ZA767496B (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2740526A1 (en) * 1976-09-09 1978-03-16 Glaxo Lab Ltd CLAVULANIC ACID COMPONENTS AND THEIR PRODUCTION
GB1587612A (en) * 1976-10-30 1981-04-08 Beecham Group Ltd Isoclavulanic acid derivatives
GB1595176A (en) * 1976-12-03 1981-08-12 Beecham Group Ltd Clavulanic acid ethers
IL53465A (en) * 1976-12-11 1980-11-30 Beecham Group Ltd Process for the preparation of clavulanic acid ethers and some novel compounds of this type
NO771106L (en) * 1977-03-10 1978-09-12 Beecham Group Ltd PROCEDURE FOR PREPARING ETHER
EP0024123B1 (en) * 1979-08-11 1983-03-16 Beecham Group Plc Process for the preparation of derivatives of clavulanic acid
GB9518917D0 (en) * 1995-09-15 1995-11-15 Smithkline Beecham Plc Compounds

Also Published As

Publication number Publication date
SE7614181L (en) 1977-06-18
FR2335222A1 (en) 1977-07-15
ZA767496B (en) 1978-02-22
JPS5293792A (en) 1977-08-06
FR2335222B1 (en) 1982-06-11
AU2064576A (en) 1978-06-22
DE2657048A1 (en) 1977-06-23
NL7613965A (en) 1977-06-21
BE849475A (en) 1977-06-16
GB1573503A (en) 1980-08-28

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