DK135130B - Analogifremgangsmåde til fremstilling af 2-substituerede adenosinderivater eller syreadditionssalte deraf. - Google Patents

Analogifremgangsmåde til fremstilling af 2-substituerede adenosinderivater eller syreadditionssalte deraf.

Info

Publication number
DK135130B
DK135130B DK621371A DK621371A DK135130B DK 135130 B DK135130 B DK 135130B DK 621371 A DK621371 A DK 621371A DK 621371 A DK621371 A DK 621371A DK 135130 B DK135130 B DK 135130B
Authority
DK
Denmark
Prior art keywords
preparation
acid addition
addition salts
analogous process
adenosine derivatives
Prior art date
Application number
DK621371A
Other languages
Danish (da)
English (en)
Other versions
DK135130C (enrdf_load_stackoverflow
Inventor
Ryuji Marumoto
Kin-Ichi Imai
Yoshio Yoshioka
Mikio Honjo
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP12407770A external-priority patent/JPS5034039B1/ja
Priority claimed from DK461771AA external-priority patent/DK126043B/da
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Priority to DK621371A priority Critical patent/DK135130B/da
Priority to CA130,670A priority patent/CA965411A/en
Priority to HUTA001164 priority patent/HU164526B/hu
Priority to NL7117845A priority patent/NL7117845A/xx
Priority to SE1669271A priority patent/SE391337B/xx
Publication of DK135130B publication Critical patent/DK135130B/da
Application granted granted Critical
Publication of DK135130C publication Critical patent/DK135130C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16Purine radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Saccharide Compounds (AREA)
DK621371A 1970-12-28 1971-12-20 Analogifremgangsmåde til fremstilling af 2-substituerede adenosinderivater eller syreadditionssalte deraf. DK135130B (da)

Priority Applications (5)

Application Number Priority Date Filing Date Title
DK621371A DK135130B (da) 1970-12-28 1971-12-20 Analogifremgangsmåde til fremstilling af 2-substituerede adenosinderivater eller syreadditionssalte deraf.
CA130,670A CA965411A (en) 1970-12-28 1971-12-21 Method for the production of 2-substituted adenosine derivative
HUTA001164 HU164526B (enrdf_load_stackoverflow) 1970-12-28 1971-12-23
NL7117845A NL7117845A (en) 1970-12-28 1971-12-24 Vasodilatory and hypotensive 2-substd adenosine prepn - by reaction of ammonia and 2,6- disubstd nebularins
SE1669271A SE391337B (sv) 1970-12-28 1971-12-27 Sett att framstella 2-substituerade adenosinderivat

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP12407770A JPS5034039B1 (enrdf_load_stackoverflow) 1970-12-28 1970-12-28
DK461771AA DK126043B (da) 1970-09-25 1971-09-22 Analogifremgangsmåde til fremstilling af 2-substituerede adenosinderivater eller syreadditionssalte deraf.
DK621371A DK135130B (da) 1970-12-28 1971-12-20 Analogifremgangsmåde til fremstilling af 2-substituerede adenosinderivater eller syreadditionssalte deraf.

Publications (2)

Publication Number Publication Date
DK135130B true DK135130B (da) 1977-03-07
DK135130C DK135130C (enrdf_load_stackoverflow) 1977-08-01

Family

ID=27222004

Family Applications (1)

Application Number Title Priority Date Filing Date
DK621371A DK135130B (da) 1970-12-28 1971-12-20 Analogifremgangsmåde til fremstilling af 2-substituerede adenosinderivater eller syreadditionssalte deraf.

Country Status (5)

Country Link
CA (1) CA965411A (enrdf_load_stackoverflow)
DK (1) DK135130B (enrdf_load_stackoverflow)
HU (1) HU164526B (enrdf_load_stackoverflow)
NL (1) NL7117845A (enrdf_load_stackoverflow)
SE (1) SE391337B (enrdf_load_stackoverflow)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6214807B1 (en) 1999-06-22 2001-04-10 Cv Therapeutics, Inc. C-pyrazole 2A A receptor agonists
USRE47351E1 (en) 1999-06-22 2019-04-16 Gilead Sciences, Inc. 2-(N-pyrazolo)adenosines with application as adenosine A2A receptor agonists
US6180615B1 (en) 1999-06-22 2001-01-30 Cv Therapeutics, Inc. Propargyl phenyl ether A2A receptor agonists
US6403567B1 (en) 1999-06-22 2002-06-11 Cv Therapeutics, Inc. N-pyrazole A2A adenosine receptor agonists
US6440948B1 (en) * 1999-06-22 2002-08-27 Cv Therapeutics, Inc. Thiophene A2A receptor agonists
US20020012946A1 (en) 2000-02-23 2002-01-31 Luiz Belardinelli Method of identifying partial agonists of the A2A receptor
US8470801B2 (en) 2002-07-29 2013-06-25 Gilead Sciences, Inc. Myocardial perfusion imaging methods and compositions
MXPA05001123A (es) 2002-07-29 2005-04-29 Cv Therapeutics Inc Formacion de imagenes por perfusion de miocardio mediante el uso de agonistas receptores de a2a.
US20050020915A1 (en) 2002-07-29 2005-01-27 Cv Therapeutics, Inc. Myocardial perfusion imaging methods and compositions
CN101076343A (zh) 2004-10-20 2007-11-21 Cv医药有限公司 A2a腺苷受体激动剂的应用
US7732595B2 (en) 2006-02-03 2010-06-08 Gilead Palo Alto, Inc. Process for preparing an A2A-adenosine receptor agonist and its polymorphs

Also Published As

Publication number Publication date
HU164526B (enrdf_load_stackoverflow) 1974-02-28
DK135130C (enrdf_load_stackoverflow) 1977-08-01
NL7117845A (en) 1972-06-30
CA965411A (en) 1975-04-01
SE391337B (sv) 1977-02-14

Similar Documents

Publication Publication Date Title
DK124547B (da) Analogifremgangsmåde til fremstilling af (3-amino-2-hydroxy-propyloxy)-thiochromanderivater eller syreadditionssalte deraf.
DK129446B (da) Analogifremgangsmåde til fremstilling af fenoxyhydroxypropylaminer eller syreadditionssalte heraf.
DK139869B (da) Analogifremgangsmåde til fremstilling af phenyl-imidazolyl-alkansyrederivater eller salte deraf.
DK131858B (da) Analogifremgangsmåde til fremstilling af 4-amino-6-arylpyrimidin-forbindelser eller syreadditionssalte deraf.
DK138324B (da) Analogifremgangsmåde til fremstilling af piperazinsubstituerede isoindolinderivater eller syreadditionssalte deraf.
DK135278B (da) Analogifremgangsmåde til fremstilling af fenoksyisopropanolaminderivater eller syreadditionssalte deraf.
DK135130B (da) Analogifremgangsmåde til fremstilling af 2-substituerede adenosinderivater eller syreadditionssalte deraf.
DK126043B (da) Analogifremgangsmåde til fremstilling af 2-substituerede adenosinderivater eller syreadditionssalte deraf.
DK127116B (da) Analogifremgangsmåde til fremstilling af imidazolidinonderivater eller syreadditionssalte deraf.
DK129513B (da) Analogifremgangsmåde til fremstilling af basisk substituerede alkylidenaminooxyalkylcarboxylsyreestere eller syreadditionssalte deraf.
DK125245B (da) Fremgangsmåde til fremstilling af γpiperidinobutyrophenonderivater eller syreadditionssalte deraf.
DK129346B (da) Analogifremgangsmåde til fremstilling af imidazolderivater eller syreadditionssalte deraf.
DK125472B (da) Analogifremgangsmåde til fremstilling af pyrimidopyridazinderivater eller syreadditionssalte deraf.
DK126327B (da) Analogifremgangsmåde til fremstilling af derivater af p-aminoalkylbenzensulfonamid eller syreadditionssalte deraf.
DK129164B (da) Analogifremgangsmåde til fremstilling af 3-alkyl-5-aryloxymethylisoxazoler eller syreadditionssalte deraf.
DK137044B (da) Analogifremgangsmåde til fremstilling af 4,4-diphenylhexahydroazepinderivater eller syreadditionssalte deraf.
DK130288B (da) Analogifremgangsmåde til fremstilling af alkanolaminderivater eller syreadditionssalte deraf.
DK127431B (da) Analogifremgangsmåde til fremstilling af thiepinderivater eller syreadditionssalte deraf.
DK136242B (da) Analogifremgangsmåde til fremstilling af substituerede benzyloxyaminer eller deres syreadditionssalte.
DK127117B (da) Analogifremgangsmåde til fremstilling af imidazolidinonderivater eller syreadditionssalte deraf.
DK131147B (da) Fremgangsmåde til fremstilling af butyrophenonderivater eller syreadditionssalte deraf.
DK137834B (da) Analogifremgangsmåde til fremstilling af triazolobenzodiazepinderivater eller syreadditionssalte deraf.
DK127642B (da) Analogifremgangsmåde til fremstilling af benzodioxanderivater eller syreadditionssalte deraf.
DK127501B (da) Analogifremgangsmåde til fremstilling af substituerede phenoxyethylaminer eller deres syreadditionssalte.
DK131570B (da) Analogifremgangsmåde til fremstilling af thienylalkanderivater eller syreadditionssalte deraf.