DE3787586D1 - Alkylsubstituiertes benzoxazinorifamycinderivat, verfahren zu seiner herstellung und dieses enthaltendes antibakterielles mittel. - Google Patents

Alkylsubstituiertes benzoxazinorifamycinderivat, verfahren zu seiner herstellung und dieses enthaltendes antibakterielles mittel.

Info

Publication number
DE3787586D1
DE3787586D1 DE87110048T DE3787586T DE3787586D1 DE 3787586 D1 DE3787586 D1 DE 3787586D1 DE 87110048 T DE87110048 T DE 87110048T DE 3787586 T DE3787586 T DE 3787586T DE 3787586 D1 DE3787586 D1 DE 3787586D1
Authority
DE
Germany
Prior art keywords
benzoxazinorifamycine
derivative
substituted
alkyl
production
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE87110048T
Other languages
English (en)
Other versions
DE3787586T2 (de
Inventor
Fumihiko Kano
Takehiko Yamane Takehik Yamane
Katsuji Yamashita
Kazunori Hosoe
Kiyoshi Watanabe
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Kanegafuchi Chemical Industry Co Ltd
Original Assignee
Kanegafuchi Chemical Industry Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kanegafuchi Chemical Industry Co Ltd filed Critical Kanegafuchi Chemical Industry Co Ltd
Application granted granted Critical
Publication of DE3787586D1 publication Critical patent/DE3787586D1/de
Publication of DE3787586T2 publication Critical patent/DE3787586T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18—Bridged systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DE87110048T 1986-07-14 1987-07-11 Alkylsubstituiertes Benzoxazinorifamycinderivat, Verfahren zu seiner Herstellung und dieses enthaltendes antibakterielles Mittel. Expired - Fee Related DE3787586T2 (de)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP16512186 1986-07-14
JP24337686 1986-10-14
JP2943687 1987-02-10
JP62062213A JP2544375B2 (ja) 1986-07-14 1987-03-17 アルキル置換ベンゾキサジノリフアマイシン誘導体

Publications (2)

Publication Number Publication Date
DE3787586D1 true DE3787586D1 (de) 1993-11-04
DE3787586T2 DE3787586T2 (de) 1994-01-27

Family

ID=27459068

Family Applications (1)

Application Number Title Priority Date Filing Date
DE87110048T Expired - Fee Related DE3787586T2 (de) 1986-07-14 1987-07-11 Alkylsubstituiertes Benzoxazinorifamycinderivat, Verfahren zu seiner Herstellung und dieses enthaltendes antibakterielles Mittel.

Country Status (6)

Country Link
US (1) US4859661A (de)
EP (1) EP0253340B1 (de)
JP (1) JP2544375B2 (de)
CN (1) CN1018833B (de)
CA (1) CA1282780C (de)
DE (1) DE3787586T2 (de)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1293503C (en) * 1988-03-18 1991-12-24 Fumihiko Kanoo Substituted benzoxazinorifamycin derivative, process for preparing the same and antibacterial agent containing the same
CA1304363C (en) * 1988-11-01 1992-06-30 Takehiko Yamane 3'-hydroxybenzoxazinorifamycin derivative, process for preparing the same and antibacterial agent containing the same
DE69829905T2 (de) * 1997-02-28 2006-03-09 Kaneka Corp. Heilmittel für durch Helicobacter verursachte Krankheit
WO2004034961A2 (en) * 2001-09-06 2004-04-29 Activbiotics, Inc. Antimicrobial agents and uses thereof
CA2465846A1 (en) * 2001-11-21 2003-06-05 Activbiotics, Inc. Targeted therapeutics and uses thereof
WO2003051299A2 (en) * 2001-12-13 2003-06-26 Activbiotics, Inc. Sulfhydryl rifamycins and uses thereof
US20040077533A1 (en) * 2002-05-23 2004-04-22 Sayada Chalom B. Methods and compositions for treating bacterial infections and diseases associated therewith
US20030236265A1 (en) * 2002-05-23 2003-12-25 Sayada Chalom B. Methods of treating bacterial infections and diseases associated therewith
US20090149453A1 (en) * 2002-05-23 2009-06-11 Activbiotics Pharma Llc Methods and compositions for treating bacterial infections and diseases associated therewith
US20040126414A1 (en) * 2002-12-12 2004-07-01 Michaelis Arthur F. Methods and compositions for treating and preventing ear infections
US20040176404A1 (en) * 2002-12-12 2004-09-09 Sayada Chalom B. Methods and reagents for treating or preventing atherosclerosis and diseases associated therewith
CA2536378A1 (en) * 2003-08-22 2005-03-10 Activbiotics, Inc. Rifamycin analogs and uses thereof
US7820652B2 (en) * 2003-09-24 2010-10-26 Activbiotics Pharma, Llc Regimen for the administration of rifamycin-class antibiotics
WO2005058231A2 (en) * 2003-12-10 2005-06-30 Activbiotics, Inc. Rifamycin analogs and uses thereof
AU2004308399A1 (en) * 2003-12-23 2005-07-14 Activbiotics, Inc. Rifamycin analogs and uses thereof
US7202246B2 (en) * 2004-06-09 2007-04-10 Cumbre Pharmaceuticals Inc. Spiro-rifamycin derivatives targeting RNA polymerase
EP3004161B1 (de) 2013-05-31 2019-10-02 Genentech, Inc. Anti-zellwand-teichonsäureantikörper und konjugate
US9803002B2 (en) 2013-05-31 2017-10-31 Genentench, Inc. Anti-wall teichoic antibodies and conjugates
KR20160015227A (ko) 2013-05-31 2016-02-12 제넨테크, 인크. 항-세포벽 테이코산 항체 및 접합체
KR20170086536A (ko) 2014-12-03 2017-07-26 제넨테크, 인크. 항-스타필로코커스 아우레우스 항체 리파마이신 접합체 및 이의 용도
MX2017007231A (es) 2014-12-03 2017-11-08 Genentech Inc Conjugados de rifamicina y anticuerpos contra el staphylococcuss aureus y usos de estos.

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL130099C (de) * 1963-10-11
US4690919A (en) * 1984-01-04 1987-09-01 Kanegafuchi Kagaku Kogyo Kabushiki Kaisha Benzoxazinorifamycin derivative, process for preparing the same and antibacterial agent containing the same
JPS63183587A (ja) * 1985-02-05 1988-07-28 Kanegafuchi Chem Ind Co Ltd ベンゾキサジノリフアマイシン誘導体

Also Published As

Publication number Publication date
CN1018833B (zh) 1992-10-28
EP0253340A1 (de) 1988-01-20
CA1282780C (en) 1991-04-09
US4859661A (en) 1989-08-22
DE3787586T2 (de) 1994-01-27
EP0253340B1 (de) 1993-09-29
JP2544375B2 (ja) 1996-10-16
CN87104870A (zh) 1988-02-17
JPS646279A (en) 1989-01-10

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Legal Events

Date Code Title Description
8364 No opposition during term of opposition
8339 Ceased/non-payment of the annual fee