DE69910983D1 - Synthese von chiralen beta-aminosäuren - Google Patents

Synthese von chiralen beta-aminosäuren

Info

Publication number
DE69910983D1
DE69910983D1 DE69910983T DE69910983T DE69910983D1 DE 69910983 D1 DE69910983 D1 DE 69910983D1 DE 69910983 T DE69910983 T DE 69910983T DE 69910983 T DE69910983 T DE 69910983T DE 69910983 D1 DE69910983 D1 DE 69910983D1
Authority
DE
Germany
Prior art keywords
synthesis
amino acids
beta amino
chiral beta
chiral
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE69910983T
Other languages
English (en)
Other versions
DE69910983T2 (de
Inventor
Pierre-Jean Colson
K Awasthi
R Nagarajan
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
GD Searle LLC
Original Assignee
GD Searle LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by GD Searle LLC filed Critical GD Searle LLC
Application granted granted Critical
Publication of DE69910983D1 publication Critical patent/DE69910983D1/de
Publication of DE69910983T2 publication Critical patent/DE69910983T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C227/30—Preparation of optical isomers
    • C07C227/32—Preparation of optical isomers by stereospecific synthesis

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DE69910983T 1998-03-04 1999-02-22 Synthese von chiralen beta-aminosäuren Expired - Fee Related DE69910983T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US7671098P 1998-03-04 1998-03-04
US76710P 1998-03-04
PCT/US1999/003280 WO1999044985A2 (en) 1998-03-04 1999-02-22 SYNTHESIS OF CHIRAL β-AMINO ACIDS

Publications (2)

Publication Number Publication Date
DE69910983D1 true DE69910983D1 (de) 2003-10-09
DE69910983T2 DE69910983T2 (de) 2004-07-15

Family

ID=22133735

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69910983T Expired - Fee Related DE69910983T2 (de) 1998-03-04 1999-02-22 Synthese von chiralen beta-aminosäuren

Country Status (15)

Country Link
US (1) US6414180B1 (de)
EP (1) EP1060159B1 (de)
JP (1) JP2002505317A (de)
AR (1) AR020056A1 (de)
AT (1) ATE248804T1 (de)
AU (1) AU2766999A (de)
CA (1) CA2322013A1 (de)
DE (1) DE69910983T2 (de)
DK (1) DK1060159T3 (de)
ES (1) ES2207181T3 (de)
MY (1) MY123317A (de)
PT (1) PT1060159E (de)
TW (1) TWI230706B (de)
WO (1) WO1999044985A2 (de)
ZA (1) ZA991105B (de)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6207854B1 (en) * 1999-12-15 2001-03-27 Eastman Chemical Company Preparation of 3-amino-3-cyclopropylpropanoate esters
US7071342B2 (en) * 2003-04-18 2006-07-04 Schering Corporation Synthesis of 2-hydroxy-N,N-dimethyl-3-[ [2-[1 (R)-(5-methyl-2-furanyl)propyl]amino]-3,4-dioxo-1-cyclobuten-1-yl]aminobenzamide
US20090263905A1 (en) * 2008-04-18 2009-10-22 Kim Scheuringer Detection test assembly for detecting the presence of a substance in a sample
US8716226B2 (en) 2012-07-18 2014-05-06 Saint Louis University 3,5 phenyl-substituted beta amino acid derivatives as integrin antagonists
JP6215324B2 (ja) 2012-07-18 2017-10-18 セントルイス ユニバーシティ インテグリンアンタゴニストとしてのβアミノ酸誘導体
CA3008023A1 (en) 2015-12-30 2017-07-06 Saint Louis University Meta-azacyclic amino benzoic acid derivatives as pan integrin antagonists

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3740439A (en) * 1968-06-24 1973-06-19 Ciba Geigy Corp Treating hypertension with beta-aminoalkane carboxylic acids
US3904681A (en) * 1971-03-30 1975-09-09 Ciba Geigy Corp Propionic acid
MX9801716A (es) * 1995-08-30 1998-05-31 Searle & Co Derivados de meta-guanidina, urea, tiourea o acido aminobenzoico azaciclico, como antagonistas de integrina.
DK0912495T3 (da) 1996-07-12 2002-05-21 Searle & Co Asymmetrisk syntese af chirale beta-aminosyrer

Also Published As

Publication number Publication date
ZA991105B (en) 2000-02-11
US6414180B1 (en) 2002-07-02
EP1060159B1 (de) 2003-09-03
ES2207181T3 (es) 2004-05-16
DE69910983T2 (de) 2004-07-15
CA2322013A1 (en) 1999-09-10
WO1999044985A2 (en) 1999-09-10
MY123317A (en) 2006-05-31
ATE248804T1 (de) 2003-09-15
AR020056A1 (es) 2002-04-10
TWI230706B (en) 2005-04-11
JP2002505317A (ja) 2002-02-19
DK1060159T3 (da) 2004-01-05
WO1999044985A3 (en) 1999-11-11
PT1060159E (pt) 2004-01-30
AU2766999A (en) 1999-09-20
EP1060159A2 (de) 2000-12-20

Similar Documents

Publication Publication Date Title
DE69924930D1 (de) Synthese von Oligonukleotiden
ATE196463T1 (de) Assymetrische synthese von (-) 6-chloro-4-
ID21981A (id) Inhibitor-inhibitor sintasis nitrik oksida
DE69916582D1 (de) Synthese von zsm-48
DE19581582T1 (de) Befestigungselement zum Anbringen von Gegenständen an Knochen
DE69505318D1 (de) Synthetische anregbare Aminosäuren
ID24458A (id) Modifikasi rheologi in-sito poliolefin
ATE198889T1 (de) Apolipoprotein-b syntheseinhibitoren
DK1533303T3 (da) Substituerede aminosalicylsyreamider (mellemprodukter)
ATE231507T1 (de) Synthese von azyklischen nukleosiden
NO20001728D0 (no) Fremgangsmåte for fremstilling av chirale forbindelser
ATE242750T1 (de) Synthese von kristallinen silicoaluminophosphaten
DE69801344D1 (de) Synthese von Bis(Phthalocyanylalumino)tetraphenyldisiloxanen
ATE230926T1 (de) Synergistische mischungen von ausgewählten aminosäuren
DE69722585D1 (de) Synthese von wellenformen
DE69800124D1 (de) Verfahren zur Reinigung von verzweigtkettigen Aminosäuren
DE69910983D1 (de) Synthese von chiralen beta-aminosäuren
ATE326443T1 (de) Verfahren zur stereoselektiven synthese zyklischer aminosäuren
FR2767824B1 (fr) Synthese d'acides carboxyalkylthiosucciniques
IT1295934B1 (it) Procedimento migliorato per la sintesi di alchilpoliglucosidi
NO20001777D0 (no) Fremgangsmåte for fremstilling av substituerte 4-fenyl-4- cyanocykloheksankarboksylsyrer
DE69624759D1 (de) Synthese von Difluormethan
NO20001896D0 (no) Fremgangsmõte for syntese av klorpurinmellomprodukter
ITTO930519A1 (it) Procedimento di sintesi di acidi cloroacetici.
BR9708718A (pt) Sínteses de aminas substituídas

Legal Events

Date Code Title Description
8364 No opposition during term of opposition
8339 Ceased/non-payment of the annual fee