DK214479A - Fremgangsmaade til fremstilling af 2,4-diamono-5-(3,5-dialkyl-4-hydroxybenzyl) pyrimidiner - Google Patents
Fremgangsmaade til fremstilling af 2,4-diamono-5-(3,5-dialkyl-4-hydroxybenzyl) pyrimidinerInfo
- Publication number
- DK214479A DK214479A DK214479A DK214479A DK214479A DK 214479 A DK214479 A DK 214479A DK 214479 A DK214479 A DK 214479A DK 214479 A DK214479 A DK 214479A DK 214479 A DK214479 A DK 214479A
- Authority
- DK
- Denmark
- Prior art keywords
- diamono
- hydroxybenzyl
- pyrimidines
- dialkyl
- preparing
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/30—Halogen atoms or nitro radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/63—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/63—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide
- A61K31/635—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide having a heterocyclic ring, e.g. sulfadiazine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/48—Two nitrogen atoms
- C07D239/49—Two nitrogen atoms with an aralkyl radical, or substituted aralkyl radical, attached in position 5, e.g. trimethoprim
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/52—Two oxygen atoms
- C07D239/54—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Oncology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB2193878 | 1978-05-24 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK214479A true DK214479A (da) | 1979-11-25 |
Family
ID=10171323
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK214479A DK214479A (da) | 1978-05-24 | 1979-05-23 | Fremgangsmaade til fremstilling af 2,4-diamono-5-(3,5-dialkyl-4-hydroxybenzyl) pyrimidiner |
Country Status (12)
| Country | Link |
|---|---|
| EP (1) | EP0006987A1 (da) |
| JP (1) | JPS54154775A (da) |
| AU (1) | AU4732579A (da) |
| DK (1) | DK214479A (da) |
| FI (1) | FI791638A (da) |
| IL (1) | IL57375A0 (da) |
| IT (1) | IT1117752B (da) |
| MA (1) | MA18450A1 (da) |
| MC (1) | MC1264A1 (da) |
| NO (1) | NO791699L (da) |
| PT (1) | PT69656A (da) |
| ZW (1) | ZW9979A1 (da) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DK523781A (da) * | 1980-11-27 | 1982-05-28 | Wellcome Found | Fremgangsmaade til fremstilling af benzylpyrimidiner samt mellemprodukt for disse |
| HU188588B (en) * | 1982-08-13 | 1986-04-28 | Egyt Gyogyszervegyeszeti Gyar | Process for the production of 2,4-diamino-5-benzyl-pyrimidine-derivatives |
| FR2652812A1 (fr) * | 1989-10-09 | 1991-04-12 | Rhone Poulenc Chimie | Procede de preparation de difluoro-2,2 benzodioxole-1,3. |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB875562A (en) * | 1957-02-21 | 1961-08-23 | Wellcome Found | Improvements in and relating to pyrimidine derivatives and the preparation thereof |
| GB1128234A (en) * | 1966-02-19 | 1968-09-25 | Wellcome Found | 5-benzylpyrimidine derivatives and process for the preparation thereof |
| CH544053A (de) * | 1966-05-09 | 1973-11-15 | Hoffmann La Roche | Verfahren zur Herstellung von Sulfonamidderivaten |
| US3684810A (en) * | 1970-03-11 | 1972-08-15 | Hoffmann La Roche | Process for 2,4-diamino-5-(3,5-dimethoxy-4-hydroxybenzyl) pyrimidine |
| GB1375162A (da) * | 1970-10-22 | 1974-11-27 | ||
| BE789904A (fr) * | 1971-10-12 | 1973-04-10 | Wellcome Found | Procedes de synthese organique |
| GB1413472A (en) * | 1971-10-12 | 1975-11-12 | Wellcome Found | 2,4-diamino pyrimidines |
| DE2546667C3 (de) * | 1975-10-17 | 1978-10-12 | Ludwig Heumann & Co Gmbh, 8500 Nuernberg | 2,4-DiamüH»-5-(3-methoxy-4-hydroxy-5-halogenbenzyl)-pyrimidine, und diese Verbindungen enthaltende Arzneimittel |
-
1979
- 1979-05-23 PT PT69656A patent/PT69656A/pt unknown
- 1979-05-23 MA MA18644A patent/MA18450A1/fr unknown
- 1979-05-23 JP JP6376279A patent/JPS54154775A/ja active Pending
- 1979-05-23 EP EP79101596A patent/EP0006987A1/en not_active Withdrawn
- 1979-05-23 DK DK214479A patent/DK214479A/da unknown
- 1979-05-23 IL IL57375A patent/IL57375A0/xx unknown
- 1979-05-23 NO NO791699A patent/NO791699L/no unknown
- 1979-05-23 IT IT49150/79A patent/IT1117752B/it active
- 1979-05-23 ZW ZW99/79A patent/ZW9979A1/xx unknown
- 1979-05-23 FI FI791638A patent/FI791638A/fi not_active Application Discontinuation
- 1979-05-23 AU AU47325/79A patent/AU4732579A/en not_active Abandoned
- 1979-05-23 MC MC791383A patent/MC1264A1/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| IL57375A0 (en) | 1979-09-30 |
| NO791699L (no) | 1979-11-27 |
| PT69656A (en) | 1979-06-01 |
| MA18450A1 (fr) | 1979-12-31 |
| EP0006987A1 (en) | 1980-01-23 |
| FI791638A (fi) | 1979-11-25 |
| MC1264A1 (fr) | 1980-03-28 |
| JPS54154775A (en) | 1979-12-06 |
| ZW9979A1 (en) | 1980-12-24 |
| AU4732579A (en) | 1979-11-29 |
| IT7949150A0 (it) | 1979-05-23 |
| IT1117752B (it) | 1986-02-24 |
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