DK170499B1 - Anvendelse af doxazosin til fremstilling af farmaceutiske præparater mod atherosclerose - Google Patents
Anvendelse af doxazosin til fremstilling af farmaceutiske præparater mod atherosclerose Download PDFInfo
- Publication number
- DK170499B1 DK170499B1 DK313688A DK313688A DK170499B1 DK 170499 B1 DK170499 B1 DK 170499B1 DK 313688 A DK313688 A DK 313688A DK 313688 A DK313688 A DK 313688A DK 170499 B1 DK170499 B1 DK 170499B1
- Authority
- DK
- Denmark
- Prior art keywords
- doxazosin
- atherosclerosis
- aortic
- acid addition
- pharmaceutically acceptable
- Prior art date
Links
- 229960001389 doxazosin Drugs 0.000 title claims abstract description 30
- RUZYUOTYCVRMRZ-UHFFFAOYSA-N doxazosin Chemical compound C1OC2=CC=CC=C2OC1C(=O)N(CC1)CCN1C1=NC(N)=C(C=C(C(OC)=C2)OC)C2=N1 RUZYUOTYCVRMRZ-UHFFFAOYSA-N 0.000 title claims abstract description 30
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Heart & Thoracic Surgery (AREA)
- Urology & Nephrology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Cardiology (AREA)
- Vascular Medicine (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US8971687 | 1987-08-26 | ||
| US07/089,716 US4758569A (en) | 1987-08-26 | 1987-08-26 | Doxazosin as an anti-atherosclerosis agent |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| DK313688D0 DK313688D0 (da) | 1988-06-09 |
| DK313688A DK313688A (da) | 1989-02-27 |
| DK170499B1 true DK170499B1 (da) | 1995-10-02 |
Family
ID=22219243
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK313688A DK170499B1 (da) | 1987-08-26 | 1988-06-09 | Anvendelse af doxazosin til fremstilling af farmaceutiske præparater mod atherosclerose |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US4758569A (enExample) |
| EP (1) | EP0305028B1 (enExample) |
| JP (1) | JPS6471817A (enExample) |
| KR (1) | KR910002145B1 (enExample) |
| AT (1) | ATE77552T1 (enExample) |
| AU (1) | AU594880B2 (enExample) |
| CA (1) | CA1323572C (enExample) |
| DE (1) | DE3872333T2 (enExample) |
| DK (1) | DK170499B1 (enExample) |
| HU (1) | HU204196B (enExample) |
| IE (1) | IE60005B1 (enExample) |
| IL (1) | IL86735A (enExample) |
| MY (1) | MY103102A (enExample) |
| NZ (1) | NZ225053A (enExample) |
| ZA (1) | ZA884237B (enExample) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4837111A (en) * | 1988-03-21 | 1989-06-06 | Alza Corporation | Dosage form for dispensing drug for human therapy |
| US5270323A (en) * | 1990-05-31 | 1993-12-14 | Pfizer Inc. | Method of treating impotence |
| US5595872A (en) * | 1992-03-06 | 1997-01-21 | Bristol-Myers Squibb Company | Nucleic acids encoding microsomal trigyceride transfer protein |
| ES2139624T3 (es) * | 1992-04-01 | 2000-02-16 | Pfizer | Metabolitos hidroxilados y derivados de doxazosin como agentes anti-ateroesclerosis. |
| US5449679A (en) * | 1994-07-29 | 1995-09-12 | Leonard; Robert J. | Process and products for reducing biological fluid levels of a lipid soluble waste |
| US6177430B1 (en) | 1997-03-27 | 2001-01-23 | Pfizer Inc | Use of α1-adrenoreceptor antagonists in the prevention and treatment of benign prostatic hyperplasia |
| IL120303A0 (en) * | 1996-03-27 | 1997-06-10 | Pfizer | Use of alpha1-adrenoreceptor antagonists in the prevention and treatment of cancer |
| WO2000045809A1 (en) * | 1999-02-05 | 2000-08-10 | Nitrosystems, Inc. | L-arginine based formulations for treating diseases and methods of using same |
| US6974806B2 (en) * | 2000-07-13 | 2005-12-13 | Takeda Pharmaceutical Company Limited | Lipid-rich plaque inhibitors |
| US20040019096A1 (en) * | 2001-10-23 | 2004-01-29 | Vlassios Andronis | Novel formulations of carvedilol |
| KR100462304B1 (ko) * | 2002-07-30 | 2004-12-17 | 씨제이 주식회사 | 암로디핀의 유기산염 |
| KR100496436B1 (ko) * | 2002-07-30 | 2005-06-20 | 씨제이 주식회사 | 암로디핀의 유기산염 |
| KR100538641B1 (ko) * | 2002-07-30 | 2005-12-22 | 씨제이 주식회사 | 암로디핀의 유기산염 |
| KR100467669B1 (ko) | 2002-08-21 | 2005-01-24 | 씨제이 주식회사 | 암로디핀의 유기산염 |
| CN100394989C (zh) | 2002-11-15 | 2008-06-18 | 华沙整形外科股份有限公司 | 包含微粒状基于胶原材料的组合物的制药应用和包含所述组合物的滑膜关节 |
| US8118779B2 (en) | 2006-06-30 | 2012-02-21 | Warsaw Orthopedic, Inc. | Collagen delivery device |
| US8399619B2 (en) | 2006-06-30 | 2013-03-19 | Warsaw Orthopedic, Inc. | Injectable collagen material |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4130647A (en) * | 1977-07-08 | 1978-12-19 | Pfizer Inc. | Methods for treating congestive heart failure and ischemic heart disease |
| US4188390A (en) * | 1977-11-05 | 1980-02-12 | Pfizer Inc. | Antihypertensive 4-amino-2-[4-(1,4-benzodioxan-2-carbonyl) piperazin-1-yl or homopiperazin-1-yl]quinazolines |
| US4361564A (en) * | 1978-11-30 | 1982-11-30 | Edwards K David G | Renoprotective treatments employing vasodilator compounds |
| US4532135A (en) * | 1981-02-09 | 1985-07-30 | Edwards K David G | Renoprotective treatments employing vasodilator compounds |
| US4582832A (en) * | 1984-10-09 | 1986-04-15 | Pfizer Inc. | Trimazosin as an anti-atherosclerosis agent |
-
1987
- 1987-08-26 US US07/089,716 patent/US4758569A/en not_active Expired - Lifetime
-
1988
- 1988-06-03 EP EP88305069A patent/EP0305028B1/en not_active Expired - Lifetime
- 1988-06-03 AT AT88305069T patent/ATE77552T1/de not_active IP Right Cessation
- 1988-06-03 DE DE8888305069T patent/DE3872333T2/de not_active Expired - Lifetime
- 1988-06-07 IE IE169588A patent/IE60005B1/en not_active IP Right Cessation
- 1988-06-09 DK DK313688A patent/DK170499B1/da not_active IP Right Cessation
- 1988-06-09 AU AU17529/88A patent/AU594880B2/en not_active Expired
- 1988-06-14 ZA ZA884237A patent/ZA884237B/xx unknown
- 1988-06-14 IL IL8673588A patent/IL86735A/en not_active IP Right Cessation
- 1988-06-15 MY MYPI88000660A patent/MY103102A/en unknown
- 1988-06-16 NZ NZ225053A patent/NZ225053A/en unknown
- 1988-06-20 HU HU883139A patent/HU204196B/hu unknown
- 1988-07-30 KR KR1019880009761A patent/KR910002145B1/ko not_active Expired
- 1988-08-23 CA CA000575443A patent/CA1323572C/en not_active Expired - Lifetime
- 1988-08-23 JP JP63209329A patent/JPS6471817A/ja active Granted
Also Published As
| Publication number | Publication date |
|---|---|
| DK313688A (da) | 1989-02-27 |
| IE60005B1 (en) | 1994-05-18 |
| AU594880B2 (en) | 1990-03-15 |
| KR910002145B1 (ko) | 1991-04-06 |
| IE881695L (en) | 1989-02-26 |
| DE3872333T2 (de) | 1992-12-03 |
| IL86735A (en) | 1994-05-30 |
| AU1752988A (en) | 1989-03-02 |
| ZA884237B (en) | 1990-02-28 |
| NZ225053A (en) | 1997-02-24 |
| HU204196B (en) | 1991-12-30 |
| EP0305028B1 (en) | 1992-06-24 |
| ATE77552T1 (de) | 1992-07-15 |
| MY103102A (en) | 1993-04-30 |
| US4758569A (en) | 1988-07-19 |
| DE3872333D1 (de) | 1992-07-30 |
| DK313688D0 (da) | 1988-06-09 |
| IL86735A0 (en) | 1988-11-30 |
| JPS6471817A (en) | 1989-03-16 |
| EP0305028A3 (en) | 1990-03-14 |
| HUT51141A (en) | 1990-04-28 |
| KR890003379A (ko) | 1989-04-14 |
| EP0305028A2 (en) | 1989-03-01 |
| JPH0575729B2 (enExample) | 1993-10-21 |
| CA1323572C (en) | 1993-10-26 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B1 | Patent granted (law 1993) | ||
| PUP | Patent expired |