DK131033B - Analogifremgangsmåde til fremstilling af kaliumsalte af 2-phenyl-6-sulfamyl-7-chlor-1,2,3,4-tetrahydro-4-quinazolinon. - Google Patents
Analogifremgangsmåde til fremstilling af kaliumsalte af 2-phenyl-6-sulfamyl-7-chlor-1,2,3,4-tetrahydro-4-quinazolinon.Info
- Publication number
- DK131033B DK131033B DK247673AA DK247673A DK131033B DK 131033 B DK131033 B DK 131033B DK 247673A A DK247673A A DK 247673AA DK 247673 A DK247673 A DK 247673A DK 131033 B DK131033 B DK 131033B
- Authority
- DK
- Denmark
- Prior art keywords
- sulfamyl
- quinazolinone
- tetrahydro
- chloro
- phenyl
- Prior art date
Links
- DBDTUXMDTSTPQZ-UHFFFAOYSA-N fenquizone Chemical class N1C=2C=C(Cl)C(S(=O)(=O)N)=CC=2C(=O)NC1C1=CC=CC=C1 DBDTUXMDTSTPQZ-UHFFFAOYSA-N 0.000 title 1
- 159000000001 potassium salts Chemical class 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
- C07D239/88—Oxygen atoms
- C07D239/91—Oxygen atoms with aryl or aralkyl radicals attached in position 2 or 3
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT2392572 | 1972-05-05 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DK131033B true DK131033B (da) | 1975-05-20 |
| DK131033C DK131033C (enExample) | 1975-10-06 |
Family
ID=11210914
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK247673AA DK131033B (da) | 1972-05-05 | 1973-05-04 | Analogifremgangsmåde til fremstilling af kaliumsalte af 2-phenyl-6-sulfamyl-7-chlor-1,2,3,4-tetrahydro-4-quinazolinon. |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US3870720A (enExample) |
| JP (1) | JPS49132221A (enExample) |
| AU (1) | AU469087B2 (enExample) |
| BE (1) | BE799087A (enExample) |
| CA (1) | CA982578A (enExample) |
| DE (1) | DE2322699C2 (enExample) |
| DK (1) | DK131033B (enExample) |
| FR (1) | FR2183806B1 (enExample) |
| GB (1) | GB1413008A (enExample) |
| NL (1) | NL7306164A (enExample) |
| SE (1) | SE400768B (enExample) |
| ZA (1) | ZA732937B (enExample) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN1681495B (zh) | 2002-08-19 | 2010-05-12 | 辉瑞产品公司 | 用于治疗过度增生性疾病的组合物 |
| US20060063803A1 (en) * | 2004-09-23 | 2006-03-23 | Pfizer Inc | 4-Amino substituted-2-substituted-1,2,3,4-tetrahydroquinoline compounds |
| US7741317B2 (en) | 2005-10-21 | 2010-06-22 | Bristol-Myers Squibb Company | LXR modulators |
| US7888376B2 (en) | 2005-11-23 | 2011-02-15 | Bristol-Myers Squibb Company | Heterocyclic CETP inhibitors |
| US8404896B2 (en) | 2006-12-01 | 2013-03-26 | Bristol-Myers Squibb Company | N-((3-benzyl)-2,2-(bis-phenyl)-propan-1-amine derivatives as CETP inhibitors for the treatment of atherosclerosis and cardiovascular diseases |
| BR112015026513A2 (pt) | 2013-04-17 | 2017-07-25 | Pfizer | derivados de n-piperidin-3-ilbenzamida para tratar as doenças cardiovasculares |
| WO2016055901A1 (en) | 2014-10-08 | 2016-04-14 | Pfizer Inc. | Substituted amide compounds |
| RS66416B1 (sr) | 2019-01-18 | 2025-02-28 | Astrazeneca Ab | 6'-[[(1s,3s)-3-[[5-(difluorometoksi)-2-pirimidinil]amino]ciklopentil]amino][1(2h),3'-bipiridin]-2-on kao inhibitor pcsk9 i metode njegove primene |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2952680A (en) * | 1960-09-13 | Derivatives of x-quevazolone | ||
| US987847A (en) * | 1910-04-12 | 1911-03-28 | Rubin W Weeks | Harness. |
| US3440244A (en) * | 1958-02-17 | 1969-04-22 | Pfizer & Co C | 3,6-disubstituted-7-sulfamyl-1,2,4-benzthiazide-1,1-dioxides |
| US3072656A (en) * | 1960-01-22 | 1963-01-08 | Ciba Geigy Corp | 2-cycloaliphatic-6-sulfamyl-7-halo(or trihalomethyl)-1, 2, 3, 4-tetrahydro-4-quinazolones |
| US3360518A (en) * | 1966-01-03 | 1967-12-26 | Wallace & Tiernan Inc | Tetrahydro-halo-sulfamyl quinazolinones |
-
1973
- 1973-05-01 ZA ZA732937A patent/ZA732937B/xx unknown
- 1973-05-02 US US356403A patent/US3870720A/en not_active Expired - Lifetime
- 1973-05-03 AU AU55161/73A patent/AU469087B2/en not_active Expired
- 1973-05-03 NL NL7306164A patent/NL7306164A/xx unknown
- 1973-05-03 JP JP48049593A patent/JPS49132221A/ja active Pending
- 1973-05-04 DK DK247673AA patent/DK131033B/da not_active IP Right Cessation
- 1973-05-04 FR FR7316142A patent/FR2183806B1/fr not_active Expired
- 1973-05-04 BE BE130734A patent/BE799087A/xx unknown
- 1973-05-04 SE SE7306244A patent/SE400768B/xx unknown
- 1973-05-04 CA CA171,105A patent/CA982578A/en not_active Expired
- 1973-05-05 DE DE2322699A patent/DE2322699C2/de not_active Expired
- 1973-05-07 GB GB2165173A patent/GB1413008A/en not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| SE400768B (sv) | 1978-04-10 |
| CA982578A (en) | 1976-01-27 |
| FR2183806A1 (enExample) | 1973-12-21 |
| NL7306164A (enExample) | 1973-11-07 |
| BE799087A (fr) | 1973-08-31 |
| ZA732937B (en) | 1974-03-27 |
| DE2322699A1 (de) | 1974-01-10 |
| AU469087B2 (en) | 1976-02-05 |
| DE2322699C2 (de) | 1983-10-27 |
| JPS49132221A (enExample) | 1974-12-18 |
| AU5516173A (en) | 1974-11-07 |
| DK131033C (enExample) | 1975-10-06 |
| FR2183806B1 (enExample) | 1976-05-14 |
| GB1413008A (en) | 1975-11-05 |
| US3870720A (en) | 1975-03-11 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PBP | Patent lapsed |