DK145228C - ANALOGY PROCEDURE FOR PREPARING 3-AMINO-4-DEOXO-4-IMINORIFAMYCIN DERIVATIVES - Google Patents

ANALOGY PROCEDURE FOR PREPARING 3-AMINO-4-DEOXO-4-IMINORIFAMYCIN DERIVATIVES

Info

Publication number
DK145228C
DK145228C DK258076A DK258076A DK145228C DK 145228 C DK145228 C DK 145228C DK 258076 A DK258076 A DK 258076A DK 258076 A DK258076 A DK 258076A DK 145228 C DK145228 C DK 145228C
Authority
DK
Denmark
Prior art keywords
iminorifamycin
deoxo
derivatives
amino
preparing
Prior art date
Application number
DK258076A
Other languages
Danish (da)
Other versions
DK145228B (en
DK258076A (en
Inventor
L Marsili
V Rossetti
C Pasqualucci
Original Assignee
Erba Farmitalia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Erba Farmitalia filed Critical Erba Farmitalia
Publication of DK258076A publication Critical patent/DK258076A/en
Publication of DK145228B publication Critical patent/DK145228B/en
Application granted granted Critical
Publication of DK145228C publication Critical patent/DK145228C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/08Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • A61P31/06Antibacterial agents for tuberculosis
DK258076A 1975-06-13 1976-06-10 ANALOGY PROCEDURE FOR PREPARING 3-AMINO-4-DEOXO-4-IMINORIFAMYCIN DERIVATIVES DK145228C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT755174A IT1056272B (en) 1975-06-13 1975-06-13 PRODUCTS DERIVED FROM AROMATIC AMINES
IT517475 1975-06-13

Publications (3)

Publication Number Publication Date
DK258076A DK258076A (en) 1976-12-14
DK145228B DK145228B (en) 1982-10-11
DK145228C true DK145228C (en) 1983-02-28

Family

ID=11118842

Family Applications (1)

Application Number Title Priority Date Filing Date
DK258076A DK145228C (en) 1975-06-13 1976-06-10 ANALOGY PROCEDURE FOR PREPARING 3-AMINO-4-DEOXO-4-IMINORIFAMYCIN DERIVATIVES

Country Status (28)

Country Link
US (2) US4086225A (en)
JP (1) JPS5236683A (en)
AR (1) AR211127A1 (en)
AU (1) AU497602B2 (en)
BE (1) BE842883A (en)
CA (1) CA1059123A (en)
CH (1) CH625524A5 (en)
CS (1) CS197271B1 (en)
DK (1) DK145228C (en)
ES (1) ES449187A1 (en)
FI (1) FI60208C (en)
FR (1) FR2314189A1 (en)
GB (1) GB1542063A (en)
HK (1) HK56083A (en)
HU (1) HU171396B (en)
IE (1) IE42998B1 (en)
IL (1) IL49701A (en)
IN (1) IN143526B (en)
IT (1) IT1056272B (en)
NL (1) NL177919C (en)
NO (1) NO148848C (en)
PH (1) PH16410A (en)
PL (1) PL99493B1 (en)
PT (1) PT65208B (en)
SE (1) SE434057B (en)
SU (1) SU680649A3 (en)
YU (1) YU39768B (en)
ZA (1) ZA763256B (en)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1056272B (en) * 1975-06-13 1982-01-30 Archifar Ind Chim Trentino PRODUCTS DERIVED FROM AROMATIC AMINES
DK345977A (en) * 1976-09-30 1978-03-31 Archifar Ind Chim Trentino G RIFAMYCIN COMPOUNDS AND PROCEDURE FOR THEIR PREPARATION
BE886395A (en) * 1980-02-13 1981-03-16 Erba Farmitalia RIFAMYCIN DERIVATIVES
IT1201963B (en) * 1983-03-24 1989-02-02 Prodotti Antibiotici Spa DERIVATIVES OF THE REFAMICINE AND PROCEDURE FOR THEIR PREPARATION
US4631290A (en) * 1985-08-29 1986-12-23 American Home Products Corporation Method of treating hepatitis
US5529994A (en) * 1993-05-05 1996-06-25 Palo Alto Medical Foundation Treatment for toxoplasmosis
ES2095772T3 (en) * 1993-05-05 1997-02-16 Palo Alto Medical Found USE OF RIFAMYCIN DERIVATIVES TO PRODUCE A MEDICINE INTENDED FOR THE TREATMENT OF TOXOPLASMOSIS.
US5981522A (en) * 1995-09-01 1999-11-09 Kaneka Corporation Treatment of disease caused by infection of Helicobacter
CA2204007A1 (en) * 1995-09-01 1997-03-13 Katsuji Yamashita Remedy for diseases caused by infection with helicobacter
JP2005510534A (en) * 2001-11-21 2005-04-21 アクティブバイオティクス インコーポレイティッド Targeted therapeutics and uses thereof
US7078399B2 (en) * 2001-12-13 2006-07-18 Activbiotics, Inc. Sulfhydryl rifamycins and uses thereof
US7820652B2 (en) * 2003-09-24 2010-10-26 Activbiotics Pharma, Llc Regimen for the administration of rifamycin-class antibiotics
US7202246B2 (en) * 2004-06-09 2007-04-10 Cumbre Pharmaceuticals Inc. Spiro-rifamycin derivatives targeting RNA polymerase
ES2246155B1 (en) * 2004-07-19 2007-03-16 Universidad De Oviedo NEW ESPIROPIPERIDILRIFAMICINAS.
EP1928890B1 (en) 2005-08-11 2013-04-03 Targanta Therapeutics Inc. Phosphonated rifamycins and uses thereof for the prevention and treatment of bone and joint infections
WO2008008480A2 (en) * 2006-07-12 2008-01-17 Cumbre Pharmaceuticals Inc. Nitroheteroaryl-containing rifamycin derivatives
CN100569778C (en) * 2006-12-05 2009-12-16 四川明欣药业有限责任公司 A kind of Rifabutin crystallization technique
US7884099B2 (en) * 2007-11-16 2011-02-08 Cumbre Ip Ventures, L.P. Quinolone carboxylic acid-substituted rifamycin derivatives
WO2010019511A2 (en) 2008-08-13 2010-02-18 Targanta Therapeutics Corp. Phosphonated rifamycins and uses thereof for the prevention and treatment of bone and joint infections
EP2890374B1 (en) 2012-08-30 2019-04-03 The Texas A&M University System Compositions and methods for drug-sensitization or inhibition of a cancer cell
PH12013000351A1 (en) 2013-11-22 2015-05-25 Joselle A Macrohon A versatile queuing management system and method
US20170202850A1 (en) 2014-07-21 2017-07-20 Hiroaki Serizawa Ophthalmic compositions of rifamycins and uses thereof
CN106279205B (en) * 2015-05-12 2020-07-21 重庆华邦胜凯制药有限公司 Process for the preparation of rifamycin S derivatives

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL130099C (en) * 1963-10-11
IT1056272B (en) * 1975-06-13 1982-01-30 Archifar Ind Chim Trentino PRODUCTS DERIVED FROM AROMATIC AMINES
DE2626296C2 (en) * 1975-06-13 1986-11-27 Farmitalia Carlo Erba S.p.A., Mailand/Milano Rifamycin compound and process for its preparation

Also Published As

Publication number Publication date
HK56083A (en) 1983-11-25
AU497602B2 (en) 1978-12-21
GB1542063A (en) 1979-03-14
DK145228B (en) 1982-10-11
ZA763256B (en) 1977-05-25
CS197271B1 (en) 1980-04-30
JPS6121957B2 (en) 1986-05-29
IE42998B1 (en) 1980-12-03
BE842883A (en) 1976-10-01
FI60208B (en) 1981-08-31
PT65208A (en) 1976-07-01
DK258076A (en) 1976-12-14
PH16410A (en) 1983-09-29
CH625524A5 (en) 1981-09-30
IL49701A0 (en) 1976-08-31
JPS5236683A (en) 1977-03-22
NO762026L (en) 1976-12-14
SU680649A3 (en) 1979-08-15
IT1056272B (en) 1982-01-30
SE7606640L (en) 1976-12-14
PL99493B1 (en) 1978-07-31
US4219478A (en) 1980-08-26
CA1059123A (en) 1979-07-24
FI761688A (en) 1976-12-14
NL177919B (en) 1985-07-16
IL49701A (en) 1979-10-31
YU39768B (en) 1985-04-30
PT65208B (en) 1977-11-23
ES449187A1 (en) 1977-07-16
IN143526B (en) 1977-12-17
NO148848B (en) 1983-09-19
US4086225A (en) 1978-04-25
NL177919C (en) 1985-12-16
AU1476976A (en) 1977-12-15
AR211127A1 (en) 1977-10-31
IE42998L (en) 1976-12-13
SE434057B (en) 1984-07-02
NO148848C (en) 1983-12-28
FR2314189B1 (en) 1980-10-31
FI60208C (en) 1981-12-10
HU171396B (en) 1978-01-28
YU140576A (en) 1982-06-30
NL7606370A (en) 1976-12-15
FR2314189A1 (en) 1977-01-07

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