DK395789D0 - USE OF ALFA AMINOBORONIC ACID DERIVATIVES FOR THE PREPARATION OF A MEDICINE FOR THERAPY OR PROPHYLAXY OF VIRUSAL DISEASES - Google Patents

USE OF ALFA AMINOBORONIC ACID DERIVATIVES FOR THE PREPARATION OF A MEDICINE FOR THERAPY OR PROPHYLAXY OF VIRUSAL DISEASES

Info

Publication number
DK395789D0
DK395789D0 DK395789A DK395789A DK395789D0 DK 395789 D0 DK395789 D0 DK 395789D0 DK 395789 A DK395789 A DK 395789A DK 395789 A DK395789 A DK 395789A DK 395789 D0 DK395789 D0 DK 395789D0
Authority
DK
Denmark
Prior art keywords
virusal
prophylaxy
alfa
therapy
diseases
Prior art date
Application number
DK395789A
Other languages
Danish (da)
Other versions
DK395789A (en
Inventor
Karin Moelling
Heinz-Werner Kleemann
Hansjoerg Urbach
Wolfgang Koenig
Dieter Ruppert
Irvin Winkler
Arnold Paessens
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of DK395789D0 publication Critical patent/DK395789D0/en
Publication of DK395789A publication Critical patent/DK395789A/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/55Protease inhibitors
    • A61K38/553Renin inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/69Boron compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
DK395789A 1988-08-12 1989-08-11 USE OF ALFA AMINOBORONIC ACID DERIVATIVES FOR THE PREPARATION OF A MEDICINE FOR THERAPY OR PROPHYLAXY OF VIRUSAL DISEASES DK395789A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE3827340A DE3827340A1 (en) 1988-08-12 1988-08-12 USE OF (ALPHA) -AMINOBORONIC ACID DERIVATIVES FOR THE PROPHYLAXIS AND TREATMENT OF VIRUS DISEASES

Publications (2)

Publication Number Publication Date
DK395789D0 true DK395789D0 (en) 1989-08-11
DK395789A DK395789A (en) 1990-02-13

Family

ID=6360676

Family Applications (1)

Application Number Title Priority Date Filing Date
DK395789A DK395789A (en) 1988-08-12 1989-08-11 USE OF ALFA AMINOBORONIC ACID DERIVATIVES FOR THE PREPARATION OF A MEDICINE FOR THERAPY OR PROPHYLAXY OF VIRUSAL DISEASES

Country Status (10)

Country Link
EP (1) EP0354522A1 (en)
JP (1) JPH0291023A (en)
KR (1) KR900002766A (en)
AU (1) AU3951389A (en)
DE (1) DE3827340A1 (en)
DK (1) DK395789A (en)
IL (1) IL91276A0 (en)
NO (1) NO893240L (en)
PT (1) PT91426A (en)
ZA (1) ZA896150B (en)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5142056A (en) * 1989-05-23 1992-08-25 Abbott Laboratories Retroviral protease inhibiting compounds
EP0315574A3 (en) * 1987-11-05 1990-08-22 Hoechst Aktiengesellschaft Renin inhibitors
US4983589A (en) * 1989-12-14 1991-01-08 Chevron Research And Technology Company Fungicidal imidazole diphenylaliphaticboranes and derivatives thereof
GB9017694D0 (en) * 1990-08-13 1990-09-26 Sandoz Ltd Improvements in or relating to organic chemistry
GB9024775D0 (en) * 1990-11-14 1991-01-02 Axis Research Chemical compounds
US5554728A (en) * 1991-07-23 1996-09-10 Nexstar Pharmaceuticals, Inc. Lipid conjugates of therapeutic peptides and protease inhibitors
DE4126485A1 (en) * 1991-08-10 1993-02-11 Bayer Ag TRIFLUOROMETHYL-CONTAINING PSEUDOPEPTIDE
US5693617A (en) * 1994-03-15 1997-12-02 Proscript, Inc. Inhibitors of the 26s proteolytic complex and the 20s proteasome contained therein
US6083903A (en) 1994-10-28 2000-07-04 Leukosite, Inc. Boronic ester and acid compounds, synthesis and uses
DE4441483C1 (en) * 1994-11-22 1996-04-04 Gsf Forschungszentrum Umwelt Use of bio-assimilated boron cpds.
US7223745B2 (en) 2003-08-14 2007-05-29 Cephalon, Inc. Proteasome inhibitors and methods of using the same
US7576206B2 (en) 2003-08-14 2009-08-18 Cephalon, Inc. Proteasome inhibitors and methods of using the same
US7468383B2 (en) 2005-02-11 2008-12-23 Cephalon, Inc. Proteasome inhibitors and methods of using the same
US7442830B1 (en) 2007-08-06 2008-10-28 Millenium Pharmaceuticals, Inc. Proteasome inhibitors
US7838673B2 (en) 2007-10-16 2010-11-23 Millennium Pharmaceuticals, Inc. Proteasome inhibitors
NZ624122A (en) 2008-06-17 2015-11-27 Millennium Pharm Inc Boronate ester compounds and pharmaceutical compositions thereof
AR075090A1 (en) 2008-09-29 2011-03-09 Millennium Pharm Inc ACID DERIVATIVES 1-AMINO-2-CYCLLOBUTILETILBORONICO PROTEOSOMA INHIBITORS, USEFUL AS ANTI-BANKER AGENTS, AND PHARMACEUTICAL COMPOSITIONS THAT UNDERSTAND THEM.
EP2516449A1 (en) 2009-12-22 2012-10-31 Cephalon, Inc. Proteasome inhibitors and processes for their preparation, purification and use
US9359398B2 (en) * 2010-03-01 2016-06-07 Onyx Therapeutics, Inc. Compounds for immunoproteasome inhibition
CN106008570A (en) 2010-03-31 2016-10-12 米伦纽姆医药公司 Derivatives of 1-amino-2-cyclopropylethylboronic acid
CN103483363B (en) * 2012-06-13 2016-12-21 上海赛迦化工产品有限公司 Multifarious chiral aminoboronic acid and its preparation method and application
CN103396426B (en) * 2013-07-12 2016-09-28 上海工程技术大学 Chirality boronic acid derivatives and its preparation method and application
CN103408572B (en) * 2013-07-12 2015-12-02 上海工程技术大学 Chiral aminoboronic acid derivative and its preparation method and application
TN2016000492A1 (en) 2014-05-20 2018-04-04 Millennium Pharm Inc Boron-containing proteasome inhibitors for use after primary cancer therapy.
EP3472151A4 (en) 2016-06-21 2020-03-04 Orion Ophthalmology LLC Carbocyclic prolinamide derivatives
EP4257191A3 (en) 2016-06-21 2023-11-22 Orion Ophthalmology LLC Heterocyclic prolinamide derivatives

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4537773A (en) * 1983-12-05 1985-08-27 E. I. Du Pont De Nemours And Company α-Aminoboronic acid derivatives
US4499082A (en) * 1983-12-05 1985-02-12 E. I. Du Pont De Nemours And Company α-Aminoboronic acid peptides
US5187157A (en) * 1987-06-05 1993-02-16 Du Pont Merck Pharmaceutical Company Peptide boronic acid inhibitors of trypsin-like proteases
EP0315574A3 (en) * 1987-11-05 1990-08-22 Hoechst Aktiengesellschaft Renin inhibitors

Also Published As

Publication number Publication date
DK395789A (en) 1990-02-13
NO893240L (en) 1990-03-27
PT91426A (en) 1990-03-08
DE3827340A1 (en) 1990-02-15
KR900002766A (en) 1990-03-31
IL91276A0 (en) 1990-03-19
EP0354522A1 (en) 1990-02-14
JPH0291023A (en) 1990-03-30
AU3951389A (en) 1990-03-29
ZA896150B (en) 1991-01-30
NO893240D0 (en) 1989-08-11

Similar Documents

Publication Publication Date Title
DK395789A (en) USE OF ALFA AMINOBORONIC ACID DERIVATIVES FOR THE PREPARATION OF A MEDICINE FOR THERAPY OR PROPHYLAXY OF VIRUSAL DISEASES
DK156376C (en) USE OF IBOGAIN FOR THE PREPARATION OF A MEDICINE FOR THE TREATMENT OF DRUGS
DK164392C (en) USE OF 3'-AZIDO-3'-DESOXYTHYMIDINE TO PREPARE A MEDICINE FOR TREATMENT OR PROPHYLAXY FOR A HUMAN RETROVIRUS INFECTION
NO861331L (en) PROCEDURE FOR THE PREPARATION OF A HYALURONIC ACID SALT.
FI102182B1 (en) Method for the preparation of human insulin analogs
ATA260690A (en) THERAPEUTIC INFUSION PREPARATION BASED ON AMINO ACID DERIVATIVES
DK195690D0 (en) USE OF COUMARIN DERIVATIVES FOR THE PREPARATION OF A MEDICINE AGAINST HUMAN IMMUNDEFECT VIRUS
DK166479C (en) USE OF FLUOXETIN, NORFLUOXETIN OR A PHARMACEUTICAL ACCEPTABLE SALT OF FLUOXETIN OR NORFLUOXETIN FOR THE PREPARATION OF A MEDICINE WITH ANXIOLYTICAL EFFECT
DK645788D0 (en) USE OF ERGOLIN DERIVATIVES FOR THE PREPARATION OF A PHARMACEUTICAL PREPARATION
NO157506C (en) PROCEDURE FOR THE PREPARATION OF HUMAN INSULIN OR TREONINB30 DERIVATIVES OF HUMAN INSULIN OR A SALT OR COMPLEX THEREOF.
NO873923L (en) PROCEDURE FOR THE PREPARATION OF A MEDICAL SKIN PREPARATION
NO865028L (en) PROCEDURE FOR THE PREPARATION OF A THERAPEUTIC SYSTEM.
DK473088D0 (en) USE OF 2-AMINO-6-TRIFLUORMETHOXYBENZOTHIAZOL FOR THE PREPARATION OF A MEDICINE
DK473288D0 (en) USE OF 2-AMINO-6-TRIFLUORMETHOXYBENZOTHIAZOL FOR THE PREPARATION OF A MEDICINE
DK425287D0 (en) PREPARATION OF A PHARMACEUTICAL PREPARATION FOR THE TREATMENT OF CONGESTIVE HEART FAILURE
DK400887A (en) USE OF 15-DEOXYSPERGUALIN FOR THE PREPARATION OF A MEDICINAL PRODUCT
DK302887A (en) USE OF TUMORNECROSE FACTOR-ALFA FOR THE PREPARATION OF ANTI-INFECTIVE MEDICINE
DK83688D0 (en) APPLICATION OF KNOWN CONNECTIONS FOR THE PREPARATION OF A MEDICINE FOR TREATMENT OF HEART DISEASES OR ORGANIC BRAIN SYNDROME
DK285589D0 (en) USE OF OXOCHINAZOLINE DERIVATIVES FOR THE PREPARATION OF A MEDICINE AGAINST HYPERLIPIDAEMIA
NO863225L (en) ANALOGUE PROCEDURE FOR THE PREPARATION OF A THERAPEUTIC EFFECTIVE BENZODIOXEPAN.
DK681288D0 (en) AENOOTROPT THERAPEUTIC MEDICINE
DK639088D0 (en) PHARMACEUTICALS FOR TREATMENT OF ISKAEMIC HEART DISEASES
DK149314C (en) PROCEDURE FOR THE PREPARATION OF HUMAN INSULIN OR THREONIN-B30 DERIVATIVES OF HUMAN INSULIN OR A SALT OR COMPLEX THEREOF
DK171089D0 (en) USE OF TETRAZOLD DERIVATIVES FOR THE PREPARATION OF MEDICINAL PRODUCTS
DK488687D0 (en) N-ALKYLBENZENESULPHONAMIDS OR A PHARMACEUTICAL ACCEPTABLE SALT THEREOF

Legal Events

Date Code Title Description
ATS Application withdrawn