DK123405B - Analogifremgangsmåde til fremstilling af et n-alkylsulfamat af tetracyclin. - Google Patents

Analogifremgangsmåde til fremstilling af et n-alkylsulfamat af tetracyclin.

Info

Publication number
DK123405B
DK123405B DK262468AA DK262468A DK123405B DK 123405 B DK123405 B DK 123405B DK 262468A A DK262468A A DK 262468AA DK 262468 A DK262468 A DK 262468A DK 123405 B DK123405 B DK 123405B
Authority
DK
Denmark
Prior art keywords
alkylsulfamate
tetracycline
preparation
analogous process
analogous
Prior art date
Application number
DK262468AA
Other languages
English (en)
Inventor
C Vazquez
Original Assignee
Hosbon Sa Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hosbon Sa Lab filed Critical Hosbon Sa Lab
Publication of DK123405B publication Critical patent/DK123405B/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/46Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with hetero atoms directly attached to the ring nitrogen atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/65Tetracyclines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C237/00Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
    • C07C237/24Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring of the carbon skeleton
    • C07C237/26Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring of the carbon skeleton of a ring being part of a condensed ring system formed by at least four rings, e.g. tetracycline
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38Nitrogen atoms
    • C07D277/42Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00Systems containing at least three condensed rings
    • C07C2603/02Ortho- or ortho- and peri-condensed systems
    • C07C2603/40Ortho- or ortho- and peri-condensed systems containing four condensed rings
    • C07C2603/42Ortho- or ortho- and peri-condensed systems containing four condensed rings containing only six-membered rings
    • C07C2603/44Naphthacenes; Hydrogenated naphthacenes
    • C07C2603/461,4,4a,5,5a,6,11,12a- Octahydronaphthacenes, e.g. tetracyclines
DK262468AA 1967-06-06 1968-06-06 Analogifremgangsmåde til fremstilling af et n-alkylsulfamat af tetracyclin. DK123405B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR109212A FR6476M (da) 1967-06-06 1967-06-06

Publications (1)

Publication Number Publication Date
DK123405B true DK123405B (da) 1972-06-19

Family

ID=8632381

Family Applications (1)

Application Number Title Priority Date Filing Date
DK262468AA DK123405B (da) 1967-06-06 1968-06-06 Analogifremgangsmåde til fremstilling af et n-alkylsulfamat af tetracyclin.

Country Status (9)

Country Link
US (2) US3536759A (da)
BE (1) BE716159A (da)
BR (1) BR6899499D0 (da)
CH (1) CH477406A (da)
DE (1) DE1767701A1 (da)
DK (1) DK123405B (da)
ES (1) ES354173A1 (da)
FR (1) FR6476M (da)
SE (1) SE352339B (da)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1997005126A1 (en) * 1995-07-29 1997-02-13 Smithkline Beecham Plc Mupirocinsulfamates with antibacterial activity
DE10114364A1 (de) 2001-03-22 2002-10-02 Heraeus Kulzer Gmbh & Co Kg Verfahren zur Herstellung von antibiotischen Kompositen
DE10114245A1 (de) * 2001-03-22 2002-10-02 Heraeus Kulzer Gmbh & Co Kg Herstellung und Verwendung einer Antibiotikum-/Antibiotika-Zubereitung
DE10114244A1 (de) 2001-03-22 2002-10-02 Heraeus Kulzer Gmbh & Co Kg Antibiotikum-/Antibiotika-Zubereitung mit retardierender Wirkstofffreisetzung
DE10227938B4 (de) 2002-06-21 2006-07-20 Heraeus Kulzer Gmbh Pharmazeutische Zubereitung, Verfahren zu ihrer Herstellung sowie deren Verwendung

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2607M (fr) * 1963-01-30 1964-06-22 Soc Ind Fab Antibiotiques Sifa Nouveau dérivé de la tétracycline.

Also Published As

Publication number Publication date
FR6476M (da) 1968-11-18
CH477406A (fr) 1969-08-31
DE1767701A1 (de) 1970-01-02
SE352339B (da) 1972-12-27
US3658989A (en) 1972-04-25
ES354173A1 (es) 1969-10-16
US3536759A (en) 1970-10-27
BR6899499D0 (pt) 1973-12-27
BE716159A (da) 1968-11-04

Similar Documents

Publication Publication Date Title
DK133618B (da) Analogifremgangsmåde til fremstilling af 1-hydroxyaryl-2-aminoalkanoler.
DK137232B (da) Analogifremgangsmåde til fremstilling af phenylethanolaminer.
DK122222B (da) Fremgangsmåde til fremstilling af alk-3-en-1-oler.
DK133783B (da) Fremgangsmåde til fremstilling af 7-halogen-7-desoxy-1-thio-alfa-D-galacto-octopyranosider.
DK120698B (da) Analogifremgangsmåde til fremstilling af acetylguanidiner.
DK124080B (da) Fremgangsmåde til fremstilling af D-6-metyl-8-cyanmetylergolin.
DK119307B (da) Fremgangsmåde til fremstilling af ketonitriler.
DK136033B (da) Fremgangsmåde til fremstilling af indolyl-3-eddikesyrer.
DK122758B (da) Fremgangsmåde til fremstilling af α-methyl-multicyclo-methylaminer.
DK123405B (da) Analogifremgangsmåde til fremstilling af et n-alkylsulfamat af tetracyclin.
DK117954B (da) Fremgangsmåde til fremstilling af 3-amino-2-cyanoacrylamid.
DK123100B (da) Fremgangsmåde til fremstilling af N-tritylimidazoler.
DK122522B (da) Fremgangsmåde til fremstilling af dichlorquinoliner.
DK115551B (da) Fremgangsmåde til fremstilling af 6-aminouracil-5-carbonamid-N-sulfonamider.
DK119976B (da) Analogifremgangsmåde til fremstilling af 18-methyl-19-nor-17α-hydroxyprogesteroner og -17-estere deraf.
DK114063B (da) Fremgangsmåde til fremstilling af 1-methyl-2-isopropyl-5-nitro-imidazol.
DK120344B (da) Fremgangsmåde til fremstilling af 5-benzyl-pyrimidiner.
DK122666B (da) Analogifremgangsmåde til fremstilling af hydrocortison-17-cyclopentancorboxylat.
DK117568B (da) Analogifremgangsmåde til fremstilling af ftalazino-ftalazindioner.
DK126378B (da) Analogifremgangsmåde til fremstilling af 17α-acyloxy-9α-chlor-11β-hydroxy-progesteroner.
DK119830B (da) Analogifremgangsmåde til fremstilling af arylsulfonylsemicarbazider.
DK123476B (da) Fremgangsmåde til fremstilling af 3-oxo-A-nor-B-homo-estra-5(10)-ener.
DK114626B (da) Fremgangsmåde til fremstilling af 2-substitueret-4-amino-5-acylamidometylpyrimidin.
DK126200B (da) Analogifremgangsmåde til fremstilling af 2-amino-3-carbamoyl-quinoxalin-di-N-oxider.
DK122278B (da) Analogifremgangsmåde til fremstilling af 3-oxogonatriener.