DK312988A - Fremgangsmaade til fremstilling af zidovudin samt mellemprodukter ved fremgangsmaaden - Google Patents

Fremgangsmaade til fremstilling af zidovudin samt mellemprodukter ved fremgangsmaaden

Info

Publication number
DK312988A
DK312988A DK312988A DK312988A DK312988A DK 312988 A DK312988 A DK 312988A DK 312988 A DK312988 A DK 312988A DK 312988 A DK312988 A DK 312988A DK 312988 A DK312988 A DK 312988A
Authority
DK
Denmark
Prior art keywords
procedure
zidovudin
intermediates
production
Prior art date
Application number
DK312988A
Other languages
English (en)
Other versions
DK312988D0 (da
Inventor
Jeffrey Douglas Wilson
Merrick Richard Almond
Janet Litster Rideout
Original Assignee
Wellcome Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB878713579A external-priority patent/GB8713579D0/en
Priority claimed from GB878716233A external-priority patent/GB8716233D0/en
Application filed by Wellcome Found filed Critical Wellcome Found
Publication of DK312988D0 publication Critical patent/DK312988D0/da
Publication of DK312988A publication Critical patent/DK312988A/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06Pyrimidine radicals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H13/00Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids
    • C07H13/12Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids by acids having the group -X-C(=X)-X-, or halides thereof, in which each X means nitrogen, oxygen, sulfur, selenium or tellurium, e.g. carbonic acid, carbamic acid

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK312988A 1987-06-10 1988-06-09 Fremgangsmaade til fremstilling af zidovudin samt mellemprodukter ved fremgangsmaaden DK312988A (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB878713579A GB8713579D0 (en) 1987-06-10 1987-06-10 Chemical process
GB878716233A GB8716233D0 (en) 1987-07-10 1987-07-10 Chemical process

Publications (2)

Publication Number Publication Date
DK312988D0 DK312988D0 (da) 1988-06-09
DK312988A true DK312988A (da) 1988-12-11

Family

ID=26292341

Family Applications (1)

Application Number Title Priority Date Filing Date
DK312988A DK312988A (da) 1987-06-10 1988-06-09 Fremgangsmaade til fremstilling af zidovudin samt mellemprodukter ved fremgangsmaaden

Country Status (8)

Country Link
EP (1) EP0295090A3 (da)
JP (1) JPS649995A (da)
KR (1) KR890000510A (da)
DK (1) DK312988A (da)
FI (1) FI882744A (da)
HU (1) HUT49626A (da)
IL (1) IL86670A0 (da)
YU (1) YU110888A (da)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH07116210B2 (ja) * 1988-02-10 1995-12-13 長谷川香料株式会社 チミン誘導体
DE4021006A1 (de) * 1990-07-02 1992-01-09 Hoechst Ag Pyrimidin-derivate, deren herstellung und verwendung sowie diese enthaltende arzneimittel
US5466787A (en) * 1993-11-15 1995-11-14 Bristol-Myers Squibb Company Process for preparing AZT
US5672698A (en) * 1993-11-15 1997-09-30 Bristol-Myers Squibb Co. Preparation of 2',3'-didehydro-3'-deoxythymidine from 5-methyluridine

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4604382A (en) * 1983-01-17 1986-08-05 Research Corporation 3'-amino-2',3'-dideoxycytidine and the pharmacologically acceptable salts thereof
EP0291633B1 (en) * 1985-03-16 1992-11-04 The Wellcome Foundation Limited Use of 3'-azido-3'-deoxythymidine in the treatment or prophylaxis of human retroviral infections
IE73219B1 (en) * 1985-03-16 1997-05-07 Wellcome Found Therapeutic nucleosides

Also Published As

Publication number Publication date
FI882744A0 (fi) 1988-06-09
DK312988D0 (da) 1988-06-09
IL86670A0 (en) 1988-11-30
YU110888A (en) 1989-08-31
EP0295090A3 (en) 1990-01-31
KR890000510A (ko) 1989-03-15
EP0295090A2 (en) 1988-12-14
HUT49626A (en) 1989-10-30
FI882744A (fi) 1988-12-11
JPS649995A (en) 1989-01-13

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Legal Events

Date Code Title Description
AHB Application shelved due to non-payment