DK137539B - Fremgangsmade til fremstilling af 11beta-fluor-4-androsten-3-oner - Google Patents

Fremgangsmade til fremstilling af 11beta-fluor-4-androsten-3-oner

Info

Publication number
DK137539B
DK137539B DK78775AA DK78775A DK137539B DK 137539 B DK137539 B DK 137539B DK 78775A A DK78775A A DK 78775AA DK 78775 A DK78775 A DK 78775A DK 137539 B DK137539 B DK 137539B
Authority
DK
Denmark
Prior art keywords
oners
11beta
androsten
fluoro
procedure
Prior art date
Application number
DK78775AA
Other languages
English (en)
Other versions
DK78775A (da
DK137539C (da
Inventor
H Hofmeister
H Laurent
R Wiechert
K Annen
H Steinbeck
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Ag filed Critical Schering Ag
Publication of DK78775A publication Critical patent/DK78775A/da
Publication of DK137539B publication Critical patent/DK137539B/da
Application granted granted Critical
Publication of DK137539C publication Critical patent/DK137539C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0003Androstane derivatives
    • C07J1/0018Androstane derivatives substituted in position 17 beta, not substituted in position 17 alfa
    • C07J1/0022Androstane derivatives substituted in position 17 beta, not substituted in position 17 alfa the substituent being an OH group free esterified or etherified
    • C07J1/0029Ethers
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0003Androstane derivatives
    • C07J1/0011Androstane derivatives substituted in position 17 by a keto group
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0003Androstane derivatives
    • C07J1/0018Androstane derivatives substituted in position 17 beta, not substituted in position 17 alfa
    • C07J1/0022Androstane derivatives substituted in position 17 beta, not substituted in position 17 alfa the substituent being an OH group free esterified or etherified
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0003Androstane derivatives
    • C07J1/0018Androstane derivatives substituted in position 17 beta, not substituted in position 17 alfa
    • C07J1/0022Androstane derivatives substituted in position 17 beta, not substituted in position 17 alfa the substituent being an OH group free esterified or etherified
    • C07J1/0025Esters
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0003Androstane derivatives
    • C07J1/0033Androstane derivatives substituted in position 17 alfa and 17 beta
    • C07J1/0037Androstane derivatives substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being a saturated hydrocarbon group
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0003Androstane derivatives
    • C07J1/0033Androstane derivatives substituted in position 17 alfa and 17 beta
    • C07J1/004Androstane derivatives substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
    • C07J1/0048Alkynyl derivatives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J53/00Steroids in which the cyclopenta(a)hydrophenanthrene skeleton has been modified by condensation with a carbocyclic rings or by formation of an additional ring by means of a direct link between two ring carbon atoms, including carboxyclic rings fused to the cyclopenta(a)hydrophenanthrene skeleton are included in this class
    • C07J53/002Carbocyclic rings fused
    • C07J53/0043 membered carbocyclic rings
    • C07J53/0053 membered carbocyclic rings in position 12
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
DK78775A 1974-03-01 1975-02-27 Fremgangsmaade til fremstilling af 11beta-fluor-4-androsten-3-oner DK137539C (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2410443A DE2410443A1 (de) 1974-03-01 1974-03-01 11beta-fluor-androstene

Publications (3)

Publication Number Publication Date
DK78775A DK78775A (da) 1975-11-03
DK137539B true DK137539B (da) 1978-03-20
DK137539C DK137539C (da) 1978-09-04

Family

ID=5909131

Family Applications (1)

Application Number Title Priority Date Filing Date
DK78775A DK137539C (da) 1974-03-01 1975-02-27 Fremgangsmaade til fremstilling af 11beta-fluor-4-androsten-3-oner

Country Status (16)

Country Link
US (1) US3966713A (da)
JP (1) JPS50121259A (da)
BE (1) BE826139A (da)
CA (1) CA1037024A (da)
CS (1) CS181779B2 (da)
DD (1) DD118623A5 (da)
DE (1) DE2410443A1 (da)
DK (1) DK137539C (da)
ES (1) ES435204A1 (da)
FR (1) FR2262528B1 (da)
GB (1) GB1504410A (da)
HU (1) HU170643B (da)
IL (1) IL46712A0 (da)
NL (1) NL7502445A (da)
SE (1) SE7502239L (da)
SU (1) SU656529A3 (da)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4943579A (en) * 1987-10-06 1990-07-24 The United States Of America As Represented By The Secretary Of The Department Of Health And Human Services Water soluble prodrugs of camptothecin
IL146284A0 (en) 1999-05-04 2002-07-25 Strakan Ltd Androgen glycosides and pharmaceutical compositions containing the same
DE10104327A1 (de) 2001-01-24 2002-07-25 Schering Ag 11beta-Halogensteroide, deren Herstellung und Verwendung zur Herstellung von Arzneimitteln sowie 11beta-Halogensteroide enthaltende pharmazeutische Präparate
EP2265629B1 (en) * 2008-03-05 2015-06-24 Evestra, Inc. Bismethylene-17 carbolactones and related uses
EP2367808A4 (en) * 2008-11-25 2012-05-09 Evestra Inc PROGESTATIVE 3- (6,6-ETHYLENE-17b-HYDROXY-3-OXO-17a-PREGNA-4-EN-17a-YL) PROPIONIC ACID g-LACTONE

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3056807A (en) * 1961-10-09 1962-10-02 Upjohn Co Process for the preparation of fluorosteroids
US3875148A (en) * 1971-07-09 1975-04-01 Glaxo Lab Ltd 9{60 -unsubstituted-11{62 -bromo-19-norsteroids
US3767685A (en) * 1972-02-02 1973-10-23 Akzona Inc Novel 11beta-halo-steroids of the oestrane series

Also Published As

Publication number Publication date
HU170643B (da) 1977-07-28
GB1504410A (en) 1978-03-22
IL46712A0 (en) 1975-04-25
AU7855175A (en) 1976-08-26
DK78775A (da) 1975-11-03
SE7502239L (da) 1975-09-02
SU656529A3 (ru) 1979-04-05
FR2262528A1 (da) 1975-09-26
NL7502445A (nl) 1975-09-03
JPS50121259A (da) 1975-09-23
DE2410443A1 (de) 1975-09-11
BE826139A (fr) 1975-08-28
CA1037024A (en) 1978-08-22
DK137539C (da) 1978-09-04
DD118623A5 (da) 1976-03-12
US3966713A (en) 1976-06-29
CS181779B2 (en) 1978-03-31
FR2262528B1 (da) 1978-06-30
ES435204A1 (es) 1976-12-16

Similar Documents

Publication Publication Date Title
DK392675A (da) Fremgangsmade til fremstilling af substituerede puriner
DK487475A (da) Fremgangsmade til fremstilling af vandkveldende polyalkylenoxid
DK244875A (da) Fremgangsmade til fremstilling af chromanderivater
DK222375A (da) Fremgangsmade til fremstilling af alkyl-tert-butylethere
DK359275A (da) Fremgangsmade til fremstilling af mellemprodukter
DK235175A (da) Fremgangsmade til fremstilling af forbindelser med ergolinskelet
DK351875A (da) Fremgangsmade til fremstilling af 7-methoxy-6-thiatetracyliner
DK250175A (da) Fremgangsmade til fremstilling af n-cycloalkylmethyldecahydroisoquino-liner
DK349175A (da) Fremgangsmade til fremstilling af ketoner
DK313175A (da) Fremgangsmade til fremstilling af indoler
DK223175A (da) Fremgangsmade til fremstilling af pyridobenzodiazepinoner
DK225075A (da) Fremgangsmade til fremstilling af alfa-6--desoxy5-hydroxytetracyclin
DK442977A (da) Fremgangsmade til fremstilling af gamma-l-glutamyltaurin
DK139820C (da) Fremgangsmaade til fremstilling af moenomycin
DK409575A (da) Fremgangsmade til fremstilling af spanplader
DK547675A (da) Fremgangsmade til fremstilling af 6-methyl-8beta-substituerede methylergoliner
DK154890C (da) Fremgangsmaade til fremstilling af 7beta-acylamino-7alfa-alkoxycephalosporiner
DK344175A (da) Fremgangsmade til fremstilling af chromanderivater
DK590275A (da) Fremgangsmade til fremstilling af pinacolon
DK283476A (da) Fremgangsmade til fremstilling af beta-acylpyrroler
DK373475A (da) Fremgangsmade til optrekning af daser
DK253175A (da) Fremgangsmade til fremstilling af skumstoffer
DK492275A (da) Fremgangsmade til fremstilling af halogenantraquinoner
DK137539B (da) Fremgangsmade til fremstilling af 11beta-fluor-4-androsten-3-oner
DK535175A (da) Fremgangsmade til fremstilling af chromonforbindelser