DK121085B - Analogifremgangsmåde til fremstilling af 2,4-diamino-6-(substitueret acylamino)-quinazolinforbindelser eller salte heraf. - Google Patents

Analogifremgangsmåde til fremstilling af 2,4-diamino-6-(substitueret acylamino)-quinazolinforbindelser eller salte heraf.

Info

Publication number
DK121085B
DK121085B DK434968AA DK434968A DK121085B DK 121085 B DK121085 B DK 121085B DK 434968A A DK434968A A DK 434968AA DK 434968 A DK434968 A DK 434968A DK 121085 B DK121085 B DK 121085B
Authority
DK
Denmark
Prior art keywords
diamino
salts
preparation
analogous process
quinazoline compounds
Prior art date
Application number
DK434968AA
Other languages
Danish (da)
English (en)
Inventor
J Davoll
Original Assignee
Parke Davis & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Parke Davis & Co filed Critical Parke Davis & Co
Publication of DK121085B publication Critical patent/DK121085B/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88Oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/86Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94Nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/95Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK434968AA 1967-09-11 1968-09-10 Analogifremgangsmåde til fremstilling af 2,4-diamino-6-(substitueret acylamino)-quinazolinforbindelser eller salte heraf. DK121085B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB41436/67A GB1161644A (en) 1967-09-11 1967-09-11 Quinazoline Compounds and process means for producing the same

Publications (1)

Publication Number Publication Date
DK121085B true DK121085B (da) 1971-09-06

Family

ID=10419677

Family Applications (1)

Application Number Title Priority Date Filing Date
DK434968AA DK121085B (da) 1967-09-11 1968-09-10 Analogifremgangsmåde til fremstilling af 2,4-diamino-6-(substitueret acylamino)-quinazolinforbindelser eller salte heraf.

Country Status (12)

Country Link
US (1) US3546224A (fr)
BE (1) BE720645A (fr)
CH (1) CH491931A (fr)
DE (1) DE1795309B2 (fr)
DK (1) DK121085B (fr)
ES (1) ES357983A1 (fr)
FR (1) FR1589711A (fr)
GB (1) GB1161644A (fr)
IL (1) IL30614A (fr)
NL (1) NL6812978A (fr)
SE (1) SE336797B (fr)
YU (1) YU32091B (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5430148A (en) * 1992-03-31 1995-07-04 Agouron Pharmaceuticals, Inc. Antiproliferative quinazolines
IL108630A0 (en) * 1993-02-18 1994-05-30 Fmc Corp Insecticidal substituted 2,4-diaminoquinazolines

Also Published As

Publication number Publication date
ES357983A1 (es) 1970-04-01
SE336797B (fr) 1971-07-19
YU32091B (en) 1974-04-30
IL30614A (en) 1972-05-30
CH491931A (fr) 1970-06-15
GB1161644A (en) 1969-08-13
US3546224A (en) 1970-12-08
DE1795309C3 (fr) 1974-10-24
DE1795309A1 (de) 1972-04-13
IL30614A0 (en) 1968-10-24
YU211068A (en) 1973-10-31
DE1795309B2 (de) 1974-03-14
NL6812978A (fr) 1969-03-13
BE720645A (fr) 1969-02-17
FR1589711A (fr) 1970-04-06

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