DK125705B - Analogifremgangsmåde til fremstilling af mod protozoinfektioner virksomme amidinourinstoffer eller syreadditionssalte heraf. - Google Patents

Analogifremgangsmåde til fremstilling af mod protozoinfektioner virksomme amidinourinstoffer eller syreadditionssalte heraf.

Info

Publication number
DK125705B
DK125705B DK349067AA DK349067A DK125705B DK 125705 B DK125705 B DK 125705B DK 349067A A DK349067A A DK 349067AA DK 349067 A DK349067 A DK 349067A DK 125705 B DK125705 B DK 125705B
Authority
DK
Denmark
Prior art keywords
amidinourine
substances
preparation
acid addition
addition salts
Prior art date
Application number
DK349067AA
Other languages
Danish (da)
English (en)
Inventor
L Walls
Original Assignee
Wellcome Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wellcome Found filed Critical Wellcome Found
Publication of DK125705B publication Critical patent/DK125705B/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C279/00Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups
    • C07C279/20Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups containing any of the groups, X being a hetero atom, Y being any atom, e.g. acylguanidines
    • C07C279/24Y being a hetero atom
    • C07C279/26X and Y being nitrogen atoms, i.e. biguanides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Structures Of Non-Positive Displacement Pumps (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK349067AA 1966-07-07 1967-07-06 Analogifremgangsmåde til fremstilling af mod protozoinfektioner virksomme amidinourinstoffer eller syreadditionssalte heraf. DK125705B (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB3047966 1966-07-07
GB19028/67A GB1194835A (en) 1966-07-07 1966-07-07 Novel 1-Amidino-3-Phenyl-Urea Derivatives, the preparation thereof and Compositions containing the same
GB5654666 1966-12-16
GB539167 1967-02-03

Publications (1)

Publication Number Publication Date
DK125705B true DK125705B (da) 1973-03-26

Family

ID=27447446

Family Applications (1)

Application Number Title Priority Date Filing Date
DK349067AA DK125705B (da) 1966-07-07 1967-07-06 Analogifremgangsmåde til fremstilling af mod protozoinfektioner virksomme amidinourinstoffer eller syreadditionssalte heraf.

Country Status (15)

Country Link
US (2) US3539616A (no)
BE (1) BE700895A (no)
CA (1) CA947316A (no)
CH (5) CH500952A (no)
DE (2) DE1793745A1 (no)
DK (1) DK125705B (no)
FR (2) FR1548340A (no)
GB (1) GB1194835A (no)
IL (1) IL28189A (no)
LU (1) LU54053A1 (no)
MC (1) MC666A1 (no)
NL (1) NL6709484A (no)
NO (1) NO126225B (no)
OA (1) OA02467A (no)
SE (1) SE330010B (no)

Families Citing this family (29)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3761597A (en) * 1967-06-30 1973-09-25 L Walls 1-amidino-3-(substituted-phenyl) urea antimalarial composition and method of use
IL37047A0 (en) * 1970-06-30 1971-08-25 Wellcome Found Substituted amidines,their preparation and pharmaceutical compositions containing them
US4488993A (en) * 1972-09-22 1984-12-18 William H. Rorer, Inc. Amidinoureas
US4220658A (en) * 1972-09-22 1980-09-02 William H. Rorer, Inc. Treatment of hypertension with amidinoureas
US4025652A (en) * 1975-03-31 1977-05-24 William H. Rorer, Inc. Amidinoureas
US4326074A (en) * 1972-09-22 1982-04-20 William H. Rorer, Inc. Amidinoureas
FR2223361B1 (no) * 1973-03-27 1977-04-29 Philagro Sa
JPS5646157B2 (no) * 1973-06-05 1981-10-31
US4060635A (en) * 1975-03-31 1977-11-29 William H. Rorer, Inc. Amidinoureas for treating diarrhea
ZA743750B (en) * 1973-07-16 1975-06-25 Rorer Inc William H Amindinoureas
US4150154A (en) * 1975-03-03 1979-04-17 William H. Rorer, Inc. Amidinoureas
US4216229A (en) * 1973-07-16 1980-08-05 William H. Rorer, Inc. Method for treating gastrointestinal hyperacidity or ulceration with amidinoureas
US4283555A (en) * 1973-07-16 1981-08-11 William H. Rorer, Inc. Amidinoureas
FR2237625B1 (no) * 1973-07-16 1978-07-28 Rorer Inc William H
US4216230A (en) * 1973-07-16 1980-08-05 William H. Rorer, Inc. Method for alleviating hypertension with amidinoureas
US4204000A (en) * 1975-03-31 1980-05-20 William H. Rorer, Inc. Anti-ulcer amidinoureas
US4203920A (en) * 1975-03-31 1980-05-20 William H. Rorer, Inc. Amidinoureas
US4242337A (en) * 1976-03-30 1980-12-30 William H. Rorer, Inc. Method for treatment of diarrheal disease conditions or symptons in mammals
US4242339A (en) * 1976-03-30 1980-12-30 William H. Rorer, Inc. Method for treatment of gastrointestinal spasmodic disease conditions or symptoms in mammals
US4058557A (en) * 1976-03-30 1977-11-15 William H. Rorer, Inc. Amidinoureas
US4353842A (en) * 1978-09-14 1982-10-12 William H. Rorer, Inc. Amidinoureas
US4440949A (en) * 1979-01-08 1984-04-03 William H. Rorer, Inc. Amidinoureas
US4340609A (en) * 1980-01-02 1982-07-20 William H. Rorer, Inc. Amidinourea derivative veterinary compositions for suppression of parasitemia
JPS58501468A (ja) * 1981-08-24 1983-09-01 ロウラ− インタ−ナシヨナル (オ−バ−シ−ズ) インコ−ポレ−テツド 複素環アミジノ置換尿素およびそれらの薬剤利用
JPS62501839A (ja) * 1985-02-15 1987-07-23 ロウラ− インタ−ナシヨナル(オ−バ−シ−ズ) インコ−ポレ−テツド アミジノ尿素の製造法および医薬用組成物
ES2110667T3 (es) * 1993-08-18 1998-02-16 Bayer Ag N-cianoaril-heterociclos nitrogenados.
DE4412079A1 (de) * 1993-08-18 1995-02-23 Bayer Ag N-Cyanoaryl-Stickstoffheterocyclen
US5681794A (en) * 1993-08-18 1997-10-28 Bayer Aktiengesellschaft N-cyanoaryl-nitrogen heterocycles
DE4335438A1 (de) * 1993-10-18 1995-04-20 Bayer Ag 4-Cyanophenyliminoheterocyclen

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3119867A (en) * 1962-01-26 1964-01-28 Clairol Inc Amino, nitro-phenyl-biguanides and amino, nitro-phenyl; guanyl-ureas

Also Published As

Publication number Publication date
FR7055M (no) 1969-06-23
GB1194835A (en) 1970-06-10
NL6709484A (no) 1968-01-08
CH500952A (de) 1970-12-31
DE1668843A1 (de) 1972-02-24
CH554318A (de) 1974-09-30
LU54053A1 (no) 1968-03-12
US3539616A (en) 1970-11-10
CA947316A (en) 1974-05-14
NO126225B (no) 1973-01-08
FR1548340A (no) 1968-12-06
CH501599A (de) 1971-01-15
DE1793745A1 (de) 1973-05-30
US3784582A (en) 1974-01-08
SE330010B (no) 1970-11-02
MC666A1 (fr) 1968-04-01
OA02467A (fr) 1970-05-05
IL28189A (en) 1971-04-28
BE700895A (no) 1968-01-04
CH501597A (de) 1971-01-15
CH501598A (de) 1971-01-15

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