DK539478A - Fremgangsmaade til fremstilling af samatostatinanaloge - Google Patents

Fremgangsmaade til fremstilling af samatostatinanaloge

Info

Publication number
DK539478A
DK539478A DK539478A DK539478A DK539478A DK 539478 A DK539478 A DK 539478A DK 539478 A DK539478 A DK 539478A DK 539478 A DK539478 A DK 539478A DK 539478 A DK539478 A DK 539478A
Authority
DK
Denmark
Prior art keywords
samatostatin
analog
preparing
procedure
samatostatin analog
Prior art date
Application number
DK539478A
Other languages
English (en)
Inventor
D F Veber
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of DK539478A publication Critical patent/DK539478A/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/655—Somatostatins
    • C07K14/6555—Somatostatins at least 1 amino acid in D-form
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/02—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S930/00—Peptide or protein sequence
    • Y10S930/01—Peptide or protein sequence
    • Y10S930/16—Somatostatin; related peptides
DK539478A 1977-12-01 1978-11-30 Fremgangsmaade til fremstilling af samatostatinanaloge DK539478A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/856,364 US4139526A (en) 1977-12-01 1977-12-01 Somatostatin analogs

Publications (1)

Publication Number Publication Date
DK539478A true DK539478A (da) 1979-06-02

Family

ID=25323425

Family Applications (1)

Application Number Title Priority Date Filing Date
DK539478A DK539478A (da) 1977-12-01 1978-11-30 Fremgangsmaade til fremstilling af samatostatinanaloge

Country Status (7)

Country Link
US (1) US4139526A (da)
EP (1) EP0002262B1 (da)
JP (1) JPS5495591A (da)
DE (1) DE2862319D1 (da)
DK (1) DK539478A (da)
IE (1) IE47683B1 (da)
IT (1) IT1158152B (da)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4191754A (en) * 1979-02-28 1980-03-04 Merck & Co., Inc. Bicyclic somatostatin analogs
US4190648A (en) * 1979-03-13 1980-02-26 Merck & Co., Inc. Peptides having somatostatin activity
CY1327A (en) * 1979-11-27 1986-06-27 Sandoz Ag Novel polypeptides,processes for their production,pharmaceutical compositions comprising said polypeptides and their use
DE3379657D1 (en) * 1982-12-06 1989-05-24 Merck & Co Inc Dicyclic hexapeptides, processes for their preparation and pharmaceutical compositions containing them
US4663435A (en) * 1982-12-06 1987-05-05 Merck & Co., Inc. Bridged cyclic hexapeptide somatostatin analogs
DE3910667A1 (de) * 1988-04-11 1989-10-19 Sandoz Ag Peptidderivate
AU2003260306A1 (en) * 2002-07-17 2004-02-02 Boehringer Ingelheim Pharma Gmbh And Co. Kg Bicyclic oligopeptides
US7101848B2 (en) * 2002-10-08 2006-09-05 Boehringer Ingelheim Pharma Gmbh & Co. Kg Bicyclic oligopeptides

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2416048A1 (de) * 1974-04-03 1975-10-30 Hoechst Ag Neue peptide mit biologischer wirkung
DE2460469A1 (de) * 1974-12-20 1976-07-01 Hoechst Ag Neue peptide mit biologischer wirkung und verfahren zu ihrer herstellung
NL7607987A (nl) * 1975-08-08 1977-02-10 Merck & Co Inc Werkwijze voor het bereiden van peptiden.
CA1083143A (en) * 1976-01-02 1980-08-05 Nedumparambil A. Abraham Carba derivatives of somatostatin and process therefor
US3997517A (en) * 1976-01-30 1976-12-14 American Home Products Corporation Cyclic somatostatin disulfide analogues

Also Published As

Publication number Publication date
IE782372L (en) 1979-06-01
EP0002262A1 (en) 1979-06-13
US4139526A (en) 1979-02-13
JPS5495591A (en) 1979-07-28
JPS6241240B2 (da) 1987-09-02
EP0002262B1 (en) 1983-09-14
IT7852161A0 (it) 1978-12-01
IE47683B1 (en) 1984-05-30
DE2862319D1 (en) 1983-10-20
IT1158152B (it) 1987-02-18

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