DK1337529T3 - Heterocyclylalkylpiperidine derivatives, their preparation and preparations containing them - Google Patents

Heterocyclylalkylpiperidine derivatives, their preparation and preparations containing them

Info

Publication number
DK1337529T3
DK1337529T3 DK01996538T DK01996538T DK1337529T3 DK 1337529 T3 DK1337529 T3 DK 1337529T3 DK 01996538 T DK01996538 T DK 01996538T DK 01996538 T DK01996538 T DK 01996538T DK 1337529 T3 DK1337529 T3 DK 1337529T3
Authority
DK
Denmark
Prior art keywords
preparation
preparations containing
heterocyclylalkylpiperidine derivatives
heterocyclylalkylpiperidine
derivatives
Prior art date
Application number
DK01996538T
Other languages
Danish (da)
Inventor
Philippe Hubert
Eric Bacqu
Jean-Christophe Carry
Youssef El-Ahmad
Michel Evers
Jean-Luc Malleron
Serge Mignani
Guy Pantel
Michel Tabart
Fabrice Viviani
Original Assignee
Novexel
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novexel filed Critical Novexel
Application granted granted Critical
Publication of DK1337529T3 publication Critical patent/DK1337529T3/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20—Oxygen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
DK01996538T 2000-11-15 2001-11-14 Heterocyclylalkylpiperidine derivatives, their preparation and preparations containing them DK1337529T3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0014738A FR2816618B1 (en) 2000-11-15 2000-11-15 HETEROCYCLYLALCOYL PIPERIDINE DERIVATIVES, THEIR PREPARATION AND THE COMPOSITIONS CONTAINING THEM

Publications (1)

Publication Number Publication Date
DK1337529T3 true DK1337529T3 (en) 2006-12-18

Family

ID=8856503

Family Applications (1)

Application Number Title Priority Date Filing Date
DK01996538T DK1337529T3 (en) 2000-11-15 2001-11-14 Heterocyclylalkylpiperidine derivatives, their preparation and preparations containing them

Country Status (28)

Country Link
EP (2) EP1695964A1 (en)
JP (1) JP2004514661A (en)
KR (1) KR100849608B1 (en)
CN (1) CN1483031A (en)
AR (1) AR034006A1 (en)
AT (1) ATE337311T1 (en)
AU (2) AU1836502A (en)
BG (1) BG107793A (en)
BR (1) BR0115312A (en)
CA (1) CA2429311A1 (en)
CZ (1) CZ20031316A3 (en)
DE (1) DE60122567T2 (en)
DK (1) DK1337529T3 (en)
EA (1) EA200300568A1 (en)
EE (1) EE200300207A (en)
ES (1) ES2271119T3 (en)
FR (1) FR2816618B1 (en)
HR (1) HRP20030379A2 (en)
HU (1) HUP0303758A3 (en)
IL (1) IL155841A0 (en)
NO (2) NO20032187L (en)
PL (1) PL363004A1 (en)
PT (1) PT1337529E (en)
SK (1) SK5822003A3 (en)
TN (1) TNSN01160A1 (en)
WO (1) WO2002040474A2 (en)
YU (1) YU46803A (en)
ZA (1) ZA200303794B (en)

Families Citing this family (37)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL366335A1 (en) 2000-07-26 2005-01-24 Smithkline Beecham P.L.C. Aminopiperidine quinolines and their azaisosteric analogues with antibacterial activity
GB0101577D0 (en) 2001-01-22 2001-03-07 Smithkline Beecham Plc Compounds
GB0112836D0 (en) 2001-05-25 2001-07-18 Smithkline Beecham Plc Medicaments
GB0112834D0 (en) 2001-05-25 2001-07-18 Smithkline Beecham Plc Medicaments
GB0118238D0 (en) * 2001-07-26 2001-09-19 Smithkline Beecham Plc Medicaments
AU2003239302A1 (en) 2002-01-29 2003-09-02 Glaxo Group Limited Aminopiperidine compounds, process for their preparation, and pharmaceutical compositions containing them
TW200406410A (en) 2002-01-29 2004-05-01 Glaxo Group Ltd Compounds
TW200406413A (en) 2002-06-26 2004-05-01 Glaxo Group Ltd Compounds
AR040336A1 (en) 2002-06-26 2005-03-30 Glaxo Group Ltd PIPERIDINE COMPOUND, USE OF THE SAME FOR THE MANUFACTURE OF A MEDICINAL PRODUCT, PHARMACEUTICAL COMPOSITION THAT INCLUDES IT AND PROCEDURE TO PREPARE SUCH COMPOUND
FR2842807A1 (en) * 2002-07-23 2004-01-30 Aventis Pharma Sa QUINOLYL PROPYL PIPERIDINE DERIVATIVES, PROCESS AND PREPARATION INTERMEDIATES AND COMPOSITIONS COMPRISING THE SAME
GB0217294D0 (en) * 2002-07-25 2002-09-04 Glaxo Group Ltd Medicaments
FR2844268B1 (en) 2002-09-11 2004-10-22 Aventis Pharma Sa QUINOLYL PROPYL PIPERIDINE DERIVATIVES, PROCESSES AND INTERMEDIATES FOR THEIR PREPARATION, AND COMPOSITIONS CONTAINING THEM
FR2844270B1 (en) 2002-09-11 2006-05-19 Aventis Pharma Sa QUINOLYL PROPYL PIPERIDINE DERIVATIVES, THEIR PROCESS AND PREPARATION INTERMEDIATES AND THE COMPOSITIONS CONTAINING THEM
DE10256405A1 (en) * 2002-12-02 2004-06-17 Morphochem Aktiengesellschaft für kombinatorische Chemie New 4-substituted quinoline derivatives, useful for treating bacterial infections, optionally including additional ring nitrogens
DE60331849D1 (en) 2002-11-05 2010-05-06 Glaxosmithkline Llc ANTIBACTERIAL ACTIVE SUBSTANCES
EP1567520B1 (en) 2002-12-04 2008-10-15 Glaxo Group Limited Quinolines and nitrogenated derivatives thereof and their use as antibacterial agents
US7232833B2 (en) 2003-03-28 2007-06-19 Novexel 4-substituted quinoline derivatives, method and intermediates for their preparation and pharmaceutical compositions containing them
FR2852954B1 (en) * 2003-03-28 2006-07-14 Aventis Pharma Sa QUINOLINE-4-SUBSTITUTED DERIVATIVES, METHODS AND PREPARATION INTERMEDIATES THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
FR2862301B1 (en) * 2003-11-17 2007-12-21 Aventis Pharma Sa NEW PROCESS FOR THE PREPARATION OF 3-FLUORINATED QUINOLINES
FR2867472B1 (en) * 2004-03-12 2008-07-18 Aventis Pharma Sa QUINOLINE-4-SUBSTITUTED DERIVATIVES, METHODS AND PREPARATION INTERMEDIATES THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
US7592334B2 (en) 2005-01-25 2009-09-22 Glaxo Group Limited Antibacterial agents
US7605169B2 (en) 2005-01-25 2009-10-20 Glaxo Group Limited Antibacterial agents
EP1845995A4 (en) 2005-01-25 2010-03-03 Glaxo Group Ltd Antibacterial agents
JP2008528586A (en) 2005-01-25 2008-07-31 グラクソ グループ リミテッド Antibacterial agent
MX2007010572A (en) 2005-03-01 2007-10-04 Wyeth Corp Cinnoline compounds and their use as liver x receptor modilators.
MY150958A (en) * 2005-06-16 2014-03-31 Astrazeneca Ab Compounds for the treatment of multi-drug resistant bacterial infections
JP2009524643A (en) 2006-01-26 2009-07-02 アクテリオン ファーマシューティカルズ リミテッド Tetrahydropyran antibiotics
JP2009532423A (en) 2006-04-06 2009-09-10 グラクソ グループ リミテッド Pyrrolo-quinoxalinone derivatives as antibacterial agents
EP1992628A1 (en) 2007-05-18 2008-11-19 Glaxo Group Limited Derivatives and analogs of N-ethylquinolones and N-ethylazaquinolones
EP2167494B1 (en) 2007-06-15 2011-08-17 Actelion Pharmaceuticals Ltd. 3-amino-6-(1-amino-ethyl)-tetrahydropyran derivatives
EP2080761A1 (en) 2008-01-18 2009-07-22 Glaxo Group Limited Compounds
WO2010043714A1 (en) 2008-10-17 2010-04-22 Glaxo Group Limited Tricyclic nitrogen compounds used as antibacterials
ES2561631T3 (en) 2009-01-15 2016-02-29 Glaxo Group Limited Naphthyridine-2 (1H) -one compounds useful as antibacterial agents
WO2014027045A1 (en) * 2012-08-15 2014-02-20 Glaxo Group Limited Chemical process
EP3182973B1 (en) 2014-08-22 2019-09-18 GlaxoSmithKline Intellectual Property Development Limited Tricyclic nitrogen containing compounds for treating neisseria gonorrhoea infection
WO2016138988A1 (en) * 2015-03-02 2016-09-09 University Of Copenhagen Piperazine inhibitors of bacterial gyrase and topoisomerase iv
TW201722965A (en) 2015-08-16 2017-07-01 葛蘭素史密斯克藍智慧財產發展有限公司 Compounds for use in antibacterial applications

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL7908031A (en) 1979-11-01 1981-06-01 Acf Chemiefarma Nv NEW QUINOLINE DERIVATIVES AND PHARMACEUTICAL PREPARATIONS CONTAINING SUCH A COMPOUND AND METHOD FOR PREPARING THESE COMPOUNDS.
JPH0239546A (en) 1988-07-29 1990-02-08 Origin Electric Co Ltd Manufacture of hybrid integrated circuit
AU623474B2 (en) 1989-01-16 1992-05-14 Laboratoire Roger Bellon New benzo(1,8)naphthyridine derivatives, their preparation and compositions containing them
AU2717899A (en) * 1998-01-26 1999-08-09 Smithkline Beecham Plc Quinoline derivatives as antibacterials
WO2000043383A1 (en) * 1999-01-20 2000-07-27 Smithkline Beecham P.L.C. Piperidinylquinolines as protein tyrosine kinase inhibitors
FR2852954B1 (en) * 2003-03-28 2006-07-14 Aventis Pharma Sa QUINOLINE-4-SUBSTITUTED DERIVATIVES, METHODS AND PREPARATION INTERMEDIATES THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM

Also Published As

Publication number Publication date
HRP20030379A2 (en) 2005-04-30
FR2816618A1 (en) 2002-05-17
SK5822003A3 (en) 2004-06-08
EP1695964A1 (en) 2006-08-30
BG107793A (en) 2004-08-31
CZ20031316A3 (en) 2003-10-15
AU2002218365B2 (en) 2007-07-05
KR20030060934A (en) 2003-07-16
EE200300207A (en) 2003-08-15
ATE337311T1 (en) 2006-09-15
AR034006A1 (en) 2004-01-21
KR100849608B1 (en) 2008-07-31
PL363004A1 (en) 2004-11-15
WO2002040474A2 (en) 2002-05-23
NO20072142L (en) 2007-04-25
TNSN01160A1 (en) 2005-11-10
PT1337529E (en) 2006-12-29
ZA200303794B (en) 2004-06-29
YU46803A (en) 2006-05-25
WO2002040474A3 (en) 2002-10-31
HUP0303758A2 (en) 2004-03-01
ES2271119T3 (en) 2007-04-16
NO20032187L (en) 2003-06-26
CN1483031A (en) 2004-03-17
DE60122567D1 (en) 2006-10-05
BR0115312A (en) 2003-09-23
AU1836502A (en) 2002-05-27
FR2816618B1 (en) 2002-12-27
EP1337529A2 (en) 2003-08-27
EA200300568A1 (en) 2003-12-25
CA2429311A1 (en) 2002-05-23
EP1337529B1 (en) 2006-08-23
IL155841A0 (en) 2003-12-23
NO20032187D0 (en) 2003-05-14
DE60122567T2 (en) 2007-08-23
JP2004514661A (en) 2004-05-20
HUP0303758A3 (en) 2009-08-28

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