DE3436380A1 - Selective fungicidal agents based on a pyrimidine derivative - Google Patents

Selective fungicidal agents based on a pyrimidine derivative

Info

Publication number
DE3436380A1
DE3436380A1 DE19843436380 DE3436380A DE3436380A1 DE 3436380 A1 DE3436380 A1 DE 3436380A1 DE 19843436380 DE19843436380 DE 19843436380 DE 3436380 A DE3436380 A DE 3436380A DE 3436380 A1 DE3436380 A1 DE 3436380A1
Authority
DE
Germany
Prior art keywords
lt
gt
alkyl
represents
bcm
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
DE19843436380
Other languages
German (de)
Inventor
Michael Dr Schwamborn
Engelbert Dr Kuehle
Erich Dr Klauke
Wilhelm Dr Brandes
Wolfram Dr Koeller
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer AG
Original Assignee
Bayer AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer AG filed Critical Bayer AG
Priority to DE19843436380 priority Critical patent/DE3436380A1/en
Publication of DE3436380A1 publication Critical patent/DE3436380A1/en
Application status is Withdrawn legal-status Critical

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulfur or nitrogen atoms
    • C07D239/60Three or more oxygen or sulfur atoms
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/541,3-Diazines; Hydrogenated 1,3-diazines
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES, AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/10Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/18Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof containing a —O—CO—N< group, or a thio analogue thereof, directly attached to a heterocyclic or cycloaliphatic ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32One oxygen, sulfur or nitrogen atom
    • C07D239/42One nitrogen atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulfur or nitrogen atoms
    • C07D239/52Two oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulfur or nitrogen atoms
    • C07D239/56One oxygen atom and one sulfur atom
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulfur or nitrogen atoms
    • C07D239/58Two sulfur atoms

Abstract

The invention relates to the use of pyrimidine derivatives, some of which are known, of the formula (I) <IMAGE> in which R represents halogen, haloalkyl, alkyl, alkoxy, alkylthio or <IMAGE> in which R<4> represents hydrogen, alkyl or alkenyl, R<5> represents hydrogen, alkyl, haloalkyl, alkenyl, cycloalkyl, alkoxyalkyl, alkoxycarbonyl, alkoxycarbonylalkyl, aryl, or aralkyl; or R<4> and R<5>, together with the nitrogen atom to which they are attached, form a saturated, optionally substituted heterocycle which can contain further heteroatoms, R<1> represents alkyl, haloalkyl, alkoxy, alkylthio, halogen or phenylthio, R<2> represents alkoxy or halogen and R<3> represents hydrogen, alkyl, alkoxy, alkylthio, phenylthio or <IMAGE> where R<4> and R<5> have the abovementioned meaning, with the proviso that one of the radicals R or R<3> represents <IMAGE> for combating BCM-resistant fungal strains, in particular in combination with BCM, BCM analogues or BCM-forming compounds.
DE19843436380 1984-10-04 1984-10-04 Selective fungicidal agents based on a pyrimidine derivative Withdrawn DE3436380A1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
DE19843436380 DE3436380A1 (en) 1984-10-04 1984-10-04 Selective fungicidal agents based on a pyrimidine derivative

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19843436380 DE3436380A1 (en) 1984-10-04 1984-10-04 Selective fungicidal agents based on a pyrimidine derivative

Publications (1)

Publication Number Publication Date
DE3436380A1 true DE3436380A1 (en) 1986-04-10

Family

ID=6247063

Family Applications (1)

Application Number Title Priority Date Filing Date
DE19843436380 Withdrawn DE3436380A1 (en) 1984-10-04 1984-10-04 Selective fungicidal agents based on a pyrimidine derivative

Country Status (1)

Country Link
DE (1) DE3436380A1 (en)

Cited By (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0303348A1 (en) * 1987-07-09 1989-02-15 Pfizer Inc. 2-Amino-5-hydroxy-4-pyrimidones
US4910204A (en) * 1988-06-28 1990-03-20 Pfizer Inc. 2-amino-5-hydroxy-4-pyrimidones
US5521184A (en) * 1992-04-03 1996-05-28 Ciba-Geigy Corporation Pyrimidine derivatives and processes for the preparation thereof
US5612340A (en) * 1993-10-01 1997-03-18 Ciba-Geigy Corporation Pyrimidineamine derivatives and processes for the preparation thereof
WO1997018714A1 (en) * 1995-11-22 1997-05-29 The Minister Of Agriculture Fisheries & Food In Her Britannic Majesty's Government Of The United Kingdom Of Great Britain And Northern Ireland Alkylphosphines as pesticidal agents
WO1997048280A1 (en) * 1996-06-20 1997-12-24 Bayer Aktiengesellschaft Use of pyrrolopyrimidines to combat pests
US5728708A (en) * 1993-10-01 1998-03-17 Novartis Corporation Pharmacologically active pyridine derivatives and processes for the preparation thereof
GB2322553A (en) * 1995-11-22 1998-09-02 Mini Agriculture & Fisheries Alkylphosphines as pesticidal agents
US6048866A (en) * 1997-03-14 2000-04-11 Celltech Therapeutics, Limited Substituted 2-anilinopryimidines useful as protein kinase inhibitors
US6552029B1 (en) 1996-10-28 2003-04-22 Celltech R&D Limited 2-pyrimidineamine derivatives and processes for their preparation
US6579983B1 (en) 1999-06-18 2003-06-17 Celltech R&D Limited 5-cyano-2-aminopyrimidine derivatives
US6600037B1 (en) 1999-10-20 2003-07-29 Celltech R & D Limited 4,5-disubstituted-2-aminopyrimidines
WO2008092199A1 (en) * 2007-01-31 2008-08-07 Cytopia Research Pty Ltd Thiopyrimidine-based compounds and uses thereof
WO2011032656A1 (en) 2009-09-18 2011-03-24 Bayer Cropscience Ag 5-fluor-2-thio-substituted pyrimidine derivatives

Cited By (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0303348A1 (en) * 1987-07-09 1989-02-15 Pfizer Inc. 2-Amino-5-hydroxy-4-pyrimidones
US4910204A (en) * 1988-06-28 1990-03-20 Pfizer Inc. 2-amino-5-hydroxy-4-pyrimidones
US5521184A (en) * 1992-04-03 1996-05-28 Ciba-Geigy Corporation Pyrimidine derivatives and processes for the preparation thereof
US5728708A (en) * 1993-10-01 1998-03-17 Novartis Corporation Pharmacologically active pyridine derivatives and processes for the preparation thereof
US5612340A (en) * 1993-10-01 1997-03-18 Ciba-Geigy Corporation Pyrimidineamine derivatives and processes for the preparation thereof
WO1997018714A1 (en) * 1995-11-22 1997-05-29 The Minister Of Agriculture Fisheries & Food In Her Britannic Majesty's Government Of The United Kingdom Of Great Britain And Northern Ireland Alkylphosphines as pesticidal agents
US6096330A (en) * 1995-11-22 2000-08-01 The Secretary Of State For Minister Of Agriculture Fisheries & Food In Her Britannic Majesty's Government Of The United Kingdom Of Great Britain And Northern Ireland Alkylphosphines as pesticidal agents
GB2322553A (en) * 1995-11-22 1998-09-02 Mini Agriculture & Fisheries Alkylphosphines as pesticidal agents
GB2322553B (en) * 1995-11-22 2000-01-19 Mini Agriculture & Fisheries Pesticidal use of aliphatic phosphines
WO1997048280A1 (en) * 1996-06-20 1997-12-24 Bayer Aktiengesellschaft Use of pyrrolopyrimidines to combat pests
US6103726A (en) * 1996-06-20 2000-08-15 Bayer Aktiengesellschaft Use of pyrrolopyrimidines for controlling pests
US6552029B1 (en) 1996-10-28 2003-04-22 Celltech R&D Limited 2-pyrimidineamine derivatives and processes for their preparation
US6048866A (en) * 1997-03-14 2000-04-11 Celltech Therapeutics, Limited Substituted 2-anilinopryimidines useful as protein kinase inhibitors
US6337335B1 (en) 1997-03-14 2002-01-08 Celltech Therapeutics Limited Substituted 2-anilinopyrimidines useful as protein kinase inhibitors
US6579983B1 (en) 1999-06-18 2003-06-17 Celltech R&D Limited 5-cyano-2-aminopyrimidine derivatives
US6600037B1 (en) 1999-10-20 2003-07-29 Celltech R & D Limited 4,5-disubstituted-2-aminopyrimidines
WO2008092199A1 (en) * 2007-01-31 2008-08-07 Cytopia Research Pty Ltd Thiopyrimidine-based compounds and uses thereof
JP2010516788A (en) * 2007-01-31 2010-05-20 サイトピア・リサーチ・ピーティーワイ・リミテッド Thiopyrimidine-based compounds and uses thereof
US20100239631A1 (en) * 2007-01-31 2010-09-23 David Gerard Bourke Thiopyrimidine-based compounds and uses thereof
AU2008210266B2 (en) * 2007-01-31 2013-09-05 Ym Biosciences Australia Pty Ltd Thiopyrimidine-based compounds and uses thereof
US8846704B2 (en) * 2007-01-31 2014-09-30 YM Biosciences Austraila Pty Ltd Thiopyrimidine-based compounds and uses thereof
US9040549B2 (en) 2007-01-31 2015-05-26 Ym Biosciences Australia Pty Ltd. Thiopyrimidine-based compounds and uses thereof
WO2011032656A1 (en) 2009-09-18 2011-03-24 Bayer Cropscience Ag 5-fluor-2-thio-substituted pyrimidine derivatives

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