DK120337B - Fremgangsmåde til fremstilling af terapeutisk aktive 3-keto-6-halogen-9β10α-Δ<4,6>-steroiddiener af androstan- eller pregnanrækken. - Google Patents
Fremgangsmåde til fremstilling af terapeutisk aktive 3-keto-6-halogen-9β10α-Δ<4,6>-steroiddiener af androstan- eller pregnanrækken.Info
- Publication number
- DK120337B DK120337B DK319165AA DK319165A DK120337B DK 120337 B DK120337 B DK 120337B DK 319165A A DK319165A A DK 319165AA DK 319165 A DK319165 A DK 319165A DK 120337 B DK120337 B DK 120337B
- Authority
- DK
- Denmark
- Prior art keywords
- androstane
- keto
- halogen
- preparation
- therapeutically active
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A61K31/568—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A61K31/568—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone
- A61K31/569—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone substituted in position 17 alpha, e.g. ethisterone
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J15/00—Stereochemically pure steroids containing carbon, hydrogen, halogen or oxygen having a partially or totally inverted skeleton, e.g. retrosteroids, L-isomers
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J5/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J75/00—Processes for the preparation of steroids in general
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Steroid Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB291965A GB1139411A (en) | 1965-01-22 | 1965-01-22 | Preparation of 10-‡-methyl steroids |
| CH846564A CH454842A (de) | 1965-05-31 | 1965-05-31 | Verfahren zur Herstellung von neuen 9B,10a-Steroiden |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK120337B true DK120337B (da) | 1971-05-17 |
Family
ID=25703347
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK319165AA DK120337B (da) | 1965-01-22 | 1965-06-23 | Fremgangsmåde til fremstilling af terapeutisk aktive 3-keto-6-halogen-9β10α-Δ<4,6>-steroiddiener af androstan- eller pregnanrækken. |
| DK324365AA DK123352B (da) | 1965-01-22 | 1965-06-25 | Analogifremgangsmåde til fremstilling af 6-halogensubstituerede 9β, 10α-steroider af androstanrækken. |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK324365AA DK123352B (da) | 1965-01-22 | 1965-06-25 | Analogifremgangsmåde til fremstilling af 6-halogensubstituerede 9β, 10α-steroider af androstanrækken. |
Country Status (14)
| Country | Link |
|---|---|
| US (2) | US3304314A (da) |
| AT (1) | AT261129B (da) |
| BE (2) | BE665762A (da) |
| BR (1) | BR6570589D0 (da) |
| CH (1) | CH464188A (da) |
| DE (2) | DE1518994A1 (da) |
| DK (2) | DK120337B (da) |
| ES (1) | ES314639A1 (da) |
| FI (1) | FI41743B (da) |
| FR (3) | FR4631M (da) |
| GB (1) | GB1087920A (da) |
| IL (2) | IL23629A (da) |
| NL (2) | NL6508148A (da) |
| SE (1) | SE331277B (da) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BE667121A (da) * | 1964-10-28 | |||
| IL23629A (en) * | 1965-01-22 | 1969-01-29 | Hoffmann La Roche | 9beta,10alpha-steroids and process for the manufacture thereof |
| GB1228801A (da) * | 1967-07-11 | 1971-04-21 | ||
| US3937700A (en) * | 1970-03-04 | 1976-02-10 | U.S. Philips Corporation | Novel 1,2-methylene-17α-acyloxy (or improved hydroxy)-9β, 10α-steroid compounds of the pregnane series, pharmaceutic preparations on the basis of the novel compounds and methods of producing said compounds and preparations |
| US4898694A (en) * | 1987-11-25 | 1990-02-06 | Schwartz Arthur G | 17-Hydroxy-steroids |
| US20070082876A1 (en) * | 2005-09-30 | 2007-04-12 | Solvay Pharmaceuticals Gmbh | Novel C18 modified retrosteroids as progesterone receptor modulator compounds |
| US20070212751A1 (en) * | 2006-01-18 | 2007-09-13 | Solvay Pharmaceuticals Gmbh | Microbial method for the 11beta hydroxylation of 9beta, 10alpha-steriods |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL252417A (da) * | 1959-06-08 | |||
| US3258473A (en) * | 1963-10-04 | 1966-06-28 | Syntex Corp | 17-dihaloacetate esters of 17alpha-hydroxy-21-desoxypregnane derivatives |
| IL23629A (en) * | 1965-01-22 | 1969-01-29 | Hoffmann La Roche | 9beta,10alpha-steroids and process for the manufacture thereof |
-
1965
- 1965-05-30 IL IL6523629A patent/IL23629A/xx unknown
- 1965-06-03 DE DE19651518994 patent/DE1518994A1/de active Pending
- 1965-06-16 FR FR20951A patent/FR4631M/fr not_active Expired
- 1965-06-22 BE BE665762D patent/BE665762A/xx unknown
- 1965-06-22 BR BR170589/65A patent/BR6570589D0/pt unknown
- 1965-06-23 CH CH876665A patent/CH464188A/de unknown
- 1965-06-23 GB GB26557/65A patent/GB1087920A/en not_active Expired
- 1965-06-23 FI FI1505/65A patent/FI41743B/fi active
- 1965-06-23 DK DK319165AA patent/DK120337B/da unknown
- 1965-06-23 IL IL6523785A patent/IL23785A/xx unknown
- 1965-06-23 SE SE08369/65A patent/SE331277B/xx unknown
- 1965-06-24 US US466818A patent/US3304314A/en not_active Expired - Lifetime
- 1965-06-24 DE DE19651543274 patent/DE1543274A1/de active Pending
- 1965-06-24 FR FR22045A patent/FR1446515A/fr not_active Expired
- 1965-06-24 US US466817A patent/US3423433A/en not_active Expired - Lifetime
- 1965-06-24 AT AT573665A patent/AT261129B/de active
- 1965-06-25 NL NL6508148A patent/NL6508148A/xx unknown
- 1965-06-25 ES ES0314639A patent/ES314639A1/es not_active Expired
- 1965-06-25 DK DK324365AA patent/DK123352B/da unknown
- 1965-06-25 NL NL6508179A patent/NL6508179A/xx unknown
- 1965-06-26 FR FR22465A patent/FR1439514A/fr not_active Expired
- 1965-06-28 BE BE666060A patent/BE666060A/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| DE1543274A1 (de) | 1969-07-24 |
| SE331277B (da) | 1970-12-21 |
| CH464188A (de) | 1968-10-31 |
| FR1446515A (fr) | 1966-07-22 |
| IL23629A (en) | 1969-01-29 |
| BE666060A (da) | 1965-12-28 |
| FR4631M (da) | 1966-11-28 |
| US3304314A (en) | 1967-02-14 |
| GB1087920A (en) | 1967-10-18 |
| AT261129B (de) | 1968-04-10 |
| FR1439514A (fr) | 1966-05-20 |
| BE665762A (da) | 1965-12-22 |
| ES314639A1 (es) | 1966-02-16 |
| NL6508148A (da) | 1966-06-27 |
| US3423433A (en) | 1969-01-21 |
| BR6570589D0 (pt) | 1973-08-02 |
| FI41743B (da) | 1969-10-31 |
| DE1518994A1 (de) | 1969-09-25 |
| NL6508179A (da) | 1965-12-27 |
| IL23785A (en) | 1969-09-25 |
| DK123352B (da) | 1972-06-12 |
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