DK114342B - Fremgangsmåde til fremstilling af 17α,21-dihydroxy-20-oxo-4,6-pregnadien-[3,2-c]pyrazol-forbindelser. - Google Patents

Fremgangsmåde til fremstilling af 17α,21-dihydroxy-20-oxo-4,6-pregnadien-[3,2-c]pyrazol-forbindelser.

Info

Publication number
DK114342B
DK114342B DK197762A DK197762A DK114342B DK 114342 B DK114342 B DK 114342B DK 197762 A DK197762 A DK 197762A DK 197762 A DK197762 A DK 197762A DK 114342 B DK114342 B DK 114342B
Authority
DK
Denmark
Prior art keywords
pregnadiene
dihydroxy
oxo
preparation
pyrazole compounds
Prior art date
Application number
DK197762A
Other languages
Danish (da)
English (en)
Inventor
M Tishler
N Steinberg
R Hirschmann
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US156478A external-priority patent/US3067194A/en
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of DK114342B publication Critical patent/DK114342B/da

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A61K31/573—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J75/00—Processes for the preparation of steroids in general

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
DK197762A 1961-05-01 1962-05-01 Fremgangsmåde til fremstilling af 17α,21-dihydroxy-20-oxo-4,6-pregnadien-[3,2-c]pyrazol-forbindelser. DK114342B (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10653961A 1961-05-01 1961-05-01
US156478A US3067194A (en) 1961-12-01 1961-12-01 4, 6-pregnadieno-[3, 2-c] pyrazoles and processes of preparing them

Publications (1)

Publication Number Publication Date
DK114342B true DK114342B (da) 1969-06-23

Family

ID=26803782

Family Applications (2)

Application Number Title Priority Date Filing Date
DK197762A DK114342B (da) 1961-05-01 1962-05-01 Fremgangsmåde til fremstilling af 17α,21-dihydroxy-20-oxo-4,6-pregnadien-[3,2-c]pyrazol-forbindelser.
DK557963A DK108168C (da) 1961-05-01 1962-05-01 Fremgangsmåde til fremstilling af 21-dihydrogenphosphatestere af 17 α,21-dihydroxy-20-oxo-4,6-pregnadien-(3,2-c)-pyrazol-forbindelser.

Family Applications After (1)

Application Number Title Priority Date Filing Date
DK557963A DK108168C (da) 1961-05-01 1962-05-01 Fremgangsmåde til fremstilling af 21-dihydrogenphosphatestere af 17 α,21-dihydroxy-20-oxo-4,6-pregnadien-(3,2-c)-pyrazol-forbindelser.

Country Status (7)

Country Link
BE (1) BE617105A (cs)
CH (1) CH423768A (cs)
DE (1) DE1468211B1 (cs)
DK (2) DK114342B (cs)
ES (1) ES277085A1 (cs)
NO (1) NO122591B (cs)
SE (1) SE309590B (cs)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1053502B (de) * 1956-01-26 1959-03-26 Syntex Sa Verfahren zur Herstellung von 2-Alkyl- und 2-Aralkylderivaten des A4-Pregnen-3, 20-dions, A4-Pregnen-17alpha-ol-3, 20-dions, A4-Pregnen-21-ol-3, 20-dions bzw. A4-Pregnen-17alpha, 21-diol-3, 20-dions
NL100550C (cs) * 1959-02-16

Also Published As

Publication number Publication date
NO122591B (cs) 1971-07-19
CH423768A (de) 1966-11-15
ES277085A1 (es) 1963-01-01
DK108168C (da) 1967-10-02
SE309590B (cs) 1969-03-31
DE1468211B1 (de) 1970-04-23
BE617105A (fr) 1962-10-30

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