DK1558931T3 - Analyse af oplöselighed og stabilitet af farmaceutisk middel - Google Patents

Analyse af oplöselighed og stabilitet af farmaceutisk middel

Info

Publication number
DK1558931T3
DK1558931T3 DK03779464T DK03779464T DK1558931T3 DK 1558931 T3 DK1558931 T3 DK 1558931T3 DK 03779464 T DK03779464 T DK 03779464T DK 03779464 T DK03779464 T DK 03779464T DK 1558931 T3 DK1558931 T3 DK 1558931T3
Authority
DK
Denmark
Prior art keywords
analysis
solubility
stability
interest
mixtures
Prior art date
Application number
DK03779464T
Other languages
English (en)
Inventor
Hongming Chen
Hector Guzman
Colin Gardner
Original Assignee
Transform Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Transform Pharmaceuticals Inc filed Critical Transform Pharmaceuticals Inc
Application granted granted Critical
Publication of DK1558931T3 publication Critical patent/DK1558931T3/da

Links

Classifications

    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J19/00—Chemical, physical or physico-chemical processes in general; Their relevant apparatus
    • B01J19/0046—Sequential or parallel reactions, e.g. for the synthesis of polypeptides or polynucleotides; Apparatus and devices for combinatorial chemistry or for making molecular arrays
    • G—PHYSICS
    • G01—MEASURING; TESTING
    • G01N—INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
    • G01N33/00—Investigating or analysing materials by specific methods not covered by groups G01N1/00 - G01N31/00
    • G01N33/48—Biological material, e.g. blood, urine; Haemocytometers
    • G01N33/50—Chemical analysis of biological material, e.g. blood, urine; Testing involving biospecific ligand binding methods; Immunological testing
    • G01N33/53—Immunoassay; Biospecific binding assay; Materials therefor
    • G01N33/5306—Improving reaction conditions, e.g. reduction of non-specific binding, promotion of specific binding
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J2219/00—Chemical, physical or physico-chemical processes in general; Their relevant apparatus
    • B01J2219/00274—Sequential or parallel reactions; Apparatus and devices for combinatorial chemistry or for making arrays; Chemical library technology
    • B01J2219/00277—Apparatus
    • B01J2219/00279—Features relating to reactor vessels
    • B01J2219/00281—Individual reactor vessels
    • B01J2219/00283—Reactor vessels with top opening
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J2219/00—Chemical, physical or physico-chemical processes in general; Their relevant apparatus
    • B01J2219/00274—Sequential or parallel reactions; Apparatus and devices for combinatorial chemistry or for making arrays; Chemical library technology
    • B01J2219/00277—Apparatus
    • B01J2219/00279—Features relating to reactor vessels
    • B01J2219/00306—Reactor vessels in a multiple arrangement
    • B01J2219/00308—Reactor vessels in a multiple arrangement interchangeably mounted in racks or blocks
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J2219/00—Chemical, physical or physico-chemical processes in general; Their relevant apparatus
    • B01J2219/00274—Sequential or parallel reactions; Apparatus and devices for combinatorial chemistry or for making arrays; Chemical library technology
    • B01J2219/00277—Apparatus
    • B01J2219/00279—Features relating to reactor vessels
    • B01J2219/00306—Reactor vessels in a multiple arrangement
    • B01J2219/00313—Reactor vessels in a multiple arrangement the reactor vessels being formed by arrays of wells in blocks
    • B01J2219/00315—Microtiter plates
    • B01J2219/00317—Microwell devices, i.e. having large numbers of wells
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J2219/00—Chemical, physical or physico-chemical processes in general; Their relevant apparatus
    • B01J2219/00274—Sequential or parallel reactions; Apparatus and devices for combinatorial chemistry or for making arrays; Chemical library technology
    • B01J2219/00277—Apparatus
    • B01J2219/00351—Means for dispensing and evacuation of reagents
    • B01J2219/00353—Pumps
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J2219/00—Chemical, physical or physico-chemical processes in general; Their relevant apparatus
    • B01J2219/00274—Sequential or parallel reactions; Apparatus and devices for combinatorial chemistry or for making arrays; Chemical library technology
    • B01J2219/00277—Apparatus
    • B01J2219/00351—Means for dispensing and evacuation of reagents
    • B01J2219/00364—Pipettes
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J2219/00—Chemical, physical or physico-chemical processes in general; Their relevant apparatus
    • B01J2219/00274—Sequential or parallel reactions; Apparatus and devices for combinatorial chemistry or for making arrays; Chemical library technology
    • B01J2219/00277—Apparatus
    • B01J2219/00495—Means for heating or cooling the reaction vessels
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J2219/00—Chemical, physical or physico-chemical processes in general; Their relevant apparatus
    • B01J2219/00274—Sequential or parallel reactions; Apparatus and devices for combinatorial chemistry or for making arrays; Chemical library technology
    • B01J2219/00583—Features relative to the processes being carried out
    • B01J2219/00585—Parallel processes
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J2219/00—Chemical, physical or physico-chemical processes in general; Their relevant apparatus
    • B01J2219/00274—Sequential or parallel reactions; Apparatus and devices for combinatorial chemistry or for making arrays; Chemical library technology
    • B01J2219/00583—Features relative to the processes being carried out
    • B01J2219/00599—Solution-phase processes
    • B—PERFORMING OPERATIONS; TRANSPORTING
    • B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
    • B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
    • B01J2219/00—Chemical, physical or physico-chemical processes in general; Their relevant apparatus
    • B01J2219/00274—Sequential or parallel reactions; Apparatus and devices for combinatorial chemistry or for making arrays; Chemical library technology
    • B01J2219/00718—Type of compounds synthesised
    • B01J2219/00756—Compositions, e.g. coatings, crystals, formulations

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Urology & Nephrology (AREA)
  • Organic Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Hematology (AREA)
  • Molecular Biology (AREA)
  • General Physics & Mathematics (AREA)
  • Biochemistry (AREA)
  • Food Science & Technology (AREA)
  • Medicinal Chemistry (AREA)
  • Microbiology (AREA)
  • Analytical Chemistry (AREA)
  • Cell Biology (AREA)
  • General Health & Medical Sciences (AREA)
  • Physics & Mathematics (AREA)
  • Pathology (AREA)
  • Biotechnology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Investigating Or Analysing Biological Materials (AREA)
  • Blow-Moulding Or Thermoforming Of Plastics Or The Like (AREA)
  • Extrusion Moulding Of Plastics Or The Like (AREA)
DK03779464T 2002-11-04 2003-11-04 Analyse af oplöselighed og stabilitet af farmaceutisk middel DK1558931T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US42336502P 2002-11-04 2002-11-04
US42336602P 2002-11-04 2002-11-04
PCT/US2003/035094 WO2004041202A2 (en) 2002-11-04 2003-11-04 Analysis of pharmaceutical solubility and stability

Publications (1)

Publication Number Publication Date
DK1558931T3 true DK1558931T3 (da) 2007-10-15

Family

ID=32314483

Family Applications (1)

Application Number Title Priority Date Filing Date
DK03779464T DK1558931T3 (da) 2002-11-04 2003-11-04 Analyse af oplöselighed og stabilitet af farmaceutisk middel

Country Status (9)

Country Link
US (1) US20040106098A1 (da)
EP (1) EP1558931B1 (da)
JP (1) JP2006513404A (da)
AT (1) ATE364840T1 (da)
AU (2) AU2003285143A1 (da)
DE (1) DE60314441T2 (da)
DK (1) DK1558931T3 (da)
ES (1) ES2287544T3 (da)
WO (2) WO2004042359A2 (da)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7889346B2 (en) * 2003-12-31 2011-02-15 University Of South Carolina Thin-layer porous optical sensors for gases and other fluids
EP1776106B1 (en) * 2004-06-22 2013-08-07 Vertex Pharmaceuticals Incorporated Heterocyclic derivatives for modulation of calcium channels
US20070201136A1 (en) * 2004-09-13 2007-08-30 University Of South Carolina Thin Film Interference Filter and Bootstrap Method for Interference Filter Thin Film Deposition Process Control
EP1879013A4 (en) * 2005-04-20 2014-05-21 Chugai Pharmaceutical Co Ltd METHOD FOR CONSTRUCTING SELF-VULGATED DRUG ORMULATIONS
WO2007061436A1 (en) * 2005-11-28 2007-05-31 University Of South Carolina Self calibration methods for optical analysis system
US20070166245A1 (en) 2005-11-28 2007-07-19 Leonard Mackles Propellant free foamable toothpaste composition
WO2007064575A1 (en) 2005-11-28 2007-06-07 Ometric Corporation Optical analysis system and method for real time multivariate optical computing
US8208147B2 (en) 2005-11-28 2012-06-26 Halliburton Energy Services, Inc. Method of high-speed monitoring based on the use of multivariate optical elements
EP2033196A2 (en) 2006-06-26 2009-03-11 University of South Carolina Data validation and classification in optical analysis systems
GB0618514D0 (en) * 2006-09-20 2006-11-01 Univ Nottingham Trent Method of detecting interactions on a microarray using nuclear magnetic resonance
WO2008057912A2 (en) * 2006-11-02 2008-05-15 University Of South Carolina Multi-analyte optical computing system
US8184295B2 (en) * 2007-03-30 2012-05-22 Halliburton Energy Services, Inc. Tablet analysis and measurement system
WO2008121684A1 (en) * 2007-03-30 2008-10-09 University Of South Carolina Novel multi-analyte optical computing system
WO2008121715A1 (en) * 2007-03-30 2008-10-09 Ometric Corporation In-line process measurement systems and methods
US8283633B2 (en) * 2007-11-30 2012-10-09 Halliburton Energy Services, Inc. Tuning D* with modified thermal detectors
US8212213B2 (en) * 2008-04-07 2012-07-03 Halliburton Energy Services, Inc. Chemically-selective detector and methods relating thereto
WO2012128603A1 (fr) 2011-03-22 2012-09-27 Aouad Salah Mohammed Dispositif automatique et procede de preparation de solutions
US20140045724A1 (en) * 2012-08-10 2014-02-13 Jon Selbo Formulation screening methods, apparatuses for performing such methods and formulations formed by such methods
MA41872B1 (fr) * 2015-08-03 2020-10-28 Mohammed Salah Aouad Dispositif et procede pour le developement de formulations
EP3532807A4 (en) * 2016-10-25 2020-07-01 Abbott Laboratories ASSESSMENT AND CONTROL OF REAGENTS IN THE AUTOMATED PREPARATION OF SLIDES

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9424125D0 (en) * 1994-11-23 1995-01-18 Univ Cranfield Electrochemical sensor and novel media for bioelectrochemical reactions
US5616621A (en) * 1995-01-30 1997-04-01 American Home Products Corporation Taste masking liquids
US5699934A (en) * 1996-01-29 1997-12-23 Universal Instruments Corporation Dispenser and method for dispensing viscous fluids
EP0907412B1 (en) * 1996-06-28 2008-08-27 Caliper Life Sciences, Inc. High-throughput screening assay systems in microscale fluidic devices
US6544193B2 (en) * 1996-09-04 2003-04-08 Marcio Marc Abreu Noninvasive measurement of chemical substances
US6004967A (en) * 1996-09-13 1999-12-21 Sugen, Inc. Psoriasis treatment with quinazoline compounds
US6109717A (en) * 1997-05-13 2000-08-29 Sarnoff Corporation Multi-element fluid delivery apparatus and methods
EP1004015B1 (en) * 1997-08-15 2004-01-02 Alexion Pharmaceuticals, Inc. Apparatus for performing assays at reaction sites
US6485703B1 (en) * 1998-07-31 2002-11-26 The Texas A&M University System Compositions and methods for analyte detection
WO2000033818A1 (en) * 1998-12-11 2000-06-15 Nostrum Pharmaceuticals, Inc. Sustained release tablet containing hydrocolloid and cellulose ether
EP1248869A2 (en) * 2000-01-07 2002-10-16 Transform Pharmaceuticals, Inc. High-throughput formation, identification, and analysis of diverse solid-forms
US20010044112A1 (en) * 2000-03-24 2001-11-22 Lyles Mark B. High throughput screening array containing porous material
CA2457408A1 (en) * 2001-07-13 2003-01-23 Pharmacopeia, Inc. System and method for aqueous solubility prediction
EP1425577A4 (en) * 2001-08-10 2004-12-29 Symyx Technologies Inc APPARATUSES AND METHODS FOR PREPARING AND TESTING PRE-FORMULATIONS AND CORRESPONDING SYSTEMS
WO2003023394A2 (en) * 2001-09-12 2003-03-20 Phares Pharmaceutical Research N.V. Kit for screening compounds with low water solubility
US20030230488A1 (en) * 2002-06-13 2003-12-18 Lawrence Lee Microfluidic device preparation system
AU2003264805A1 (en) * 2002-10-18 2004-05-04 Brian David Bissett Automated kinetci solubility assay apparatus and method

Also Published As

Publication number Publication date
US20040106098A1 (en) 2004-06-03
ES2287544T3 (es) 2007-12-16
WO2004042359A3 (en) 2004-08-05
AU2003285143A8 (en) 2004-06-07
AU2003287491A8 (en) 2004-06-07
ATE364840T1 (de) 2007-07-15
EP1558931A2 (en) 2005-08-03
AU2003285143A1 (en) 2004-06-07
WO2004041202A2 (en) 2004-05-21
EP1558931B1 (en) 2007-06-13
DE60314441T2 (de) 2008-02-21
DE60314441D1 (de) 2007-07-26
AU2003287491A1 (en) 2004-06-07
WO2004042359A2 (en) 2004-05-21
JP2006513404A (ja) 2006-04-20
WO2004041202A3 (en) 2004-07-22
EP1558931A4 (en) 2006-08-30

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