DK3770165T3 - Posaconazolphosphatestermonocholinsalt, fremgangsmåde til fremstilling deraf og anvendelse deraf - Google Patents
Posaconazolphosphatestermonocholinsalt, fremgangsmåde til fremstilling deraf og anvendelse deraf Download PDFInfo
- Publication number
- DK3770165T3 DK3770165T3 DK18933805.6T DK18933805T DK3770165T3 DK 3770165 T3 DK3770165 T3 DK 3770165T3 DK 18933805 T DK18933805 T DK 18933805T DK 3770165 T3 DK3770165 T3 DK 3770165T3
- Authority
- DK
- Denmark
- Prior art keywords
- posaconazol
- preparation
- phosphate ester
- monocholine salt
- monocholine
- Prior art date
Links
- 229910019142 PO4 Inorganic materials 0.000 title 1
- -1 POSACONAZOL PHOSPHATE ESTER Chemical class 0.000 title 1
- 239000010452 phosphate Substances 0.000 title 1
- 229960001589 posaconazole Drugs 0.000 title 1
- 150000003839 salts Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6558—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
- C07F9/65586—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system at least one of the hetero rings does not contain nitrogen as ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Molecular Biology (AREA)
- Biochemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oncology (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Communicable Diseases (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN201811107484.4A CN110938093B (zh) | 2018-09-21 | 2018-09-21 | 一种泊沙康唑磷酸酯单胆碱盐及其制备方法和用途 |
| PCT/CN2018/123343 WO2020056974A1 (zh) | 2018-09-21 | 2018-12-25 | 一种泊沙康唑磷酸酯单胆碱盐及其制备方法和用途 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK3770165T3 true DK3770165T3 (da) | 2022-08-22 |
Family
ID=69888213
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK18933805.6T DK3770165T3 (da) | 2018-09-21 | 2018-12-25 | Posaconazolphosphatestermonocholinsalt, fremgangsmåde til fremstilling deraf og anvendelse deraf |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20210147455A1 (da) |
| EP (1) | EP3770165B1 (da) |
| JP (1) | JP7026264B2 (da) |
| CN (1) | CN110938093B (da) |
| AU (1) | AU2018441838B2 (da) |
| DK (1) | DK3770165T3 (da) |
| ES (1) | ES2923683T3 (da) |
| WO (1) | WO2020056974A1 (da) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN112778369B (zh) * | 2019-11-05 | 2024-01-26 | 华创合成制药股份有限公司 | 一种三唑类衍生物及其制备方法和用途 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU681753B2 (en) * | 1993-12-21 | 1997-09-04 | Merck Sharp & Dohme Corp. | Tetrahydrofuran antifungals |
| ATE240319T1 (de) * | 1995-06-02 | 2003-05-15 | Schering Corp | Antifungale tetrahydrofurane |
| JO2691B1 (en) * | 2005-05-03 | 2013-03-03 | ايساي آر آند دي مانجمنت كو.، ليمتد | Monolysine salts for azole compounds |
| CN105287403A (zh) * | 2014-08-02 | 2016-02-03 | 陕西合成药业股份有限公司 | 一种泊沙康唑前体药物的冻干组合物及其制备方法和用途 |
| CN106432338A (zh) * | 2015-08-08 | 2017-02-22 | 陕西合成药业股份有限公司 | 泊沙康唑衍生物、合成和在长效制剂中的用途 |
| CN107033186B (zh) * | 2016-02-04 | 2020-06-09 | 武汉朗来科技发展有限公司 | 泊沙康唑衍生物、其药物组合物和用途 |
| NL2017545B1 (en) * | 2016-09-28 | 2018-04-06 | Eucaryo Beheer B V | Composition comprising a bioactive molecule |
-
2018
- 2018-09-21 CN CN201811107484.4A patent/CN110938093B/zh active Active
- 2018-12-25 EP EP18933805.6A patent/EP3770165B1/en active Active
- 2018-12-25 AU AU2018441838A patent/AU2018441838B2/en active Active
- 2018-12-25 DK DK18933805.6T patent/DK3770165T3/da active
- 2018-12-25 ES ES18933805T patent/ES2923683T3/es active Active
- 2018-12-25 US US17/048,745 patent/US20210147455A1/en active Pending
- 2018-12-25 WO PCT/CN2018/123343 patent/WO2020056974A1/zh unknown
- 2018-12-25 JP JP2020570616A patent/JP7026264B2/ja active Active
Also Published As
| Publication number | Publication date |
|---|---|
| EP3770165A1 (en) | 2021-01-27 |
| JP7026264B2 (ja) | 2022-02-25 |
| AU2018441838A1 (en) | 2020-11-12 |
| CN110938093B (zh) | 2022-08-19 |
| WO2020056974A1 (zh) | 2020-03-26 |
| JP2021515049A (ja) | 2021-06-17 |
| US20210147455A1 (en) | 2021-05-20 |
| EP3770165B1 (en) | 2022-06-08 |
| CN110938093A (zh) | 2020-03-31 |
| AU2018441838B2 (en) | 2021-10-07 |
| ES2923683T3 (es) | 2022-09-29 |
| EP3770165A4 (en) | 2021-04-28 |
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