DK1436280T3 - Fremgangsmåde til fremstilling af 4-(hydroxy)-[1,4']bipiperidinyl-1'-carboxylsyre-tert-butylester - Google Patents

Fremgangsmåde til fremstilling af 4-(hydroxy)-[1,4']bipiperidinyl-1'-carboxylsyre-tert-butylester

Info

Publication number
DK1436280T3
DK1436280T3 DK02773120T DK02773120T DK1436280T3 DK 1436280 T3 DK1436280 T3 DK 1436280T3 DK 02773120 T DK02773120 T DK 02773120T DK 02773120 T DK02773120 T DK 02773120T DK 1436280 T3 DK1436280 T3 DK 1436280T3
Authority
DK
Denmark
Prior art keywords
bipiperidinyl
hydroxy
carboxylic acid
butyl ester
acid tert
Prior art date
Application number
DK02773120T
Other languages
English (en)
Inventor
Philip O'keefe
Mark Purdie
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Application granted granted Critical
Publication of DK1436280T3 publication Critical patent/DK1436280T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40—Oxygen atoms
    • C07D211/44—Oxygen atoms attached in position 4
    • C07D211/46—Oxygen atoms attached in position 4 having a hydrogen atom as the second substituent in position 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Hydrogenated Pyridines (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK02773120T 2001-10-05 2002-10-02 Fremgangsmåde til fremstilling af 4-(hydroxy)-[1,4']bipiperidinyl-1'-carboxylsyre-tert-butylester DK1436280T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0124020.9A GB0124020D0 (en) 2001-10-05 2001-10-05 Chemical compounds
PCT/SE2002/001802 WO2003031433A1 (en) 2001-10-05 2002-10-02 A process for preparing 4-(hydroxy)-[1,4']bipiperidinyl-l'carboxylic acid tert-butyl ester

Publications (1)

Publication Number Publication Date
DK1436280T3 true DK1436280T3 (da) 2005-08-29

Family

ID=9923349

Family Applications (1)

Application Number Title Priority Date Filing Date
DK02773120T DK1436280T3 (da) 2001-10-05 2002-10-02 Fremgangsmåde til fremstilling af 4-(hydroxy)-[1,4']bipiperidinyl-1'-carboxylsyre-tert-butylester

Country Status (10)

Country Link
US (1) US7276609B2 (da)
EP (1) EP1436280B1 (da)
JP (1) JP2005509614A (da)
AT (1) ATE296822T1 (da)
DE (1) DE60204473T2 (da)
DK (1) DK1436280T3 (da)
ES (1) ES2240804T3 (da)
GB (1) GB0124020D0 (da)
PT (1) PT1436280E (da)
WO (1) WO2003031433A1 (da)

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE9703378D0 (sv) * 1997-09-18 1997-09-18 Astra Ab New compounds
WO1999052894A1 (fr) * 1998-04-09 1999-10-21 Meiji Seika Kaisha, Ltd. Composes heterocycliques a base d'azote anti-agregation plaquettaire et leur utilisation medicale
US6294554B1 (en) * 1999-09-22 2001-09-25 Schering Corporation Muscarinic antagonists
AR033517A1 (es) * 2000-04-08 2003-12-26 Astrazeneca Ab Derivados de piperidina, proceso para su preparacion y uso de estos derivados en la fabricacion de medicamentos

Also Published As

Publication number Publication date
ES2240804T3 (es) 2005-10-16
EP1436280A1 (en) 2004-07-14
ATE296822T1 (de) 2005-06-15
DE60204473T2 (de) 2006-05-11
WO2003031433A1 (en) 2003-04-17
PT1436280E (pt) 2005-09-30
US20040235895A1 (en) 2004-11-25
US7276609B2 (en) 2007-10-02
JP2005509614A (ja) 2005-04-14
DE60204473D1 (de) 2005-07-07
EP1436280B1 (en) 2005-06-01
GB0124020D0 (en) 2001-11-28

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